P1 Aspartate-Based Peptide .alpha.-((2,6-Dichlorobenzoyl)oxy)methyl Ketones as Potent Time-Dependent Inhibitors of Interleukin-1.beta.-Converting Enzyme
Dolle, Roland E, Hoyer, Denton, Prasad, C. V. C, Schmidt, Stanley J, Helaszek, Carla T, Miller, Robert E, Ator, Mark A
Published in Journal of medicinal chemistry (01.03.1994)
Published in Journal of medicinal chemistry (01.03.1994)
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Journal Article
Studies on the acid-catalyzed homonuclear steroidal diene isomerization
Dolle, Roland E, Schmidt, Stanley J, Eggleston, Drake, Kruse, Lawrence I
Published in Journal of organic chemistry (01.04.1988)
Published in Journal of organic chemistry (01.04.1988)
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Journal Article
Comprehensive Survey of Combinatorial Library Synthesis: 2005
Dolle, Roland E, Le Bourdonnec, Bertrand, Morales, Guillermo A, Moriarty, Kevin J, Salvino, Joseph M
Published in Journal of combinatorial chemistry (01.09.2006)
Published in Journal of combinatorial chemistry (01.09.2006)
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Journal Article
Pyridazinodiazepines as a High-Affinity, P2−P3 Peptidomimetic Class of Interleukin-1β-Converting Enzyme Inhibitor
Dolle, Roland E, Prasad, C. V. C, Prouty, Catherine P, Salvino, Joseph M, Awad, Mohamed M. A, Schmidt, Stanley J, Hoyer, Denton, Ross, Tina Morgan, Graybill, Todd L, Speier, Gary J, Uhl, Joanne, Helaszek, Carla T, Ator, Mark A
Published in Journal of medicinal chemistry (20.06.1997)
Published in Journal of medicinal chemistry (20.06.1997)
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Journal Article
Design of potent non-peptide competitive antagonists of the human bradykinin B2 receptor
Salvino, Joseph M, Seoane, Peter R, Douty, Brent D, Awad, Mohamad M. A, Dolle, Roland E, Houck, Wayne T, Faunce, David M, Sawutz, David G
Published in Journal of medicinal chemistry (01.08.1993)
Published in Journal of medicinal chemistry (01.08.1993)
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Journal Article
First Examples of Peptidomimetic Inhibitors of Interleukin-1β Converting Enzyme
Dolle, Roland E, Prouty, Catherine P, Prasad, C. V. C, Cook, Ewell, Saha, Ashis, Ross, Tina Morgan, Salvino, Joseph M, Helaszek, Carla T, Ator, Mark A
Published in Journal of medicinal chemistry (21.06.1996)
Published in Journal of medicinal chemistry (21.06.1996)
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Journal Article
SPIROCYCLIC HETEROCYCLIC DERIVATIVES AND METHODS OF THEIR USE
LE BOURDONNEC BERTRAND, ZHOU JEAN Q, LEISTER LARA K, DOLLE ROLAND E, AJELLO CHRISTOPHER W, CHU GUO HUA, GU MINGHUA, TUTHILL PAUL ANSON
Year of Publication 06.02.2014
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Year of Publication 06.02.2014
Patent
Application of the intramolecular azomethine imine cycloaddition to the construction of a novel, orthogonally protected spirodiamino acid scaffold
Dolle, Roland E, Barden, Michael C, Brennan, Paul E, Ahmed, Gulzar, Tran, Vinh, Ho, Douglas M
Published in Tetrahedron letters (09.04.1999)
Published in Tetrahedron letters (09.04.1999)
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Journal Article
ATP-Citrate Lyase as a Target for Hypolipidemic Intervention. 2. Synthesis and Evaluation of (3R,5S)-ω-Substituted-3-carboxy-3,5-dihydroxyalkanoic Acids and Their γ-Lactone Prodrugs as Inhibitors of the Enzyme in Vitro and in Vivo
Gribble, Andrew D, Ife, Robert J, Shaw, Antony, McNair, David, Novelli, Christine E, Bakewell, Susan, Shah, Virendra P, Dolle, Roland E, Groot, Pieter H, Pearce, Nigel, Yates, John, Tew, David, Boyd, Helen, Ashman, Stephen, Eggleston, Drake S, Haltiwanger, R. Curtis, Okafo, George
Published in Journal of medicinal chemistry (10.09.1998)
Published in Journal of medicinal chemistry (10.09.1998)
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Journal Article
ATP-Citrate Lyase as a Target for Hypolipidemic Intervention. Design and Synthesis of 2-Substituted Butanedioic Acids as Novel, Potent Inhibitors of the Enzyme
Gribble, Andrew D, Dolle, Roland E, Shaw, Antony, McNair, David, Novelli, Riccardo, Novelli, Christine E, Slingsby, Brian P, Shah, Virendra P, Tew, David, Saxty, Barbara A, Allen, Mark, Groot, Pieter H, Pearce, Nigel, Yates, John
Published in Journal of medicinal chemistry (30.08.1996)
Published in Journal of medicinal chemistry (30.08.1996)
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Journal Article
Discovery of lndazole Derivatives as a Novel Class of Bacterial Gyrase B Inhibitors
Zhang, Jing, Yang, Qingyi, Romero, Jan Antoinette C., Cross, Jason, Wang, Bin, Poutsiaka, Katherine M., Epie, Felix, Bevan, Douglas, Wu, Yuchuan, Moy, Terence, Daniel, Anu, Chamberlain, Brian, Carter, Nicole, Shotwell, Joseph, Arya, Anu, Kumar, Vipul, Silverman, Jared, Kien Nguyen, Metcalf, Chester A., Ryan, Dominic, Lippa, Blaise, Dolle, Roland E.
Published in ACS medicinal chemistry letters (01.10.2015)
Published in ACS medicinal chemistry letters (01.10.2015)
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