Search Results - "DOLLE, Roland E." :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery of a series of aminopiperidines as novel iNOS inhibitors

Discovery of a series of aminopiperidines as novel iNOS inhibitors

by Bourdonnec, Bertrand Le, Leister, Lara K., Ajello, Christopher A., Cassel, Joel A., Seida, Pamela R., O’Hare, Heather, Gu, Minghua, Chu, Guo-Hua, Tuthill, Paul A., DeHaven, Robert N., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry (2008)

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Journal Article

Further studies of tyrosine surrogates in opioid receptor peptide ligands

Further studies of tyrosine surrogates in opioid receptor peptide ligands

by Dolle, Roland E., Michaut, Mathieu, Martinez-Teipel, Blanca, Belanger, Serge, Graczyk, Thomas M., DeHaven, Robert N.
Published in Bioorganic & medicinal chemistry letters (01.05.2007)

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Journal Article

Sulfonamido-aryl ethers as bradykinin B1 receptor antagonists

Sulfonamido-aryl ethers as bradykinin B1 receptor antagonists

by Cole, Andrew G., Metzger, Axel, Brescia, Marc-Raleigh, Qin, Lan-Ying, Appell, Kenneth C., Brain, Christopher T., Hallett, Allan, Ganju, Pam, Denholm, Alastair A., Wareing, James R., Ritchie, Timothy J., Drake, Gillian M., Bevan, Stuart J., MacGloinn, Aisling, McBryde, Andrew, Patel, Viral, Oakley, Paul J., Nunez, Ximena, Gstach, Hubert, Schneider, Peter, Baldwin, John J., Dolle, Roland E., McDonald, Edward, Henderson, Ian
Published in Bioorganic & medicinal chemistry letters (2009)

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Journal Article

Novel trans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidines as μ opioid receptor antagonists with improved opioid receptor selectivity profiles

Novel trans-3,4-dimethyl-4-(3-hydroxyphenyl)piperidines as μ opioid receptor antagonists with improved opioid receptor selectivity profiles

by Le Bourdonnec, Bertrand, Barker, William M., Belanger, Serge, Wiant, Daniel D., Conway-James, Nathalie C., Cassel, Joel A., O’Neill, Timothy J., Little, Patrick J., DeHaven, Robert N., DeHaven-Hudkins, Diane L., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry (15.03.2008)

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Journal Article

Comprehensive survey of chemical libraries yielding enzyme inhibitors, receptor agonists and antagonists, and other biologically active agents: 1992 through 1997

Comprehensive survey of chemical libraries yielding enzyme inhibitors, receptor agonists and antagonists, and other biologically active agents: 1992 through 1997

by Dolle, R E
Published in Molecular diversity (1997)

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Journal Article

Small molecule biaryl FSH receptor agonists. Part 1: Lead discovery via encoded combinatorial synthesis

Small molecule biaryl FSH receptor agonists. Part 1: Lead discovery via encoded combinatorial synthesis

by Guo, Tao, Adang, Anton E.P., Dolle, Roland E., Dong, Guizhen, Fitzpatrick, Dan, Geng, Peng, Ho, Koc-Kan, Kultgen, Steven G., Liu, Ruiyan, McDonald, Edward, McGuinness, Brian F., Saionz, Kurt W., Valenzano, Kenneth J., van Straten, Nicole C.R., Xie, Dan, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (05.04.2004)

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Journal Article

(4-Carboxamido)phenylalanine is a surrogate for tyrosine in opioid receptor peptide ligands

(4-Carboxamido)phenylalanine is a surrogate for tyrosine in opioid receptor peptide ligands

by Dolle, Roland E., Machaut, Mathieu, Martinez-Teipel, Blanca, Belanger, Serge, Cassel, Joel A., Stabley, Gabriel J., Graczyk, Thomas M., DeHaven, Robert N.
Published in Bioorganic & medicinal chemistry letters (05.07.2004)

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Journal Article

Enantiospecific synthesis of (-)-tabtoxinine .beta.-lactam

Enantiospecific synthesis of (-)-tabtoxinine .beta.-lactam

by Dolle, Roland E, Li, Chun Sing, Novelli, Riccardo, Kruse, Lawrence I, Eggleston, Drake
Published in Journal of organic chemistry (01.01.1992)

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Journal Article

Solid-phase synthesis of α-hydroxy phosphonates and hydroxystatine amides. Transition-state isosteres derived from resin-bound amino acid aldehydes

Solid-phase synthesis of α-hydroxy phosphonates and hydroxystatine amides. Transition-state isosteres derived from resin-bound amino acid aldehydes

by Dolle, Roland E, Herpin, Timothy F, Shimshock, Yvonne Class
Published in Tetrahedron letters (04.03.2001)

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Journal Article

trans-3,4-Dimethyl-4-(3-carboxamidophenyl)piperidines: A novel class of μ-selective opioid antagonists

trans-3,4-Dimethyl-4-(3-carboxamidophenyl)piperidines: A novel class of μ-selective opioid antagonists

by LE BOURDONNEC, Bertrand, BELANGER, Serge, CASSEL, Joel A, STABLEY, Gabriel J, DEHAVEN, Robert N, DOLLE, Roland E
Published in Bioorganic & medicinal chemistry letters (15.12.2003)

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Journal Article

Arylacetamide κ opioid receptor agonists with reduced cytochrome P450 2D6 inhibitory activity

Arylacetamide κ opioid receptor agonists with reduced cytochrome P450 2D6 inhibitory activity

by Le Bourdonnec, Bertrand, Ajello, Christopher W., Seida, Pamela R., Susnow, Roberta G., Cassel, Joel A., Belanger, Serge, Stabley, Gabriel J., DeHaven, Robert N., DeHaven-Hudkins, Diane L., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (16.05.2005)

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Journal Article

Azepinone as a conformational constraint in the design of κ-opioid receptor agonists

Azepinone as a conformational constraint in the design of κ-opioid receptor agonists

by TUTHILL, Paul A, SEIDA, Pamela R, DOLLE, Roland E, BARKER, William, CASSEL, Joel A, BELANGER, Serge, DEHAVEN, Robert N, KOBLISH, Michael, GOTTSHALL, Susan L, LITTLE, Patrick J, DEHAVEN-HUDKINS, Diane L
Published in Bioorganic & medicinal chemistry letters (15.11.2004)

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Journal Article

The copper sites of dopamine .beta.-hydroxylase: an x-ray absorption spectroscopic study

The copper sites of dopamine .beta.-hydroxylase: an x-ray absorption spectroscopic study

by Scott, Robert A, Sullivan, Richard J, DeWolf, Walter E, Dolle, Roland E, Kruse, Lawrence I
Published in Biochemistry (Easton) (01.07.1988)

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Journal Article

Discovery of 6-Phenylhexanamide Derivatives as Potent Stereoselective Mitofusin Activators for the Treatment of Mitochondria! Diseases

Discovery of 6-Phenylhexanamide Derivatives as Potent Stereoselective Mitofusin Activators for the Treatment of Mitochondria! Diseases

by Dang, Xiawei, Zhang, Lihong, Franco, Antonietta, Li, Jiajia, Rocha, Agostinho G., Devanathan, Sriram, Dolle, Roland E., Bernstein, Peter R., Dorn, Gerald W.
Published in Journal of medicinal chemistry (09.07.2020)

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Journal Article

Inactivation of dopamine .beta.-hydroxylase by p-cresol: isolation and characterization of covalently modified active site peptides

Inactivation of dopamine .beta.-hydroxylase by p-cresol: isolation and characterization of covalently modified active site peptides

by DeWolf, Walter E, Carr, Steven A, Varrichio, Angela, Goodhart, Paula J, Mentzer, Mary A, Roberts, Gerald D, Southan, Christopher, Dolle, Roland E, Kruse, Lawrence I
Published in Biochemistry (Easton) (01.12.1988)

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Journal Article

The development and application of tetrafluorophenol-activated resins for rapid amine derivatization

The development and application of tetrafluorophenol-activated resins for rapid amine derivatization

by Salvino, Joseph M, Dolle, Roland E
Published in Methods in enzymology (2003)

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Journal Article

Synthesis and structure–activity relationships of a new series of 2α-substituted trans-4,5-dimethyl-4-(3-hydroxyphenyl)piperidine as μ-selective opioid antagonists

Synthesis and structure–activity relationships of a new series of 2α-substituted trans-4,5-dimethyl-4-(3-hydroxyphenyl)piperidine as μ-selective opioid antagonists

by Le Bourdonnec, Bertrand, Goodman, Allan J., Michaut, Mathieu, Ye, Hai-Fen, Graczyk, Thomas M., Belanger, Serge, DeHaven, Robert N., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (15.02.2006)

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Journal Article

Novel phenylamino acetamide derivatives as potent and selective κ opioid receptor agonists

Novel phenylamino acetamide derivatives as potent and selective κ opioid receptor agonists

by Chu, Guo-Hua, Gu, Minghua, Cassel, Joel A., Belanger, Serge, Stabley, Gabriel. J., DeHaven, Robert N., Conway-James, Nathalie, Koblish, Mike, Little, Patrick J., DeHaven-Hudkins, Diane L., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (01.02.2006)

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Journal Article

Design and Synthesis of Imidazopyrimidine Derivatives as Potent iNOS Dimerization Inhibitors

Design and Synthesis of Imidazopyrimidine Derivatives as Potent iNOS Dimerization Inhibitors

by Chu, Guo-Hua, Le Bourdonnec, Bertrand, Gu, Minghua, Ajello, Christopher W, Leister, Lara K, Sellitto, Ian, Cassel, Joel A, Tuthill, Paul A, O' Hare, Heather, Dehaven, Robert N, Dolle, Roland E
Published in The open medicinal chemistry journal (18.11.2009)

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Journal Article

(S)-2-BENZYL-3-((3R,4R)-4-(3-CARBAMOYLPHENYL)-3,4-DIMETHYLPIPERIDINYL)PROPANOIC ACID AND SALT THEROF AS ANTAGONISTS OF THE OPIOID RECEPTORS

(S)-2-BENZYL-3-((3R,4R)-4-(3-CARBAMOYLPHENYL)-3,4-DIMETHYLPIPERIDINYL)PROPANOIC ACID AND SALT THEROF AS ANTAGONISTS OF THE OPIOID RECEPTORS

by LE BOURDONNEC BERTRAND, DOLLE ROLAND E
Year of Publication 06.02.2014

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