The development of highly potent and selective small molecule correctors of Z alpha 1-antitrypsin misfolding
Liddle, John, Pearce, Andrew C., Arico-Muendel, Christopher, Belyanskaya, Svetlana, Brewster, Andrew, Brown, Murray, Chung, Chun-wa, Denis, Alexis, Dodic, Nerina, Dossang, Anthony, Eddershaw, Peter, Klimaszewska, Diana, Haq, Imran, Holmes, Duncan S., Jagger, Alistair, Jakhria, Toral, Jigorel, Emilie, Lind, Ken, Messer, Jeff, Neu, Margaret, Olszewski, Allison, Ronzoni, Riccardo, Rowedder, James, Rudiger, Martin, Skinner, Steve, Smith, Kathrine J., Trottet, Lionel, Uings, Iain, Zhu, Zhengrong, Irving, James A., Lomas, David A.
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
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Development of a small molecule that corrects misfolding and increases secretion of Z α1‐antitrypsin
Lomas, David A, Irving, James A, Arico‐Muendel, Christopher, Belyanskaya, Svetlana, Brewster, Andrew, Brown, Murray, Chung, Chun‐wa, Dave, Hitesh, Denis, Alexis, Dodic, Nerina, Dossang, Anthony, Eddershaw, Peter, Klimaszewska, Diana, Haq, Imran, Holmes, Duncan S, Hutchinson, Jonathan P, Jagger, Alistair M, Jakhria, Toral, Jigorel, Emilie, Liddle, John, Lind, Ken, Marciniak, Stefan J, Messer, Jeff, Neu, Margaret, Olszewski, Allison, Ordonez, Adriana, Ronzoni, Riccardo, Rowedder, James, Rüdiger, Martin, Skinner, Steve, Smith, Kathrine J, Terry, Rebecca, Trottet, Lionel, Uings, Iain, Wilson, Steve, Zhu, Zhengrong, Pearce, Andrew C
Published in EMBO molecular medicine (05.03.2021)
Published in EMBO molecular medicine (05.03.2021)
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Journal Article
The development of highly potent and selective small molecule correctors of Z α1-antitrypsin misfolding
Liddle, John, Pearce, Andrew C., Arico-Muendel, Christopher, Belyanskaya, Svetlana, Brewster, Andrew, Brown, Murray, Chung, Chun-wa, Denis, Alexis, Dodic, Nerina, Dossang, Anthony, Eddershaw, Peter, Klimaszewska, Diana, Haq, Imran, Holmes, Duncan S., Jagger, Alistair, Jakhria, Toral, Jigorel, Emilie, Lind, Ken, Messer, Jeff, Neu, Margaret, Olszewski, Allison, Ronzoni, Riccardo, Rowedder, James, Rüdiger, Martin, Skinner, Steve, Smith, Kathrine J., Trottet, Lionel, Uings, Iain, Zhu, Zhengrong, Irving, James A., Lomas, David A.
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
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거대고리 RIP2 키나제 억제제
DENIS ALEXIS, DAOUBI KHAMLICHI MOURAD, BENDERITTER PASCAL ANDRE RENE, TAP AURELIEN, DODIC NERINA, LAMOTTE YANN, BRUSQ JEAN MARIE
Year of Publication 09.01.2023
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Year of Publication 09.01.2023
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Structurally Diverse Mitochondrial Branched Chain Aminotransferase (BCATm) Leads with Varying Binding Modes Identified by Fragment Screening
Borthwick, Jennifer A, Ancellin, Nicolas, Bertrand, Sophie M, Bingham, Ryan P, Carter, Paul S, Chung, Chun-wa, Churcher, Ian, Dodic, Nerina, Fournier, Charlène, Francis, Peter L, Hobbs, Andrew, Jamieson, Craig, Pickett, Stephen D, Smith, Sarah E, Somers, Donald O’N, Spitzfaden, Claus, Suckling, Colin J, Young, Robert J
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Published in Journal of medicinal chemistry (24.03.2016)
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The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits
Bertrand, Sophie M, Ancellin, Nicolas, Beaufils, Benjamin, Bingham, Ryan P, Borthwick, Jennifer A, Boullay, Anne-Bénédicte, Boursier, Eric, Carter, Paul S, Chung, Chun-wa, Churcher, Ian, Dodic, Nerina, Fouchet, Marie-Hélène, Fournier, Charlène, Francis, Peter L, Gummer, Laura A, Herry, Kenny, Hobbs, Andrew, Hobbs, Clare I, Homes, Paul, Jamieson, Craig, Nicodeme, Edwige, Pickett, Stephen D, Reid, Iain H, Simpson, Graham L, Sloan, Lisa A, Smith, Sarah E, Somers, Donald O’N, Spitzfaden, Claus, Suckling, Colin J, Valko, Klara, Washio, Yoshiaki, Young, Robert J
Published in Journal of medicinal chemistry (24.09.2015)
Published in Journal of medicinal chemistry (24.09.2015)
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Development of a small molecule that corrects misfolding and increases secretion of Z α 1 -antitrypsin
Lomas, David A, Irving, James A, Arico-Muendel, Christopher, Belyanskaya, Svetlana, Brewster, Andrew, Brown, Murray, Chung, Chun-Wa, Dave, Hitesh, Denis, Alexis, Dodic, Nerina, Dossang, Anthony, Eddershaw, Peter, Klimaszewska, Diana, Haq, Imran, Holmes, Duncan S, Hutchinson, Jonathan P, Jagger, Alistair M, Jakhria, Toral, Jigorel, Emilie, Liddle, John, Lind, Ken, Marciniak, Stefan J, Messer, Jeff, Neu, Margaret, Olszewski, Allison, Ordonez, Adriana, Ronzoni, Riccardo, Rowedder, James, Rüdiger, Martin, Skinner, Steve, Smith, Kathrine J, Terry, Rebecca, Trottet, Lionel, Uings, Iain, Wilson, Steve, Zhu, Zhengrong, Pearce, Andrew C
Published in EMBO molecular medicine (05.03.2021)
Published in EMBO molecular medicine (05.03.2021)
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Abstract 1398: Structure-based design of small macrocyclic CDK9 degraders as chemical biology tools and beyond
Dodic, Nerina, Ancellin, Nicolas, Bordessoules, Morgane, Bouillot, Anne, Butin, Nathan, Charrier, Cedric, Fouchet, Marie-Helene, Laroze, Alain, Luzy, Anne-Pascale, Moquette, Alexandre, Pilot, Julia, Serin, Guillaume, Mirjolet, Jean-François, Viviani, Fabrice, Parsy, Christophe
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Design and evaluation of a novel series of 2,3-oxidosqualene cyclase inhibitors with low systemic exposure, relationship between pharmacokinetic properties and ocular toxicity
Fouchet, Marie-Hélène, Donche, Frédéric, Martin, Christelle, Bouillot, Anne, Junot, Christophe, Boullay, Anne-Bénédicte, Potvain, Florent, Magny, Sylvie Demaria, Coste, Hervé, Walker, Max, Issandou, Marc, Dodic, Nérina
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
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Discovery and Optimization of Potent, Selective, and in Vivo Efficacious 2‑Aryl Benzimidazole BCATm Inhibitors
Deng, Hongfeng, Zhou, Jingye, Sundersingh, Flora, Messer, Jeffrey A, Somers, Donald O, Ajakane, Myriam, Arico-Muendel, Christopher C, Beljean, Arthur, Belyanskaya, Svetlana L, Bingham, Ryan, Blazensky, Emily, Boullay, Anne-Benedicte, Boursier, Eric, Chai, Jing, Carter, Paul, Chung, Chun-Wa, Daugan, Alain, Ding, Yun, Herry, Kenny, Hobbs, Clare, Humphries, Eric, Kollmann, Christopher, Nguyen, Van Loc, Nicodeme, Edwige, Smith, Sarah E, Dodic, Nerina, Ancellin, Nicolas
Published in ACS medicinal chemistry letters (14.04.2016)
Published in ACS medicinal chemistry letters (14.04.2016)
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Comparison of soluble guanylate cyclase stimulators and activators in models of cardiovascular disease associated with oxidative stress
Costell, Melissa H, Ancellin, Nicolas, Bernard, Roberta E, Zhao, Shufang, Upson, John J, Morgan, Lisa A, Maniscalco, Kristeen, Olzinski, Alan R, Ballard, Victoria L T, Herry, Kenny, Grondin, Pascal, Dodic, Nerina, Mirguet, Olivier, Bouillot, Anne, Gellibert, Francoise, Coatney, Robert W, Lepore, John J, Jucker, Beat M, Jolivette, Larry J, Willette, Robert N, Schnackenberg, Christine G, Behm, David J
Published in Frontiers in pharmacology (01.01.2012)
Published in Frontiers in pharmacology (01.01.2012)
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NOVEL SOLUBLE GUANYLATE CYCLASE ACTIVATORS AND THEIR USE
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Year of Publication 05.03.2024
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Year of Publication 27.10.2022
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