The Process Development of Ravuconazole: An Efficient Multikilogram Scale Preparation of an Antifungal Agent
Pesti, Jaan, Chen, Chien-Kuang, Spangler, Lori, DelMonte, Albert J, Benoit, Serge, Berglund, Derek, Bien, Jeffrey, Brodfuehrer, Paul, Chan, Yeung, Corbett, Elisabeth, Costello, Carrie, DeMena, Paul, Discordia, Robert P, Doubleday, Wendel, Gao, Zhinong, Gingras, Stephane, Grosso, John, Haas, Oscar, Kacsur, David, Lai, Chiajen, Leung, Simon, Miller, Melanie, Muslehiddinoglu, Jale, Nguyen, Nina, Qiu, Jun, Olzog, Martina, Reiff, Emily, Thoraval, Dominique, Totleben, Michael, Vanyo, Dale, Vemishetti, Purushotham, Wasylak, John, Wei, Chenkou
Published in Organic process research & development (17.07.2009)
Published in Organic process research & development (17.07.2009)
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Amination of Heterocyclic Compounds with O-Benzoylhydroxylamine Derivatives
Parlanti, Luca, Discordia, Robert P, Hynes, John, Miller, Michael M, O'Grady, Harold R, Shi, Zhongping
Published in Organic letters (13.09.2007)
Published in Organic letters (13.09.2007)
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A tellurium transposition route to allylic alcohols: overcoming some limitations of the Sharpless-Katsuki asymmetric epoxidation
Dittmer, Donald C, Discordia, Robert P, Zhang, Yanzhi, Murphy, Christopher K, Kumar, Archana, Pepito, Aurora S, Wang, Yuesheng
Published in Journal of organic chemistry (1993)
Published in Journal of organic chemistry (1993)
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Practical synthesis of the rebeccamycin aglycone and related analogs by oxidative cyclization of bisindolylmaleimides with a Wacker-type catalytic system
Wang, Jianji, Rosingana, Miguel, Watson, Daniel J, Dowdy, Eric D, Discordia, Robert P, Soundarajan, Nachimuthu, Li, Wen-Sen
Published in Tetrahedron letters (17.12.2001)
Published in Tetrahedron letters (17.12.2001)
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Journal Article
Preparation and pharmacokinetics of 11C labeled stavudine (d4T)
Livni, Eli, Berker, Mark, Hillier, Shawn, Waller, Stephen C, Ogan, Marc D, Discordia, Robert P, Rienhart, J.Kent, Rubin, Robert H, Fischman, Alan J
Published in Nuclear medicine and biology (01.07.2004)
Published in Nuclear medicine and biology (01.07.2004)
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Concomitant Epoxide Deoxygenation and Deacetylation of Glycidyl Acetates Induced by Telluride Ion
Dittmer, Donald C, Zhang, Yanzhi, Discordia, Robert P
Published in Journal of organic chemistry (01.03.1994)
Published in Journal of organic chemistry (01.03.1994)
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A mild and efficient synthesis of 4-aryl-quinolin-2(1 H)-ones via a tandem amidation/Knoevenagel condensation of 2-amino-benzophenones with esters or lactones
Wang, Jianji, Discordia, Robert P., Crispino, Gerard A., Li, Jun, Grosso, John A., Polniaszek, Richard, Truc, Vu C.
Published in Tetrahedron letters (26.05.2003)
Published in Tetrahedron letters (26.05.2003)
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Efficient Synthesis of the Anticancer Drug Etoposide 4‘-Phosphate: Use of Benzylic Ether-Protecting Groups on the Carbohydrate Segment 1
Silverberg, Lee J., Dillon, John L., Vemishetti, Purushotham, Sleezer, Paul D., Discordia, Robert P., Hartung, Kerry B., Gao, Qi
Published in Organic process research & development (01.01.2000)
Published in Organic process research & development (01.01.2000)
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Synthesis of a radiolabeled enniatin cyclodepsipeptide [3H-methyl]JES 1798
Pleiss, U., Turberg, A., Harder, A., Londershausen, M., Jeschke, P., Boheim, G.
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.1996)
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.1996)
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PROCESS FOR THE PREPARATION OF Y(1R), 2S -2-AMINOPROPIONIC ACID 2-Y4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLOY2,1-f Y1,2,4 TRIAZIN-6-YLOXY -1-METHYLETHYL ESTER
LEAHY DAVID K, LOBBEN PAUL C, THORNTON JOHN E, MUSLEHIDDINOGLU JALE, HAMEDI MOURAD, XU ZHONGMIN, DISCORDIA ROBERT P, LAI CHIAJEN, CRISPINO GERARD A, PESTI JAAN A, SPANGLER LORI ANN, LAPORTE THOMAS L
Year of Publication 28.06.2013
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Year of Publication 28.06.2013
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PROCESS FOR THE PREPARATION OF Ý(1R), 2S¨-2-AMINOPROPIONIC ACID 2-Ý4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLOÝ2,1-f¨Ý1,2,4¨TRIAZIN-6-YLOXY¨-1-METHYLETHYL ESTER
LAPORTE, THOMAS L, LEAHY, DAVID K, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, LOBBEN, PAUL C, DISCORDIA, ROBERT P, PESTI, JAAN A, HAMEDI, MOURAD, THORNTON, JOHN E, XU, ZHONGMIN, SPANGLER, LORI ANN
Year of Publication 30.04.2013
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Year of Publication 30.04.2013
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PROCESS FOR THE PREPARATION OF [(1R), 2S]-2-AMINOPROPIONIC ACID 2-[4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLO]2,1-f-[1,2,4-TRIAZIN-6-YLOXY]-1-METHYLETHYL ESTER
LAPORTE, THOMAS L, LEAHY, DAVID K, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, LOBBEN, PAUL C, DISCORDIA, ROBERT P, PESTI, JAAN A, HAMEDI, MOURAD, THORNTON, JOHN E, XU, ZHONGMIN, SPANGLER, LORI ANN
Year of Publication 31.03.2013
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Year of Publication 31.03.2013
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PROCESS FOR THE PREPARATION OF Ý(1R), 2S¨-2-AMINOPROPIONIC ACID 2-Ý4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-5-METHYLPYRROLOÝ2,1-f¨Ý1,2,4¨TRIAZIN-6-YLOXY¨-1-METHYLETHYL ESTER
LAPORTE, THOMAS L, LEAHY, DAVID K, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, LOBBEN, PAUL C, DISCORDIA, ROBERT P, PESTI, JAAN A, HAMEDI, MOURAD, THORNTON, JOHN E, XU, ZHONGMIN, SPANGLER, LORI ANN
Year of Publication 05.12.2012
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Year of Publication 05.12.2012
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Process for the preparation of [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester
LEAHY, DAVID K, LAPORTE, THOMAS L, MUSLEHIDDINOGLU, JALE, LAI, CHIAJEN, CRISPINO, GERARD A, DISCORDIA, ROBERT P, LOBBEN, PAUL C, PESTI, JAAN A, HAMEDI, MOURAD, XU, ZHONGMIN, THORNTON, JOHN E, SPANGLER, LORI ANN
Year of Publication 12.04.2012
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Year of Publication 12.04.2012
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