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Inhibitors of Cholesterol Biosynthesis. 2. Hypocholesterolemic and Antioxidant Activities of Benzopyran and Tetrahydronaphthalene Analogs of the Tocotrienols
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Quinazoline derivatives as MC-I inhibitors: Evaluation of myocardial uptake using Positron Emission Tomography in rat and non-human primate
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Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Lead Pig for Use with Screw Cap Vials
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[18F](R)-5-chloro-1-(1-cyclopropyl-2-methoxyethyl)-3-(4-(2-fluoroethoxy)-2,5-dimethyl phenylamino)pyrazin-2(1H)-one: Introduction of N3-phenylpyrazinones as potential CRF-R1 PET imaging agents
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Published in Bioorganic & medicinal chemistry letters (01.11.2012)
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In vitro and in vivo metabolism of a gamma-secretase inhibitor BMS-299897 and generation of active metabolites in milligram quantities with a microbial bioreactor
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Published in Current drug metabolism (01.12.2006)
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Identification of a Binding Site on Hsc70 for the Immunosuppressant 15-Deoxyspergualin
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pH-Dependent Changes in Photoaffinity Labeling Patterns of the H1 Influenza Virus Hemagglutinin by Using an Inhibitor of Viral Fusion
Cianci, C, Yu, K L, Dischino, D D, Harte, W, Deshpande, M, Luo, G, Colonno, R J, Meanwell, N A, Krystal, M
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Published in Journal of labelled compounds & radiopharmaceuticals (01.02.2003)
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Development of a photoaffinity label for respiratory syncytial virus inhibitors
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Published in Journal of labelled compounds & radiopharmaceuticals (31.10.2003)
Published in Journal of labelled compounds & radiopharmaceuticals (31.10.2003)
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CONTRAST AGENTS FOR MYOCARDIAL PERFUSION IMAGING
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Year of Publication 30.03.2012
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Year of Publication 30.03.2012
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Synthesis of carbon-14 labeled (R)-3-fluoro-4-(2′-(5′′, 6′′, 7′′, 8′′-tetrahydro-5′′, 5′′, 8′′, 8′′-tetramethyl-2′′-naphthyl)-[2′-hydroxy-14C])[carbonyl-14C]acetamidobenzoic acid
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Published in Journal of labelled compounds & radiopharmaceuticals (01.02.2003)
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Microwave-assisted synthesis and chiral HPLC separation of 18F-labeled MaxiPost™. An agent for post-stroke neuroprotection
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Synthesis and Biologic Evaluation of a Novel ^sup 18^F-Labeled Adnectin as a PET Radioligand for Imaging PD-L1 Expression
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Published in The Journal of nuclear medicine (1978) (01.03.2018)
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Published in The Journal of nuclear medicine (1978) (01.03.2018)
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[F-18](R)-5-chloro-1-(1-cyclopropyl-2-methoxyethyl)-3-(4-(2-fluoroethoxy)-2,5-dimethyl phenylamino)pyrazin-2(1H)-one: Introduction of N-3-phenylpyrazinones as potential CRF-R1 PET imaging agents
Deskus, Jeffrey A., Dischino, Douglas D., Mattson, Ronald J., Ditta, Jonathan L., Parker, Michael F., Denhart, Derek J., Zuev, Dmitry, Huang, Hong, Hartz, Richard A., Ahuja, Vijay T., Wong, Henry, Mattson, Gail K., Molski, Thaddeus F., Grace, James E., Zueva, Larisa, Nielsen, Julia M., Dulac, Heidi, Li, Yu-Wen, Guaraldi, Mary, Azure, Michael, Onthank, David, Hayes, Megan, Wexler, Eric, McDonald, Jennifer, Lodge, Nicholas J., Bronson, Joanne J., Macor, John E.
Published in Bioorganic & medicinal chemistry letters (01.11.2012)
Published in Bioorganic & medicinal chemistry letters (01.11.2012)
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Synthesis and Biologic Evaluation of a Novel 18F-Labeled Adnectin as a PET Radioligand for Imaging PD-L1 Expression
Donnelly, David J, Smith, R Adam, Morin, Paul, Lipovšek, Daša, Gokemeijer, Jochem, Cohen, Daniel, Lafont, Virginie, Tran, Tritin, Cole, Erin L, Wright, Martin, Kim, Joonyoung, Pena, Adrienne, Kukral, Daniel, Dischino, Douglas D, Chow, Patrick, Gan, Jinping, Adelakun, Olufemi, Wang, Xi-Tao, Cao, Kai, Leung, David, Bonacorsi, Samuel J, Hayes, Wendy
Published in The Journal of nuclear medicine (1978) (01.03.2018)
Published in The Journal of nuclear medicine (1978) (01.03.2018)
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