A study of the molecular mechanism of binding kinetics and long residence times of human CCR5 receptor small molecule allosteric ligands
Swinney, David C, Beavis, Paul, Chuang, Kai‐Ting, Zheng, Yue, Lee, Ina, Gee, Peter, Deval, Jerome, Rotstein, David M, Dioszegi, Marianna, Ravendran, Palani, Zhang, Jun, Sankuratri, Surya, Kondru, Rama, Vauquelin, Georges
Published in British journal of pharmacology (01.07.2014)
Published in British journal of pharmacology (01.07.2014)
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Development of Tetravalent, Bispecific CCR5 Antibodies with Antiviral Activity against CCR5 Monoclonal Antibody-Resistant HIV-1 Strains
Schanzer, Jürgen, Jekle, Andreas, Nezu, Junichi, Lochner, Adriane, Croasdale, Rebecca, Dioszegi, Marianna, Zhang, Jun, Hoffmann, Eike, Dormeyer, Wilma, Stracke, Jan, Schäfer, Wolfgang, Ji, Changhua, Heilek, Gabrielle, Cammack, Nick, Brandt, Michael, Umana, Pablo, Brinkmann, Ulrich
Published in Antimicrobial Agents and Chemotherapy (01.05.2011)
Published in Antimicrobial Agents and Chemotherapy (01.05.2011)
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CCR5 Small-Molecule Antagonists and Monoclonal Antibodies Exert Potent Synergistic Antiviral Effects by Cobinding to the Receptor
Ji, Changhua, Zhang, Jun, Dioszegi, Marianna, Chiu, Sophie, Rao, Eileen, Derosier, Andre, Cammack, Nick, Brandt, Michael, Sankuratri, Surya
Published in Molecular pharmacology (01.07.2007)
Published in Molecular pharmacology (01.07.2007)
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The Second Extracellular Loop of CCR5 Contains the Dominant Epitopes for Highly Potent Anti-Human Immunodeficiency Virus Monoclonal Antibodies
JUN ZHANG, RAO, Eileen, CHANGHUA JI, DIOSZEGI, Marianna, KONDRU, Rama, DEROSIER, Andre, CHAN, Eva, SCHWOERER, Stephan, CAMMACK, Nick, BRANDT, Michael, SANKURATRI, Surya
Published in Antimicrobial Agents and Chemotherapy (01.04.2007)
Published in Antimicrobial Agents and Chemotherapy (01.04.2007)
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Analyzing ligand and small molecule binding activity of solubilized GPCRs using biosensor technology
Navratilova, Iva, Dioszegi, Marianna, Myszka, David G.
Published in Analytical biochemistry (01.08.2006)
Published in Analytical biochemistry (01.08.2006)
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Increased bone density in sclerosteosis is due to the deficiency of a novel secreted protein (SOST)
BALEMANS, Wendy, EBELING, Martin, PAES-ALVES, Auristela F, HILL, Suvimol, BUENO, Manuel, RAMOS, Feliciano J, TACCONI, Paoio, DIKKERS, Frederik G, STRATAKIS, Constantine, LINDPAINTNER, Klaus, VICKERY, Brian, FOERNZLER, Dorothee, PATEL, Neela, VAN HUL, Wim, VAN HUL, Els, OLSON, Pam, DIOSZEGI, Marianna, LACZA, Charlemagne, WUYTS, Wim, VAN DEN ENDE, Jenneke, WILLEMS, Patrick
Published in Human molecular genetics (01.03.2001)
Published in Human molecular genetics (01.03.2001)
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Journal Article
A study of the molecular mechanism of binding kinetics and long residence times of human CCR 5 receptor small molecule allosteric ligands
Swinney, David C, Beavis, Paul, Chuang, Kai‐Ting, Zheng, Yue, Lee, Ina, Gee, Peter, Deval, Jerome, Rotstein, David M, Dioszegi, Marianna, Ravendran, Palani, Zhang, Jun, Sankuratri, Surya, Kondru, Rama, Vauquelin, Georges
Published in British journal of pharmacology (01.07.2014)
Published in British journal of pharmacology (01.07.2014)
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Journal Article
Spiropiperidine CCR5 antagonists
Rotstein, David M., Gabriel, Stephen D., Makra, Ferenc, Filonova, Lubov, Gleason, Shelley, Brotherton-Pleiss, Christine, Setti, Lina Q., Trejo-Martin, Alejandra, Lee, Eun Kyung, Sankuratri, Surya, Ji, Changhua, deRosier, Andre, Dioszegi, Marianna, Heilek, Gabrielle, Jekle, Andreas, Berry, Pamela, Weller, Paul, Mau, Cheng-I.
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
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Synthesis, SAR and evaluation of [1,4′]-bipiperidinyl-4-yl-imidazolidin-2-one derivatives as novel CCR5 antagonists
Rotstein, David M., Gabriel, Stephen D., Manser, Nicole, Filonova, Lubov, Padilla, Fernando, Sankuratri, Surya, Ji, Changhua, deRosier, Andre, Dioszegi, Marianna, Heilek, Gabrielle, Jekle, Andreas, Weller, Paul, Berry, Pamela
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
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Novel CCR5 monoclonal antibodies with potent and broad-spectrum anti-HIV activities
Ji, Changhua, Brandt, Michael, Dioszegi, Marianna, Jekle, Andreas, Schwoerer, Stephan, Challand, Steven, Zhang, Jun, Chen, Yun, Zautke, Lisa, Achhammer, Gunthar, Baehner, Monika, Kroetz, Sandra, Heilek-Snyder, Gabrielle, Schumacher, Ralf, Cammack, Nick, Sankuratri, Surya
Published in Antiviral research (01.05.2007)
Published in Antiviral research (01.05.2007)
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Journal Article
Novel hexahydropyrrolo[3,4- c]pyrrole CCR5 antagonists
Rotstein, David M., Melville, Chris R., Padilla, Fernando, Cournoyer, Dick, Lee, Eun K., Lemoine, Remy, Petersen, Ann C., Setti, Lina Q., Wanner, Jutta, Chen, Lijing, Filonova, Lubov, Loughhead, David G., Manka, Jason, Lin, Xiao-Fa, Gleason, Shelley, Sankuratri, Surya, Ji, Changhua, deRosier, Andre, Dioszegi, Marianna, Heilek, Gabrielle, Jekle, Andreas, Berry, Pamela, Mau, Cheng-I, Weller, Paul
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Journal Article
Characterization of 58-kilodalton human neutrophil collagenase: comparison with human fibroblast collagenase
Mallya, Satish K, Mookhtiar, Kasim A, Gao, Yi, Brew, Keith, Dioszegi, Marianna, Birkedal-Hansen, Henning, Van Wart, Harold E
Published in Biochemistry (Easton) (01.11.1990)
Published in Biochemistry (Easton) (01.11.1990)
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Improved process for the preparation of tripeptide aldehydes
ATTILA JUHASZ, EMILIA USKERT, ERNOE ORBAN, EVA TOMORI, MARIANNA DIOSZEGI, ATTILA NAGY, GYULA HORVATH, ZSUZSANNA LANG, ERZSEBET SZELL, GYOERGY SOMOGYI, KATALIN SZILAGYI, SANDOR ELEK, ZSUZSA PESTI, LAJOS ILA, TIBOR BALOGH, KATALIN PAL, TIBOR LANG, EVA BARABAS
Year of Publication 19.01.1994
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Year of Publication 19.01.1994
Patent
PREPARATION OF TRIPEPTIDE ALDEHYDES
JUHASZ, ATTILA, SZELL, ERZSEBET, PAL, KATALIN, SOMOGYI, GYORGY, ORBAN, ERNO, LANG, TIBOR, BARABAS, EVA, DIOSZEGI, MARIANNA, PESTI, ZSUZSA, HORVATH, GYULA, ELEK, SANDOR, NAGY, ATTILA, BALOGH, TIBOR, LANG, ZSUZSANNA, SZILAGYI, KATALIN, ILA, LAJOS, TOMOR
Year of Publication 26.08.1993
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Year of Publication 26.08.1993
Patent
Preparation of tripeptide aldehydes
ATTILA JUHASZ, GYORGY SOMOGYI, EVA TOMORI, MARIANNA DIOSZEGI, ATTILA NAGY, GYULA HORVATH, ZSUZSANNA LANG, ERZSEBET SZELL, DR EMILIA USKERT, KATALIN SZILAGYI, ERNO ORBAN, SANDOR ELEK, ZSUZSA PESTI, LAJOS ILA, TIBOR BALOGH, KATALIN PAL, TIBOR LANG, EVA BARABAS
Year of Publication 18.12.1991
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Year of Publication 18.12.1991
Patent
IMPROVED PROCESS FOR THE PREPARATION OF TRIPEPTIDE ALDEHYDES
ATTILA, JUHASZ DR, ERZSEBET, SZELL, GYOERGY, SOMOGYI, EVA, BARABAS DR, LAJOS, ILA DR, ERNO, ORBAN DR, TIBOR, LANG DR, KATALIN, PAL DR, ATTILA, NAGY, MARIANNA, DIOSZEGI, ZSUZSA, PESTI, EMILIA, USKERT DR, KATALIN, SZILAGYI DR, ZSUZSANA, LANG, TIBOR, BALOGH DR, SANDOR, ELEK DR, GYULA, HORVATH DR, EVA, TOMORI DR
Year of Publication 07.07.2003
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Year of Publication 07.07.2003
Patent
Fremgangsmåte ved fremstilling av tripeptidaldehyder
JUHASZ, ATTILA, SZELL, ERZSEBET, PAL, KATALIN, SOMOGYI, GYORGY, ORBAN, ERNO, LANG, TIBOR, BARABAS, EVA, DIOSZEGI, MARIANNA, PESTI, ZSUZSA, HORVATH, GYULA, ELEK, SANDOR, NAGY, ATTILA, BALOGH, TIBOR, USKERT, EMILIA, LANG, ZSUZSANNA, SZILAGYI, KATALIN, TOMORI, EVA, ILA, LAJOS
Year of Publication 10.05.1995
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Year of Publication 10.05.1995
Patent
Fremgangsmåte ved fremstilling av tripeptidaldehyder
JUHASZ, ATTILA, SZELL, ERZSEBET, PAL, KATALIN, SOMOGYI, GYORGY, ORBAN, ERNO, LANG, TIBOR, BARABAS, EVA, DIOSZEGI, MARIANNA, PESTI, ZSUZSA, HORVATH, GYULA, ELEK, SANDOR, NAGY, ATTILA, BALOGH, TIBOR, USKERT, EMILIA, LANG, ZSUZSANNA, SZILAGYI, KATALIN, TOMORI, EVA, ILA, LAJOS
Year of Publication 30.01.1995
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Year of Publication 30.01.1995
Patent