PARP1 Trapping by PARP Inhibitors Drives Cytotoxicity in Both Cancer Cells and Healthy Bone Marrow
Hopkins, Todd A, Ainsworth, William B, Ellis, Paul A, Donawho, Cherrie K, DiGiammarino, Enrico L, Panchal, Sanjay C, Abraham, Vivek C, Algire, Mikkel A, Shi, Yan, Olson, Amanda M, Johnson, Eric F, Wilsbacher, Julie L, Maag, David
Published in Molecular cancer research (01.02.2019)
Published in Molecular cancer research (01.02.2019)
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Journal Article
Mechanistic Dissection of PARP1 Trapping and the Impact on In Vivo Tolerability and Efficacy of PARP Inhibitors
Hopkins, Todd A, Shi, Yan, Rodriguez, Luis E, Solomon, Larry R, Donawho, Cherrie K, DiGiammarino, Enrico L, Panchal, Sanjay C, Wilsbacher, Julie L, Gao, Wenqing, Olson, Amanda M, Stolarik, DeAnne F, Osterling, Donald J, Johnson, Eric F, Maag, David
Published in Molecular cancer research (01.11.2015)
Published in Molecular cancer research (01.11.2015)
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Journal Article
Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours
Lasko, Loren M., Jakob, Clarissa G., Edalji, Rohinton P., Qiu, Wei, Montgomery, Debra, Digiammarino, Enrico L., Hansen, T. Matt, Risi, Roberto M., Frey, Robin, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Hessler, Paul, Lam, Lloyd T., Uziel, Tamar, Faivre, Emily, Ferguson, Debra, Buchanan, Fritz G., Martin, Ruth L., Torrent, Maricel, Chiang, Gary G., Karukurichi, Kannan, Langston, J. William, Weinert, Brian T., Choudhary, Chunaram, de Vries, Peter, Kluge, Arthur F., Patane, Michael A., Van Drie, John H., Wang, Ce, McElligott, David, Kesicki, Ed, Marmorstein, Ronen, Sun, Chaohong, Cole, Philip A., Rosenberg, Saul H., Michaelides, Michael R., Lai, Albert, Bromberg, Kenneth D.
Published in Nature (London) (05.10.2017)
Published in Nature (London) (05.10.2017)
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Journal Article
Ligand association rates to the inner-variable-domain of a dual-variable-domain immunoglobulin are significantly impacted by linker design
DiGiammarino, Enrico L., Harlan, John E., Walter, Karl A., Ladror, Uri S., Edalji, Rohinton P., Hutchins, Charles W., Lake, Marc R., Greischar, Amy J., Liu, Junjian, Ghayur, Tariq, Jakob, Clarissa G.
Published in mAbs (01.09.2011)
Published in mAbs (01.09.2011)
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Journal Article
Reversible Amyloid Formation by the p53 Tetramerization Domain and a Cancer-associated Mutant
Lee, Amanda S., Galea, Charles, DiGiammarino, Enrico L., Jun, Bokkyoo, Murti, Gopal, Ribeiro, Raul C., Zambetti, Gerard, Schultz, Christian P., Kriwacki, Richard W.
Published in Journal of molecular biology (28.03.2003)
Published in Journal of molecular biology (28.03.2003)
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Characterization of ABT-806, a Humanized Tumor-Specific Anti-EGFR Monoclonal Antibody
Reilly, Edward B, Phillips, Andrew C, Buchanan, Fritz G, Kingsbury, Gillian, Zhang, Yumin, Meulbroek, Jonathan A, Cole, Todd B, DeVries, Peter J, Falls, Hugh D, Beam, Christine, Gu, Jinming, Digiammarino, Enrico L, Palma, Joann P, Donawho, Cherrie K, Goodwin, Neal C, Scott, Andrew M
Published in Molecular cancer therapeutics (01.05.2015)
Published in Molecular cancer therapeutics (01.05.2015)
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ABT-165, a Dual Variable Domain Immunoglobulin (DVD-Ig) Targeting DLL4 and VEGF, Demonstrates Superior Efficacy and Favorable Safety Profiles in Preclinical Models
Li, Yingchun, Hickson, Jonathan A, Ambrosi, Dominic J, Haasch, Deanna L, Foster-Duke, Kelly D, Eaton, Lucia J, DiGiammarino, Enrico L, Panchal, Sanjay C, Jiang, Fang, Mudd, Sarah R, Zhang, Catherine, Akella, Surekha S, Gao, Wenqing, Ralston, Sherry L, Naumovski, Louie, Gu, Jijie, Morgan-Lappe, Susan E
Published in Molecular cancer therapeutics (01.05.2018)
Published in Molecular cancer therapeutics (01.05.2018)
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Author Correction: Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours
Lasko, Loren M., Jakob, Clarissa G., Edalji, Rohinton P., Qiu, Wei, Montgomery, Debra, Digiammarino, Enrico L., Hansen, T. Matt, Risi, Roberto M., Frey, Robin, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Hessler, Paul, Lam, Lloyd T., Uziel, Tamar, Faivre, Emily, Ferguson, Debra, Buchanan, Fritz G., Martin, Ruth L., Torrent, Maricel, Chiang, Gary G., Karukurichi, Kannan, Langston, J. William, Weinert, Brian T., Choudhary, Chunaram, de Vries, Peter, Kluge, Arthur F., Patane, Michael A., Van Drie, John H., Wang, Ce, McElligott, David, Kesicki, Edward A., Marmorstein, Ronen, Sun, Chaohong, Cole, Philip A., Rosenberg, Saul H., Michaelides, Michael R., Lai, Albert, Bromberg, Kenneth D.
Published in Nature (London) (01.06.2018)
Published in Nature (London) (01.06.2018)
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Journal Article
A novel mechanism of tumorigenesis involving pH-dependent destabilization of a mutant p53 tetramer
Kriwacki, Richard W, DiGiammarino, Enrico L, Lee, Amanda S, Cadwell, Craig, Zhang, Weixing, Bothner, Brian, Ribeiro, Raul C, Zambetti, Gerard
Published in Nature structural & molecular biology (01.01.2002)
Published in Nature structural & molecular biology (01.01.2002)
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Journal Article
Cooperative Signals Governing ARF-Mdm2 Interaction and Nucleolar Localization of the Complex
Weber, Jason D., Kuo, Mei-Ling, Bothner, Brian, DiGiammarino, Enrico L., Kriwacki, Richard W., Roussel, Martine F., Sherr, Charles J.
Published in Molecular and Cellular Biology (01.04.2000)
Published in Molecular and Cellular Biology (01.04.2000)
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Defining the molecular basis of Arf and Hdm2 interactions
Bothner, B, Lewis, W S, DiGiammarino, E L, Weber, J D, Bothner, S J, Kriwacki, R W
Published in Journal of molecular biology (23.11.2001)
Published in Journal of molecular biology (23.11.2001)
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Journal Article
ANTIBODIES TO RECEPTOR OF ADVANCED GLYCATION END PRODUCTS (RAGE) AND USES THEREOF
DIGIAMMARINO ENRICO L, NIMMRICH VOLKER, HSIEH CHUNG MING, SCHMIDT MARTIN, WU ZHEN, MUELLER REINHOLD, GU JIJIE, LUO FENG, FOX GERARD B, EBERT ULRICH, HARLAN JOHN E, LOEBBERT RALF
Year of Publication 13.09.2016
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Year of Publication 13.09.2016
Patent
Solution Studies of Isepamicin and Conformational Comparisons between Isepamicin and Butirosin A When Bound to an Aminoglycoside 6‘-N-Acetyltransferase Determined by NMR Spectroscopy
DiGiammarino, Enrico L, Draker, Kari-ann, Wright, Gerard D, Serpersu, Engin H
Published in Biochemistry (Easton) (17.03.1998)
Published in Biochemistry (Easton) (17.03.1998)
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ANTIBODIES TO RECEPTOR OF ADVANCED GLYCATION END PRODUCTS (RAGE) AND USES THEREOF
DIGIAMMARINO ENRICO L, NIMMRICH VOLKER, HSIEH CHUNG MING, SCHMIDT MARTIN, WU ZHEN, MUELLER REINHOLD, GU JIJIE, LUO FENG, FOX GERARD B, EBERT ULRICH, HARLAN JOHN E, LOEBBERT RALF
Year of Publication 22.03.2016
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Year of Publication 22.03.2016
Patent
ANTIBODIES TO RECEPTOR OF ADVANCED GLYCATION END PRODUCTS (RAGE) AND USES THEREOF
DIGIAMMARINO ENRICO L, NIMMRICH VOLKER, HSIEH CHUNG MING, SCHMIDT MARTIN, WU ZHEN, MUELLER REINHOLD, GU JIJIE, LUO FENG, FOX GERARD B, EBERT ULRICH, HARLAN JOHN E, LOEBBERT RALF
Year of Publication 03.11.2015
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Year of Publication 03.11.2015
Patent
PROLACTIN RECEPTOR BINDING PROTEINS AND USES THEREOF
LONGENECKER KENTON L, HUTCHINS CHARLES W, DIGIAMMARINO ENRICO L, HSIEH CHUNG MING, ANDERSON MARK, REILLY EDWARD B, ZHANG QIAN, JUDGE RUSSELL A, EGAN DAVID A, THAKUR ARCHANA, CHAO DEBRA, WANG JIEYI
Year of Publication 02.09.2015
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Year of Publication 02.09.2015
Patent
Solution Structure of the p53 Regulatory Domain of the p19Arf Tumor Suppressor Protein
DiGiammarino, Enrico L, Filippov, Igor, Weber, Jason D, Bothner, Brian, Kriwacki, Richard W
Published in Biochemistry (Easton) (27.02.2001)
Published in Biochemistry (Easton) (27.02.2001)
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Journal Article
Abstract 2850: Talazoparib (BMN-673) possesses greater PARP1 trapping activity than structurally distinct PARP inhibitors with identical PARP1 binding properties
Hopkins, Todd A., Shi, Yan Y., DiGiammarino, Enrico L., Panchal, Sanjay C., Zhu, Gui-Dong G., Penning, Thomas D., Johnson, Eric F., Maag, David
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Abstract C52: PARP1 trapping activity of PARP inhibitors is associated with cytotoxicity in both cancer cells and healthy bone marrow
Hopkins, Todd A., Wilsbacher, Julie L., DiGiammarino, Enrico L., Panchal, Sanjay C., Zhu, Gui-Dong, Penning, Thomas D., Johnson, Eric F., Maag, David
Published in Molecular cancer therapeutics (01.12.2015)
Published in Molecular cancer therapeutics (01.12.2015)
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