Identification and Preliminary Characterization of a Potent, Safe, and Orally Efficacious Inhibitor of Acyl-CoA:Diacylglycerol Acyltransferase 1
Yeh, Vince S. C, Beno, David W. A, Brodjian, Sevan, Brune, Michael E, Cullen, Steven C, Dayton, Brian D, Dhaon, Madhup K, Falls, Hugh D, Gao, Ju, Grihalde, Nelson, Hajduk, Philip, Hansen, T. Matthew, Judd, Andrew S, King, Andrew J, Klix, Russel C, Larson, Kelly J, Lau, Yau Y, Marsh, Kennan C, Mittelstadt, Scott W, Plata, Dan, Rozema, Michael J, Segreti, Jason A, Stoner, Eric J, Voorbach, Martin J, Wang, Xiaojun, Xin, Xili, Zhao, Gang, Collins, Christine A, Cox, Bryan F, Reilly, Regina M, Kym, Philip R, Souers, Andrew J
Published in Journal of medicinal chemistry (23.02.2012)
Published in Journal of medicinal chemistry (23.02.2012)
Get full text
Journal Article
Normal phase and reverse phase HPLC-UV-MS analysis of process impurities for rapamycin analog ABT-578: Application to active pharmaceutical ingredient process development
Chen, Yong, Brill, Gregory M., Benz, Nancy J., Leanna, M. Robert, Dhaon, Madhup K., Rasmussen, Michael, Zhou, Casey Chun, Bruzek, James A., Bellettini, John R.
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.10.2007)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.10.2007)
Get full text
Journal Article
BOP-Cl mediated synthesis of the cyclosporine A 8-11 tetrapeptide fragment
Tung, Roger D, Dhaon, Madhup K, Rich, Daniel H
Published in Journal of organic chemistry (01.08.1986)
Published in Journal of organic chemistry (01.08.1986)
Get full text
Journal Article
ONE POT SYNTHESIS OF TETRAZOLE DERIVATIVES OF SIROLIMUS
CHEN YONG, BURKAR SANJAY, PATEL SUBHASH, DHAON MADHUP, HSIAO CHU NUNG, BONK PETER
Year of Publication 05.09.2017
Get full text
Year of Publication 05.09.2017
Patent
ONE POT SYNTHESIS OF TETRAZOLE DERIVATIVES OF SIROLIMUS
CHEN YONG, BURKAR SANJAY, PATEL SUBHASH, DHAON MADHUP, HSIAO CHU NUNG, BONK PETER
Year of Publication 25.01.2017
Get full text
Year of Publication 25.01.2017
Patent
Synthesis, isolation, and characterization of ABT-578 equilibrium isomers
Dhaon, Madhup K., Zhou, Casey C., Chemburkar, Sanjay, Morton, Howard
Published in Tetrahedron letters (05.02.2007)
Published in Tetrahedron letters (05.02.2007)
Get full text
Journal Article
ONE POT SYNTHESIS OF TETRAZOLE DERIVATIVES OF SIROLIMUS
CHEN YONG, BURKAR SANJAY, PATEL SUBHASH, DHAON MADHUP, HSIAO CHU NUNG, BONK PETER
Year of Publication 08.01.2016
Get full text
Year of Publication 08.01.2016
Patent
ONE POT SYNTHESIS OF TETRAZOLE DERIVATIVES OF SIROLIMUS
CHEN YONG, BURKAR SANJAY, PATEL SUBHASH, DHAON MADHUP, HSIAO CHU NUNG, BONK PETER
Year of Publication 27.05.2015
Get full text
Year of Publication 27.05.2015
Patent
ONE POT SYNTHESIS OF TETRAZOLE DERIVATIVES OF SIROLIMUS
CHEN YONG, BURKAR SANJAY, PATEL SUBHASH, DHAON MADHUP, HSIAO CHU NUNG, BONK PETER
Year of Publication 07.01.2015
Get full text
Year of Publication 07.01.2015
Patent
A short synthesis of enantiomerically pure (2S,3R,4R,6E)-3-hydroxy-4-methyl-2-(methylamino)-6-octenoic acid, the unusual C9 amino acid found in the immunosuppressive peptide cyclosporine
Aebi, Johannes D, Dhaon, Madhup K, Rich, Daniel H
Published in Journal of organic chemistry (01.06.1987)
Published in Journal of organic chemistry (01.06.1987)
Get full text
Journal Article
ONE POT SYNTHESIS OF TETRAZOLE DERIVATIVES OF SIROLIMUS
CHEN YONG, BURKAR SANJAY, PATEL SUBHASH, DHAON MADHUP, HSIAO CHU NUNG, BONK PETER
Year of Publication 06.11.2013
Get full text
Year of Publication 06.11.2013
Patent
ONE POT SYNTHESIS OF TETRAZOLE DERIVATIVES OF SIROLIMUS
BURKAR, SANJAY, BONK, PETER, PATEL, SUBHASH, CHEN, YONG, HSIAO, CHI-NUNG, DHAON, MADHUP
Year of Publication 17.04.2018
Get full text
Year of Publication 17.04.2018
Patent
ONE POT SYNTHESIS OF TETRAZOLE DERIVATIVES OF SIROLIMUS
PATEL, Subhash, DHAON, Madhup, CHEN, Yong, HSIAO, Chu-nung, BONK, Peter, BURKAR, Sanjay
Year of Publication 28.02.2018
Get full text
Year of Publication 28.02.2018
Patent
Síntesis en un solo reactor de derivados tetrazólicos de sirolimus
Chen, Yong, Hsiao, Chu-nung, Patel, Subhash, Dhaon, Madhup, Chemburkar, Sanjay, Bonk, Peter
Year of Publication 15.11.2017
Get full text
Year of Publication 15.11.2017
Patent
One pot synthesis of tetrazole derivatives of sirolimus
Chen, Yong, Hsiao, Chu-nung, Patel, Subhash, Dhaon, Madhup, Chemburkar, Sanjay, Bonk, Peter
Year of Publication 06.09.2017
Get full text
Year of Publication 06.09.2017
Patent