Differential targeting of brain stress circuits with a selective glucocorticoid receptor modulator
Zalachoras, Ioannis, Houtman, René, Atucha, Erika, Devos, Rene, Tijssen, Ans M. I., Hu, Pu, Lockey, Peter M., Datson, Nicole A., Belanoff, Joseph K., Lucassen, Paul J., Joëls, Marian, de Kloet, E. Ronald, Roozendaal, Benno, Hunt, Hazel, Meijer, Onno C.
Published in Proceedings of the National Academy of Sciences - PNAS (07.05.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (07.05.2013)
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The Novel Nucleoside Analog R1479 (4′-Azidocytidine) Is a Potent Inhibitor of NS5B-dependent RNA Synthesis and Hepatitis C Virus Replication in Cell Culture
Klumpp, Klaus, Lévêque, Vincent, Le Pogam, Sophie, Ma, Han, Jiang, Wen-Rong, Kang, Hyunsoon, Granycome, Caroline, Singer, Margaret, Laxton, Carl, Hang, Julie Qi, Sarma, Keshab, Smith, David B., Heindl, Dieter, Hobbs, Chris J., Merrett, John H., Symons, Julian, Cammack, Nick, Martin, Joseph A., Devos, Rene, Nájera, Isabel
Published in The Journal of biological chemistry (17.02.2006)
Published in The Journal of biological chemistry (17.02.2006)
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Journal Article
Recombinant mouse OB protein: evidence for a peripheral signal linking adiposity and central neural networks
Campfield, L.A. (Hoffmann-La Roche Incorporated, Nutley, NJ.), Smith, F.J, Guisez, Y, Devos, R, Burn, P
Published in Science (American Association for the Advancement of Science) (28.07.1995)
Published in Science (American Association for the Advancement of Science) (28.07.1995)
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Journal Article
Identification and expression cloning of a leptin receptor, OB-R
Tartaglia, Louis A., Dembski, Marlene, Weng, Xun, Deng, Nanhua, Culpepper, Janice, Devos, Rene, Richards, Grayson J., Campfield, L.Arthur, Clark, Frederick T., Deeds, Jim, Muir, Craig, Sanker, Sean, Moriarty, Ann, Moore, Karen J., Smutko, John S., Mays, Gail G., Wool, Elizabeth A., Monroe, Cheryl A., Tepper, Robert I.
Published in Cell (29.12.1995)
Published in Cell (29.12.1995)
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Journal Article
Discovery and optimization of novel, non-steroidal glucocorticoid receptor modulators
Ray, Nicholas C., Clark, Robin D., Clark, David E., Williams, Karen, Hickin, H.G., Crackett, Peter H., Dyke, Hazel J., Lockey, Peter M., Wong, Melanie, Devos, René, White, Anne, Belanoff, Joseph K.
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Journal Article
Role of IFN-gamma in the Inhibition of the Allergic Airway Inflammation Caused by IL-12
Brusselle, Guy G, Kips, Johan C, Peleman, Renaat A, Joos, Guy F, Devos, Rene R, Tavernier, Jan H, Pauwels, Romain A
Published in American journal of respiratory cell and molecular biology (01.12.1997)
Published in American journal of respiratory cell and molecular biology (01.12.1997)
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Journal Article
Leptin Receptor (OB-R) Signaling
White, David W., Kuropatwinski, Karen K., Devos, Rene, Baumann, Heinz, Tartaglia, Louis A.
Published in The Journal of biological chemistry (14.02.1997)
Published in The Journal of biological chemistry (14.02.1997)
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Journal Article
Ligand-independent Dimerization of the Extracellular Domain of the Leptin Receptor and Determination of the Stoichiometry of Leptin Binding
Devos, René, Guisez, Yves, Van der Heyden, José, White, David W., Kalai, Michael, Fountoulakis, Michael, Plaetinck, Geert
Published in The Journal of biological chemistry (18.07.1997)
Published in The Journal of biological chemistry (18.07.1997)
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Journal Article
Abstract 5137: Parallel approaches to the discovery of novel BRD4 inhibitors
Jones, David H., Groot, Marcel J. de, Heald, Robert, Arhin, Ebenezer, Goodwin, Ria, Burton, Brenda, Kulagowski, Jan, Brown, David, Irving, Steven, Bazin, Richard, Bruce, Deborah, Devos, Rene, Price, Steven, Ray, Nick, Lockey, Peter, Montana, John, Albertella, Mark R., Green, Simon R.
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Journal Article
Design, synthesis, and antiviral properties of 4′-substituted ribonucleosides as inhibitors of hepatitis C virus replication: The discovery of R1479
Smith, David B., Martin, Joseph A., Klumpp, Klaus, Baker, Stewart J., Blomgren, Peter A., Devos, Rene, Granycome, Caroline, Hang, Julie, Hobbs, Christopher J., Jiang, Wen-Rong, Laxton, Carl, Pogam, Sophie Le, Leveque, Vincent, Ma, Han, Maile, Graham, Merrett, John H., Pichota, Arkadius, Sarma, Keshab, Smith, Mark, Swallow, Steven, Symons, Julian, Vesey, David, Najera, Isabel, Cammack, Nick
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
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Journal Article
High-level expression of human interferon gamma in Escherichia coli under control of the pL promoter of bacteriophage lambda
Simons, Guus, Remaut, Erik, Allet, Bernard, Devos, Rene, Fiers, Walter
Published in Gene (01.04.1984)
Published in Gene (01.04.1984)
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Journal Article
1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity
CLARK, Robin D, RAY, Nicholas C, DEVOS, Rene, WONG, Melanie, PORRES, Soraya S, BRIGHT, Colin P, JENKINS, Robert E, BELANOFF, Joseph, WILLIAMS, Karen, BLANEY, Paul, WARD, Stuart, CRACKETT, Peter H, HURLEY, Christopher, DYKE, Hazel J, CLARK, David E, LOCKEY, Peter
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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Journal Article
Leptin receptor (OB-R) signaling: cytoplasmic domain mutational analysis and evidence for receptor homo-oligomerization
White, D.W. (Millennium Pharmaceuticals, Cambridge, MA.), Kuropatwinski, K.K, Devos, R, Baumann, H, Tartaglia, L.A
Published in The Journal of biological chemistry (14.02.1997)
Published in The Journal of biological chemistry (14.02.1997)
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Journal Article
A human leptin mutant induces weight gain in normal mice
Verploegen, Sandra A.B.W., Plaetinck, Geert, Devos, René, Van der Heyden, José, Guisez, Yves
Published in FEBS letters (24.03.1997)
Published in FEBS letters (24.03.1997)
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Journal Article
Comparison of R128Q Mutations in Human, Ovine, and Chicken Leptins
Raver, Nina, Vardy, Eyal, Livnah, Oded, Devos, Rene, Gertler, Arieh
Published in General and comparative endocrinology (01.03.2002)
Published in General and comparative endocrinology (01.03.2002)
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Journal Article
2-Benzenesulfonyl-8a-benzyl-hexahydro-2H-isoquinolin-6-ones as selective glucocorticoid receptor antagonists
Clark, Robin D., Ray, Nicholas C., Blaney, Paul, Crackett, Peter H., Hurley, Christopher, Williams, Karen, Dyke, Hazel J., Clark, David E., Lockey, Peter M., Devos, Rene, Wong, Melanie, White, Anne, Belanoff, Joseph K.
Published in Bioorganic & medicinal chemistry letters (15.10.2007)
Published in Bioorganic & medicinal chemistry letters (15.10.2007)
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Journal Article
1 H-Pyrazolo[3,4- g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity
Clark, Robin D., Ray, Nicholas C., Williams, Karen, Blaney, Paul, Ward, Stuart, Crackett, Peter H., Hurley, Christopher, Dyke, Hazel J., Clark, David E., Lockey, Peter, Devos, Rene, Wong, Melanie, Porres, Soraya S., Bright, Colin P., Jenkins, Robert E., Belanoff, Joseph
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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Journal Article
OB protein binds specifically to the choroid plexus of mice and rats
Devos, R. (Roche Research Gent, Gent, Belgium.), Richards, J.G, Campfield, L.A, Tartaglia, L.A, Guisez, Y, Heyden, J. van der, Travernier, J, Plaetinck, G, Burn, P
Published in Proceedings of the National Academy of Sciences - PNAS (28.05.1996)
Published in Proceedings of the National Academy of Sciences - PNAS (28.05.1996)
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