Crystal structure, biochemical and cellular activities demonstrate separate functions of MTH1 and MTH2
Carter, Megan, Jemth, Ann-Sofie, Hagenkort, Anna, Page, Brent D G, Gustafsson, Robert, Griese, Julia J, Gad, Helge, Valerie, Nicholas C K, Desroses, Matthieu, Boström, Johan, Warpman Berglund, Ulrika, Helleday, Thomas, Stenmark, Pål
Published in Nature communications (04.08.2015)
Published in Nature communications (04.08.2015)
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Journal Article
A microwave-assisted, propylphosphonic anhydride (T3P®) mediated one-pot Fischer indole synthesis
Desroses, Matthieu, Wieckowski, Krzysztof, Stevens, Marc, Odell, Luke R.
Published in Tetrahedron letters (24.08.2011)
Published in Tetrahedron letters (24.08.2011)
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Journal Article
Crystal structure of human MTH1 and the 8-oxo-dGMP product complex
Svensson, Linda M., Jemth, Ann-Sofie, Desroses, Matthieu, Loseva, Olga, Helleday, Thomas, Högbom, Martin, Stenmark, Pål
Published in FEBS letters (19.08.2011)
Published in FEBS letters (19.08.2011)
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Journal Article
Development of a chemical probe against NUDT15
Zhang, Si Min, Desroses, Matthieu, Hagenkort, Anna, Valerie, Nicholas C K, Rehling, Daniel, Carter, Megan, Wallner, Olov, Koolmeister, Tobias, Throup, Adam, Jemth, Ann-Sofie, Almlöf, Ingrid, Loseva, Olga, Lundbäck, Thomas, Axelsson, Hanna, Regmi, Shruti, Sarno, Antonio, Krämer, Andreas, Pudelko, Linda, Bräutigam, Lars, Rasti, Azita, Göttmann, Mona, Wiita, Elisée, Kutzner, Juliane, Schaller, Torsten, Kalderén, Christina, Cázares-Körner, Armando, Page, Brent D G, Krimpenfort, Rosa, Eshtad, Saeed, Altun, Mikael, Rudd, Sean G, Knapp, Stefan, Scobie, Martin, Homan, Evert J, Berglund, Ulrika Warpman, Stenmark, Pål, Helleday, Thomas
Published in Nature chemical biology (01.10.2020)
Published in Nature chemical biology (01.10.2020)
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Journal Article
STAT3 differential scanning fluorimetry and differential scanning light scattering assays: Addressing a missing link in the characterization of STAT3 inhibitor interactions
Desroses, Matthieu, Busker, Sander, Astorga-Wells, Juan, Attarha, Sanaz, Kolosenko, Iryna, Zubarev, Roman A., Helleday, Thomas, Grandér, Dan, Page, Brent D.G.
Published in Journal of pharmaceutical and biomedical analysis (25.10.2018)
Published in Journal of pharmaceutical and biomedical analysis (25.10.2018)
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Journal Article
dUTPase inhibition augments replication defects of 5-Fluorouracil
Hagenkort, Anna, Paulin, Cynthia B J, Desroses, Matthieu, Sarno, Antonio, Wiita, Elisée, Mortusewicz, Oliver, Koolmeister, Tobias, Loseva, Olga, Jemth, Ann-Sofie, Almlöf, Ingrid, Homan, Evert, Lundbäck, Thomas, Gustavsson, Anna-Lena, Scobie, Martin, Helleday, Thomas
Published in Oncotarget (04.04.2017)
Published in Oncotarget (04.04.2017)
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Journal Article
Exploring Drug Target Flexibility Using in Situ Click Chemistry: Application to a Mycobacterial Transcriptional Regulator
Willand, Nicolas, Desroses, Matthieu, Toto, Patrick, Dirié, Bertrand, Lens, Zoé, Villeret, Vincent, Rucktooa, Prakash, Locht, Camille, Baulard, Alain, Deprez, Benoit
Published in ACS chemical biology (19.11.2010)
Published in ACS chemical biology (19.11.2010)
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Journal Article
A Convenient Microwave-Assisted Propylphosphonic Anhydride (T3P®) Mediated One-Pot Pyrazolone Synthesis
Desroses, Matthieu, Jacques-Cordonnier, Marie-Caroline, Llona-Minguez, Sabin, Jacques, Sylvain, Koolmeister, Tobias, Helleday, Thomas, Scobie, Martin
Published in European journal of organic chemistry (01.09.2013)
Published in European journal of organic chemistry (01.09.2013)
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Journal Article
MTH1 inhibition eradicates cancer by preventing sanitation of the dNTP pool
Gad, Helge, Koolmeister, Tobias, Jemth, Ann-Sofie, Eshtad, Saeed, Jacques, Sylvain A, Ström, Cecilia E, Svensson, Linda M, Schultz, Niklas, Lundbäck, Thomas, Einarsdottir, Berglind Osk, Saleh, Aljona, Göktürk, Camilla, Baranczewski, Pawel, Svensson, Richard, Berntsson, Ronnie P-A, Gustafsson, Robert, Strömberg, Kia, Sanjiv, Kumar, Jacques-Cordonnier, Marie-Caroline, Desroses, Matthieu, Gustavsson, Anna-Lena, Olofsson, Roger, Johansson, Fredrik, Homan, Evert J, Loseva, Olga, Bräutigam, Lars, Johansson, Lars, Höglund, Andreas, Hagenkort, Anna, Pham, Therese, Altun, Mikael, Gaugaz, Fabienne Z, Vikingsson, Svante, Evers, Bastiaan, Henriksson, Martin, Vallin, Karl S A, Wallner, Olov A, Hammarström, Lars G J, Wiita, Elisee, Almlöf, Ingrid, Kalderén, Christina, Axelsson, Hanna, Djureinovic, Tatjana, Puigvert, Jordi Carreras, Häggblad, Maria, Jeppsson, Fredrik, Martens, Ulf, Lundin, Cecilia, Lundgren, Bo, Granelli, Ingrid, Jensen, Annika Jenmalm, Artursson, Per, Nilsson, Jonas A, Stenmark, Pål, Scobie, Martin, Berglund, Ulrika Warpman, Helleday, Thomas
Published in Nature (London) (10.04.2014)
Published in Nature (London) (10.04.2014)
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Journal Article
Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420
Blondiaux, Nicolas, Moune, Martin, Desroses, Matthieu, Frita, Rosangela, Flipo, Marion, Mathys, Vanessa, Soetaert, Karine, Kiass, Mehdi, Delorme, Vincent, Djaout, Kamel, Trebosc, Vincent, Kemmer, Christian, Wintjens, René, Wohlkönig, Alexandre, Antoine, Rudy, Huot, Ludovic, Hot, David, Coscolla, Mireia, Feldmann, Julia, Gagneux, Sebastien, Locht, Camille, Brodin, Priscille, Gitzinger, Marc, Déprez, Benoit, Willand, Nicolas, Baulard, Alain R.
Published in Science (American Association for the Advancement of Science) (17.03.2017)
Published in Science (American Association for the Advancement of Science) (17.03.2017)
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Journal Article
Front Cover: Synthesis of Substituted Indazole Acetic Acids by N−N Bond Forming Reactions (Eur. J. Org. Chem. 29/2023)
Odell, Luke R., Skillinghaug, Bobo, Matt, Christof, Wu, Peng, Koolmeister, Tobias, Desroses, Matthieu, Llona‐Minguez, Sabin, Wallner, Olov, Helleday, Thomas, Scobie, Martin
Published in European journal of organic chemistry (01.08.2023)
Published in European journal of organic chemistry (01.08.2023)
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Journal Article
A new concise synthesis of 2,3-dihydroquinazolin-4(1H)-one derivatives
Desroses, Matthieu, Scobie, Martin, Helleday, Thomas
Published in New journal of chemistry (01.01.2013)
Published in New journal of chemistry (01.01.2013)
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Journal Article
Synthesis of Substituted Indazole Acetic Acids by N−N Bond Forming Reactions
Odell, Luke R., Skillinghaug, Bobo, Matt, Christof, Wu, Peng, Koolmeister, Tobias, Desroses, Matthieu, Llona‐Minguez, Sabin, Wallner, Olov, Helleday, Thomas, Scobie, Martin
Published in European journal of organic chemistry (01.08.2023)
Published in European journal of organic chemistry (01.08.2023)
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Journal Article
Validating Signal Transducer and Activator of Transcription (STAT) Protein–Inhibitor Interactions Using Biochemical and Cellular Thermal Shift Assays
Attarha, Sanaz, Reithmeier, Anja, Busker, Sander, Desroses, Matthieu, Page, Brent D. G
Published in ACS chemical biology (17.07.2020)
Published in ACS chemical biology (17.07.2020)
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Journal Article
Synthetic EthR inhibitors boost antituberculous activity of ethionamide
Baulard, Alain R, Willand, Nicolas, Dirié, Bertrand, Carette, Xavier, Bifani, Pablo, Singhal, Amit, Desroses, Matthieu, Leroux, Florence, Willery, Eve, Mathys, Vanessa, Déprez-Poulain, Rebecca, Delcroix, Guy, Frénois, Frédéric, Aumercier, Marc, Locht, Camille, Villeret, Vincent, Déprez, Benoit
Published in Nature Medicine (01.05.2009)
Published in Nature Medicine (01.05.2009)
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Journal Article
Magazine Article
NUDT15-mediated hydrolysis limits the efficacy of anti-HCMV drug ganciclovir
Zhang, Si Min, Rehling, Daniel, Jemth, Ann-Sofie, Throup, Adam, Landázuri, Natalia, Almlöf, Ingrid, Göttmann, Mona, Valerie, Nicholas C.K., Borhade, Sanjay R., Wakchaure, Prasad, Page, Brent D.G., Desroses, Matthieu, Homan, Evert J., Scobie, Martin, Rudd, Sean G., Berglund, Ulrika Warpman, Söderberg-Nauclér, Cecilia, Stenmark, Pål, Helleday, Thomas
Published in Cell chemical biology (16.12.2021)
Published in Cell chemical biology (16.12.2021)
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Journal Article
Crystal structures of NUDT15 variants enabled by a potent inhibitor reveal the structural basis for thiopurine sensitivity
Rehling, Daniel, Zhang, Si Min, Jemth, Ann-Sofie, Koolmeister, Tobias, Throup, Adam, Wallner, Olov, Scaletti, Emma, Moriyama, Takaya, Nishii, Rina, Davies, Jonathan, Desroses, Matthieu, Rudd, Sean G., Scobie, Martin, Homan, Evert, Berglund, Ulrika Warpman, Yang, Jun J., Helleday, Thomas, Stenmark, Pål
Published in The Journal of biological chemistry (01.01.2021)
Published in The Journal of biological chemistry (01.01.2021)
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Journal Article
Ethionamide Boosters: Synthesis, Biological Activity, and Structure−Activity Relationships of a Series of 1,2,4-Oxadiazole EthR Inhibitors
Flipo, Marion, Desroses, Matthieu, Lecat-Guillet, Nathalie, Dirié, Bertrand, Carette, Xavier, Leroux, Florence, Piveteau, Catherine, Demirkaya, Fatma, Lens, Zoé, Rucktooa, Prakash, Villeret, Vincent, Christophe, Thierry, Jeon, Hee Kyoung, Locht, Camille, Brodin, Priscille, Déprez, Benoit, Baulard, Alain R, Willand, Nicolas
Published in Journal of medicinal chemistry (28.04.2011)
Published in Journal of medicinal chemistry (28.04.2011)
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Journal Article
Ethionamide Boosters. 2. Combining Bioisosteric Replacement and Structure-Based Drug Design To Solve Pharmacokinetic Issues in a Series of Potent 1,2,4-Oxadiazole EthR Inhibitors
Flipo, Marion, Desroses, Matthieu, Lecat-Guillet, Nathalie, Villemagne, Baptiste, Blondiaux, Nicolas, Leroux, Florence, Piveteau, Catherine, Mathys, Vanessa, Flament, Marie-Pierre, Siepmann, Juergen, Villeret, Vincent, Wohlkönig, Alexandre, Wintjens, René, Soror, Sameh H, Christophe, Thierry, Jeon, Hee Kyoung, Locht, Camille, Brodin, Priscille, Déprez, Benoit, Baulard, Alain R, Willand, Nicolas
Published in Journal of medicinal chemistry (12.01.2012)
Published in Journal of medicinal chemistry (12.01.2012)
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