Phosphinanes and Azaphosphinanes as Potent and Selective Inhibitors of Activated Thrombin-Activatable Fibrinolysis Inhibitor (TAFIa)
Schaffner, Arnaud-Pierre, Sansilvestri-Morel, Patricia, Despaux, Nicole, Ruano, Elisabeth, Persigand, Thierry, Rupin, Alain, Mennecier, Philippe, Vallez, Marie-Odile, Raimbaud, Eric, Desos, Patrice, Gloanec, Philippe
Published in Journal of medicinal chemistry (08.04.2021)
Published in Journal of medicinal chemistry (08.04.2021)
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Improvement in the Selectivity and Metabolic Stability of the Serotonin 5-HT1A Ligand, S 15535: A Series of cis- and trans-2-(Arylcycloalkylamine) 1-Indanols
Peglion, Jean-Louis, Goument, Bertrand, Despaux, Nicole, Charlot, Valérie, Giraud, Hélène, Nisole, Christian, Newman-Tancredi, Adrian, Dekeyne, Anne, Bertrand, Marc, Genissel, Patrick, Millan, Mark J
Published in Journal of medicinal chemistry (03.01.2002)
Published in Journal of medicinal chemistry (03.01.2002)
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Tetracyclic analogues of [+]-S 14297 : Synthesis and determination of affinity and selectivity at cloned human dopamine D3 vs D2 receptors
PEGLION, J.-L, VIAN, J, GOUMENT, B, DESPAUX, N, AUDINOT, V, MILLAN, M. J
Published in Bioorganic & medicinal chemistry letters (08.04.1997)
Published in Bioorganic & medicinal chemistry letters (08.04.1997)
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Improvement in the selectivity and metabolic stability of the serotonin 5-HT(1A) ligand, S 15535: a series of cis- and trans-2-(arylcycloalkylamine) 1-indanols
Peglion, Jean-Louis, Goument, Bertrand, Despaux, Nicole, Charlot, Valérie, Giraud, Hélène, Nisole, Christian, Newman-Tancredi, Adrian, Dekeyne, Anne, Bertrand, Marc, Genissel, Patrick, Millan, Mark J
Published in Journal of medicinal chemistry (03.01.2002)
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Published in Journal of medicinal chemistry (03.01.2002)
Journal Article
Improvement in the Selectivity and Metabolic Stability of the Serotonin 5-HT 1A Ligand, S 15535: A Series of cis - and trans -2-(Arylcycloalkylamine) 1-Indanols
Peglion, Jean-Louis, Goument, Bertrand, Despaux, Nicole, Charlot, Valérie, Giraud, Hélène, Nisole, Christian, Newman-Tancredi, Adrian, Dekeyne, Anne, Bertrand, Marc, Genissel, Patrick, Millan, Mark J.
Published in Journal of medicinal chemistry (01.01.2002)
Published in Journal of medicinal chemistry (01.01.2002)
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S18327 (1-{2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)piperid-1-yl]ethyl}3-phenyl imidazolin-2-one), a Novel, Potential Antipsychotic Displaying Marked Antagonist Properties at α1- and α2-Adrenergic Receptors: II. Functional Profile and a Multiparametric Comparison with Haloperidol, Clozapine, and 11 Other Antipsychotic Agents
Mark J. Millan, Mauricette Brocco, Jean-Michel Rivet, Valérie Audinot, Adrian Newman-Tancredi, Lisa Maiofiss, Sophie Queriaux, Nicole Despaux, Jean-Louis Peglion, Anne Dekeyne
Published in The Journal of pharmacology and experimental therapeutics (01.01.2000)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.2000)
Journal Article
S18327 (1-{2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)piperid-1-yl]ethyl}3-phenyl imidazolin-2-one), a Novel, Potential Antipsychotic Displaying Marked Antagonist Properties at α1- and α2-Adrenergic Receptors: I. Receptorial, Neurochemical, and Electrophysiological Profile
Mark J. Millan, Alain Gobert, Adrian Newman-Tancredi, Françoise Lejeune, Didier Cussac, Jean-Michel Rivet, Valérie Audinot, Agnès Adhumeau, Mauricette Brocco, Jean-Paul Nicolas, Jean A. Boutin, Nicole Despaux, Jean-Louis Peglion
Published in The Journal of pharmacology and experimental therapeutics (01.01.2000)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.2000)
Journal Article
Tetracyclic analogues of [+]-S 14297: Synthesis and determination of affinity and selectivity at cloned human dopamine D 3 vs D 2 receptors
Peglion, Jean-Louis, Vian, Joël, Goument, Bertrand, Despaux, Nicole, Audinot, Valérie, Millan, Mark J.
Published in Bioorganic & medicinal chemistry letters (1997)
Published in Bioorganic & medicinal chemistry letters (1997)
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Immunoturbidimetric assay of δ aminolevulimc acid dehydratase (ALA D) on a centrifugal fast analyser
Despaux-Pages, Nicole, Comoy, Etienne, Bohuon, Claude, Boudene, Claude
Published in Clinica chimica acta (15.04.1985)
Published in Clinica chimica acta (15.04.1985)
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