A novel DYRK1A (Dual specificity tyrosine phosphorylation‐regulated kinase 1A) inhibitor for the treatment of Alzheimer's disease: effect on Tau and amyloid pathologies in vitro
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Published in Journal of neurochemistry (01.05.2015)
Published in Journal of neurochemistry (01.05.2015)
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Wnt signalling regulates adult hippocampal neurogenesis
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Published in Nature (27.10.2005)
Published in Nature (27.10.2005)
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DYRK1A controls the transition from proliferation to quiescence during lymphoid development by destabilizing Cyclin D3
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Published in The Journal of experimental medicine (01.06.2015)
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Etazolate, a neuroprotective drug linking GABAA receptor pharmacology to amyloid precursor protein processing
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Published in Journal of neurochemistry (01.07.2008)
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Inhibition of the Rho GTPase, Rac1, decreases estrogen receptor levels and is a novel therapeutic strategy in breast cancer
Rosenblatt, Adena E, Garcia, Maria Ines, Lyons, Leah, Xie, Yingqiu, Maiorino, Carol, Désiré, Laurent, Slingerland, Joyce, Burnstein, Kerry L
Published in Endocrine-related cancer (01.04.2011)
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RAC1 Inhibition Targets Amyloid Precursor Protein Processing by γ-Secretase and Decreases Aβ Production in Vitro and in Vivo
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Published in The Journal of biological chemistry (11.11.2005)
Published in The Journal of biological chemistry (11.11.2005)
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An Unusual Binding Model of the Methyl 9‑Anilinothiazolo[5,4‑f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases
Chaikuad, Apirat, Diharce, Julien, Schröder, Martin, Foucourt, Alicia, Leblond, Bertrand, Casagrande, Anne-Sophie, Désiré, Laurent, Bonnet, Pascal, Knapp, Stefan, Besson, Thierry
Published in Journal of medicinal chemistry (23.11.2016)
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Design and synthesis of thiazolo[5,4-f]quinazolines as DYRK1A inhibitors, part I
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Published in Molecules (Basel, Switzerland) (29.09.2014)
Published in Molecules (Basel, Switzerland) (29.09.2014)
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Rap1-Rac1 Circuits Potentiate Platelet Activation
Stefanini, Lucia, Boulaftali, Yacine, Ouellette, Timothy D, Holinstat, Michael, Désiré, Laurent, Leblond, Bertrand, Andre, Patrick, Conley, Pamela B, Bergmeier, Wolfgang
Published in Arteriosclerosis, thrombosis, and vascular biology (01.02.2012)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.02.2012)
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Design and synthesis of thiazolo[5,4-f]quinazolines as DYRK1A inhibitors, part II
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Published in Molecules (Basel, Switzerland) (26.09.2014)
Published in Molecules (Basel, Switzerland) (26.09.2014)
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Rare association of thermal burns of the knee and ankle with wounds of the patellar and achilles tendons
Essomba, Laurent Désiré Ndzié, Sanogo, Téredjou Fatou, Moussa, Abdoul Kadri
Published in Burns open : an international open access journal for burn injuries (01.07.2023)
Published in Burns open : an international open access journal for burn injuries (01.07.2023)
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Therapeutic sensitivity to Rac GTPase inhibition requires consequential suppression of mTORC1, AKT, and MEK signaling in breast cancer
Hampsch, Riley A, Shee, Kevin, Bates, Darcy, Lewis, Lionel D, Désiré, Laurent, Leblond, Bertrand, Demidenko, Eugene, Stefan, Kurtis, Huang, Yina H, Miller, Todd W
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Multiplex Antibody Detection for Noninvasive Genus-Level Diagnosis of Prosthetic Joint Infection
Marmor, Simon, Bauer, Thomas, Desplaces, Nicole, Heym, Beate, Roux, Anne-Laure, Sol, Olivier, Rogé, Julie, Mahé, Florence, Désiré, Laurent, Aegerter, Philippe, Ghout, Idir, Ropers, Jacques, Gaillard, Jean-Louis, Rottman, Martin
Published in Journal of clinical microbiology (01.04.2016)
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Validation of AclarusDx™, a blood-based transcriptomic signature for the diagnosis of Alzheimer's disease
Fehlbaum-Beurdeley, Pascale, Sol, Olivier, Désiré, Laurent, Touchon, Jacques, Dantoine, Thierry, Vercelletto, Martine, Gabelle, Audrey, Jarrige, Anne-Charlotte, Haddad, Raphaël, Lemarié, Jean Christophe, Zhou, Weiyin, Hampel, Harald, Einstein, Richard, Vellas, Bruno
Published in Journal of Alzheimer's disease (01.01.2012)
Published in Journal of Alzheimer's disease (01.01.2012)
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A Novel Immersive Anatomy Education System (Anat_Hub): Redefining Blended Learning for the Musculoskeletal System
Boomgaard, Ayesha, Fritz, Kaylyn A., Isafiade, Omowunmi E., Kotze, Retha Christina M., Ekpo, Okobi, Smith, Marjorie, Gessler, Tyler, Filton, Kayleigh J., Cupido, Christiaan C., Aden, Bahija, Yokwe, Ntokozo, Mayekiso, Luyanda, Gxowa, Siyamthanda, Levitt, Annelize, Dlodlo, Lilitha, Madushana, Nosicelo, de Laroche Souvestre, Desiré Laurent
Published in Applied sciences (03.06.2022)
Published in Applied sciences (03.06.2022)
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Blood transcriptomic biomarkers of Alzheimer's disease patients treated with EHT 0202
Désiré, Laurent, Blondiaux, Elodie, Carrière, Jennifer, Haddad, Raphael, Sol, Olivier, Fehlbaum-Beurdeley, Pascale, Einstein, Rich, Zhou, Weiyin, Pando, Matthew P
Published in Journal of Alzheimer's disease (01.01.2013)
Published in Journal of Alzheimer's disease (01.01.2013)
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