Interactions between Penicillin-Binding Proteins (PBPs) and Two Novel Classes of PBP Inhibitors, Arylalkylidene Rhodanines and Arylalkylidene Iminothiazolidin-4-ones
ZERVOSEN, Astrid, LU, Wei-Ping, ZHOULIANG CHEN, WHITE, Ronald E, DEMUTH, Thomas P, FRERE, Jean-Marie
Published in Antimicrobial Agents and Chemotherapy (01.03.2004)
Published in Antimicrobial Agents and Chemotherapy (01.03.2004)
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Design and synthesis of novel N-sulfonyl-2-indole carboxamides as potent PPAR-γ binding agents with potential application to the treatment of osteoporosis
Hopkins, Corey R., O’Neil, Steven V., Laufersweiler, Michael C., Wang, Yili, Pokross, Matthew, Mekel, Marlene, Evdokimov, Artem, Walter, Richard, Kontoyianni, Maria, Petrey, Maria E., Sabatakos, Georgios, Roesgen, Jeff T., Richardson, Eloise, Demuth, Thomas P.
Published in Bioorganic & medicinal chemistry letters (01.11.2006)
Published in Bioorganic & medicinal chemistry letters (01.11.2006)
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Development of a screening assay to measure the loss of antibacterial activity in the presence of proteins: its use in optimizing compound structure
Roychoudhury, Siddhartha, Brill, Jessica L, Lu, Wei-Ping, White, Ronald E, Chen, Zhuoliang, Demuth, Jr, Thomas P
Published in Journal of biomolecular screening (01.10.2003)
Published in Journal of biomolecular screening (01.10.2003)
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Synthesis and evaluation of unsaturated caprolactams as interleukin-1β converting enzyme (ICE) inhibitors
Wang, Yili, O’Neil, Steven V., Wos, John A., Oppong, Kofi A., Laufersweiler, Michael C., Soper, David L., Ellis, Christopher D., Baize, Mark W., Fancher, Amy N., Lu, Wei, Suchanek, Maureen K., Wang, Richard L., Schwecke, William P., Cruze, Charles A., Buchalova, Maria, Belkin, Marina, De, Biswanath, Demuth, Thomas P.
Published in Bioorganic & medicinal chemistry (01.02.2007)
Published in Bioorganic & medicinal chemistry (01.02.2007)
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Synthesis and evaluation of thiazepines as interleukin-1β converting enzyme (ICE) inhibitors
Ellis, Christopher D., Oppong, Kofi A., Laufersweiler, Michael C., O’Neil, Steven V., Soper, David L., Wang, Yili, Wos, John A., Fancher, Amy N., Lu, Wei, Suchanek, Maureen K., Wang, Richard L., De, Biswanath, Demuth, Thomas P.
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
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Synthesis and evaluation of novel 8,5-fused bicyclic peptidomimetic compounds as interleukin-1β converting enzyme (ICE) inhibitors
Soper, David L., Sheville, Justin X., O’Neil, Steven V., Wang, Yili, Laufersweiler, Michael C., Oppong, Kofi A., Wos, John A., Ellis, Christopher D., Baize, Mark W., Chen, Jack J., Fancher, Amy N., Lu, Wei, Suchanek, Maureen K., Wang, Richard L., Schwecke, William P., Cruze, Charles A., Buchalova, Maria, Belkin, Marina, Wireko, Fred, Ritter, Amanda, De, Biswanath, Wang, Difei, Demuth, Thomas P.
Published in Bioorganic & medicinal chemistry (01.12.2006)
Published in Bioorganic & medicinal chemistry (01.12.2006)
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Discovery of novel conformationally restricted diazocan peptidomimetics as inhibitors of interleukin-1β synthesis
Oppong, Kofi A., Ellis, Christopher D., Laufersweiler, Michael C., O’Neil, Steven V., Wang, Yili, Soper, David L., Baize, Mark W., Wos, John A., De, Biswanath, Bosch, Gregory K., Fancher, Amy N., Lu, Wei, Suchanek, Maureen K., Wang, Richard L., Demuth, Thomas P.
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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Synthesis and evaluation of novel 8,6-fused bicyclic peptidomimetic compounds as interleukin-1β converting enzyme inhibitors
O’Neil, Steven V., Wang, Yili, Laufersweiler, Michael C., Oppong, Kofi A., Soper, David L., Wos, John A., Ellis, Christopher D., Baize, Mark W., Bosch, Gregory K., Fancher, Amy N., Lu, Wei, Suchanek, Maureen K., Wang, Richard L., De, Biswanath, Demuth, Thomas P.
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
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Synthesis and evaluation of novel 1-(2-acylhydrazinocarbonyl)-cycloalkyl carboxamides as interleukin-1β converting enzyme (ICE) inhibitors
Soper, David L., Sheville, Justin, O’Neil, Steven V., Wang, Yili, Laufersweiler, Michael C., Oppong, Kofi A., Wos, John A., Ellis, Christopher D., Fancher, Amy N., Lu, Wei, Suchanek, Maureen K., Wang, Richard L., De, Biswanath, Demuth, Thomas P.
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
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Preparation and Antimicrobial Assessment of 2-Thioether-linked Quinolonyl-carbapenems
HERSHBERGER, PAUL M., SWITZER, A. GREG, YELM, KENNETH E., COLEMAN, MILT C., DEVRIES, CAROL A., ROURKE, F. JAMES, DAVIS, BARB W., KRAFT, WILLIAM G., TWINEM, TRACY L., KOENIGS, PAULA M., PAULE, SUZANNE M., SIEHNEL, RICHARD J., ZOUTENDAM, PAUL H., IMBUS, REBECCA, DEMUTH, THOMAS P. Jr
Published in Journal of antibiotics (1998)
Published in Journal of antibiotics (1998)
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Stereoselective synthesis and antibacterial evaluation of 4-amido-isothiazolidinone oxides
Chen, Zhuoliang, Demuth, Thomas P, Wireko, Fred C
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Synthesis and evaluation of tricyclic pyrrolopyrimidinones as dipeptide mimetics: Inhibition of interleukin-1β-converting enzyme
Laufersweiler, Michael C., Wang, Yili, Soper, David L., Suchanek, Maureen K., Fancher, Amy N., Lu, Wei, Wang, Richard L., Oppong, Kofi A., Ellis, Christopher D., Baize, Mark W., O’Neil, Steven V., Wos, John A., Demuth, Thomas P.
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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Journal Article
Synthesis and evaluation of thiazepines as interleukin-1beta converting enzyme (ICE) inhibitors
Ellis, Christopher D, Oppong, Kofi A, Laufersweiler, Michael C, O'Neil, Steven V, Soper, David L, Wang, Yili, Wos, John A, Fancher, Amy N, Lu, Wei, Suchanek, Maureen K, Wang, Richard L, De, Biswanath, Demuth, Jr, Thomas P
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
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Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Journal Article
Synthesis and evaluation of unsaturated caprolactams as interleukin-1beta converting enzyme (ICE) inhibitors
Wang, Yili, O'Neil, Steven V, Wos, John A, Oppong, Kofi A, Laufersweiler, Michael C, Soper, David L, Ellis, Christopher D, Baize, Mark W, Fancher, Amy N, Lu, Wei, Suchanek, Maureen K, Wang, Richard L, Schwecke, William P, Cruze, Charles A, Buchalova, Maria, Belkin, Marina, De, Biswanath, Demuth, Jr, Thomas P
Published in Bioorganic & medicinal chemistry (01.02.2007)
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Published in Bioorganic & medicinal chemistry (01.02.2007)
Journal Article
Synthesis and evaluation of novel 8,5-fused bicyclic peptidomimetic compounds as interleukin-1beta converting enzyme (ICE) inhibitors
Soper, David L, Sheville, Justin X, O'Neil, Steven V, Wang, Yili, Laufersweiler, Michael C, Oppong, Kofi A, Wos, John A, Ellis, Christopher D, Baize, Mark W, Chen, Jack J, Fancher, Amy N, Lu, Wei, Suchanek, Maureen K, Wang, Richard L, Schwecke, William P, Cruze, Charles A, Buchalova, Maria, Belkin, Marina, Wireko, Fred, Ritter, Amanda, De, Biswanath, Wang, Difei, Demuth, Jr, Thomas P
Published in Bioorganic & medicinal chemistry (01.12.2006)
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Published in Bioorganic & medicinal chemistry (01.12.2006)
Journal Article
Synthesis and evaluation of tricyclic pyrrolopyrimidinones as dipeptide mimetics: inhibition of interleukin-1beta-converting enzyme
Laufersweiler, Michael C, Wang, Yili, Soper, David L, Suchanek, Maureen K, Fancher, Amy N, Lu, Wei, Wang, Richard L, Oppong, Kofi A, Ellis, Christopher D, Baize, Mark W, O'Neil, Steven V, Wos, John A, Demuth, Jr, Thomas P
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Journal Article
Synthesis and evaluation of novel 1-(2-acylhydrazinocarbonyl)-cycloalkyl carboxamides as interleukin-1beta converting enzyme (ICE) inhibitors
Soper, David L, Sheville, Justin, O'Neil, Steven V, Wang, Yili, Laufersweiler, Michael C, Oppong, Kofi A, Wos, John A, Ellis, Christopher D, Fancher, Amy N, Lu, Wei, Suchanek, Maureen K, Wang, Richard L, De, Biswanath, Demuth, Jr, Thomas P
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
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Published in Bioorganic & medicinal chemistry letters (15.08.2006)
Journal Article
Synthesis and evaluation of novel 8,6-fused bicyclic peptidomimetic compounds as interleukin-1beta converting enzyme inhibitors
O'Neil, Steven V, Wang, Yili, Laufersweiler, Michael C, Oppong, Kofi A, Soper, David L, Wos, John A, Ellis, Christopher D, Baize, Mark W, Bosch, Gregory K, Fancher, Amy N, Lu, Wei, Suchanek, Maureen K, Wang, Richard L, De, Biswanath, Demuth, Jr, Thomas P
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
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Published in Bioorganic & medicinal chemistry letters (15.12.2005)
Journal Article
Discovery of novel conformationally restricted diazocan peptidomimetics as inhibitors of interleukin-1beta synthesis
Oppong, Kofi A, Ellis, Christopher D, Laufersweiler, Michael C, O'Neil, Steven V, Wang, Yili, Soper, David L, Baize, Mark W, Wos, John A, De, Biswanath, Bosch, Gregory K, Fancher, Amy N, Lu, Wei, Suchanek, Maureen K, Wang, Richard L, Demuth, Jr, Thomas P
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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