Inhaled mosliciguat (BAY 1237592): targeting pulmonary vasculature via activating apo-sGC
Becker-Pelster, Eva M., Hahn, Michael G., Delbeck, Martina, Dietz, Lisa, Hüser, Jörg, Kopf, Johannes, Kraemer, Thomas, Marquardt, Tobias, Mondritzki, Thomas, Nagelschmitz, Johannes, Nikkho, Sylvia M., Pires, Philippe V., Tinel, Hanna, Weimann, Gerrit, Wunder, Frank, Sandner, Peter, Schuhmacher, Joachim, Stasch, Johannes-Peter, Truebel, Hubert K. F.
Published in Respiratory research (01.10.2022)
Published in Respiratory research (01.10.2022)
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Journal Article
A role for coagulation factor Xa in experimental pulmonary arterial hypertension
Delbeck, Martina, Nickel, Katrin F., Perzborn, Elisabeth, Ellinghaus, Peter, Strassburger, Julia, Kast, Raimund, Laux, Volker, Schäfer, Stefan, Schermuly, Ralph T., von Degenfeld, Georges
Published in Cardiovascular research (01.10.2011)
Published in Cardiovascular research (01.10.2011)
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Journal Article
Finerenone, a novel selective nonsteroidal mineralocorticoid receptor antagonist protects from rat cardiorenal injury
Kolkhof, Peter, Delbeck, Martina, Kretschmer, Axel, Steinke, Wolfram, Hartmann, Elke, Bärfacker, Lars, Eitner, Frank, Albrecht-Küpper, Barbara, Schäfer, Stefan
Published in Journal of cardiovascular pharmacology (01.07.2014)
Published in Journal of cardiovascular pharmacology (01.07.2014)
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Journal Article
Topical Potassium Channel Blockage Improves Pharyngeal Collapsibility
Osman, Amal M., Mukherjee, Sutapa, Altree, Thomas J., Delbeck, Martina, Gehring, Doris, Hahn, Michael, Lang, Tina, Xing, Charles, Muller, Thomas, Weimann, Gerrit, Eckert, Danny J.
Published in Chest (01.04.2023)
Published in Chest (01.04.2023)
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Journal Article
Topical Potassium Channel Blockage Improves Pharyngeal Collapsibility: A Translational, Placebo-Controlled Trial
Osman, Amal M, Mukherjee, Sutapa, Altree, Thomas J, Delbeck, Martina, Gehring, Doris, Hahn, Michael, Lang, Tina, Xing, Charles, Muller, Thomas, Weimann, Gerrit, Eckert, Danny J
Published in Chest (01.04.2023)
Published in Chest (01.04.2023)
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Journal Article
A novel TASK channel antagonist nasal spray reduces sleep apnea severity in physiological responders: a randomized, blinded, trial
Osman, Amal M, Toson, Barbara, Naik, Ganesh R, Mukherjee, Sutapa, Delbeck, Martina, Hahn, Michael, Muller, Thomas, Weimann, Gerrit, Eckert, Danny J
Published in American journal of physiology. Heart and circulatory physiology (01.03.2024)
Published in American journal of physiology. Heart and circulatory physiology (01.03.2024)
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Journal Article
A critical review of fundamental controversies in the field of GPR30 research
Langer, Gernot, Bader, Benjamin, Meoli, Luca, Isensee, Jörg, Delbeck, Martina, Noppinger, Patricia Ruiz, Otto, Christiane
Published in Steroids (01.08.2010)
Published in Steroids (01.08.2010)
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Journal Article
Conference Proceeding
Novel non-xanthine antagonist of the A(2B) adenosine receptor: From HTS hit to lead structure
Haerter, Michael, Kalthof, Bernd, Delbeck, Martina, Lustig, Klemens, Gerisch, Michael, Schulz, Simone, Kast, Raimund, Meibom, Daniel, Lindner, Niels
Published in European journal of medicinal chemistry (01.02.2019)
Published in European journal of medicinal chemistry (01.02.2019)
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Journal Article
A lower X-gate in TASK channels traps inhibitors within the vestibule
Rödström, Karin E J, Kiper, Aytuğ K, Zhang, Wei, Rinné, Susanne, Pike, Ashley C W, Goldstein, Matthias, Conrad, Linus J, Delbeck, Martina, Hahn, Michael G, Meier, Heinrich, Platzk, Magdalena, Quigley, Andrew, Speedman, David, Shrestha, Leela, Mukhopadhyay, Shubhashish M M, Burgess-Brown, Nicola A, Tucker, Stephen J, Müller, Thomas, Decher, Niels, Carpenter, Elisabeth P
Published in Nature (London) (18.06.2020)
Published in Nature (London) (18.06.2020)
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Journal Article
Novel non-xanthine antagonist of the A2B adenosine receptor: From HTS hit to lead structure
Härter, Michael, Kalthof, Bernd, Delbeck, Martina, Lustig, Klemens, Gerisch, Michael, Schulz, Simone, Kast, Raimund, Meibom, Daniel, Lindner, Niels
Published in European journal of medicinal chemistry (01.02.2019)
Published in European journal of medicinal chemistry (01.02.2019)
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Journal Article
Vascular Protection and Decongestion Without Renin-Angiotensin-Aldosterone System Stimulation Mediated by a Novel Dual-Acting Vasopressin V1a/V2 Receptor Antagonist
Kolkhof, Peter, Pook, Elisabeth, Pavkovic, Mira, Kretschmer, Axel, Buchmüller, Anja, Tinel, Hanna, Delbeck, Martina, Mondritzki, Thomas, Wasnaire, Pierre, Dinh, Wilfried, Truebel, Hubert, Hüser, Jörg, Schmeck, Carsten
Published in Journal of cardiovascular pharmacology (01.07.2019)
Published in Journal of cardiovascular pharmacology (01.07.2019)
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Journal Article
Freezing the Bioactive Conformation to Boost Potency: The Identification of BAY85-8501, a Selective and Potent Inhibitor of Human Neutrophil Elastase for Pulmonary Diseases
von Nussbaum, Franz, Li, Volkhart M. -J., Allerheiligen, Swen, Anlauf, Sonja, Baerfacker, Lars, Bechem, Martin, Delbeck, Martina, Fitzgerald, Mary F., Gerisch, Michael, Gielen-Haertwig, Heike, Haning, Helmut, Karthaus, Dagmar, Lang, Dieter, Lustig, Klemens, Meibom, Daniel, Mittendorf, Joachim, Rosentreter, Ulrich, Schaefer, Martina, Schaefer, Stefan, Schamberger, Jens, Telan, Leila A., Tersteegen, Adrian
Published in ChemMedChem (01.07.2015)
Published in ChemMedChem (01.07.2015)
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Journal Article
Potent and Selective Human Neutrophil Elastase Inhibitors with Novel Equatorial Ring Topology: in vivo Efficacy of the Polar Pyrimidopyridazine BAY-8040 in a Pulmonary Arterial Hypertension Rat Model
von Nussbaum, Franz, Li, Volkhart M., Meibom, Daniel, Anlauf, Sonja, Bechem, Martin, Delbeck, Martina, Gerisch, Michael, Harrenga, Axel, Karthaus, Dagmar, Lang, Dieter, Lustig, Klemens, Mittendorf, Joachim, Schäfer, Martina, Schäfer, Stefan, Schamberger, Jens
Published in ChemMedChem (19.01.2016)
Published in ChemMedChem (19.01.2016)
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Journal Article
아드레날린수용체 ADRAC2의 억제제
DELBECK MARTINA, DIETZ LISA, BUCHGRABER PHILIPP, MEIBOM DANIEL, PLATZK MAGDALENA, BECKER PELSTER EVA MARIA, HAHN MICHAEL, MUELLER THOMAS, SCHMECK CARSTEN, LINDNER NIELS
Year of Publication 11.07.2022
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Year of Publication 11.07.2022
Patent
Novel non-xanthine antagonist of the A 2B adenosine receptor: From HTS hit to lead structure
Härter, Michael, Kalthof, Bernd, Delbeck, Martina, Lustig, Klemens, Gerisch, Michael, Schulz, Simone, Kast, Raimund, Meibom, Daniel, Lindner, Niels
Published in European journal of medicinal chemistry (20.11.2018)
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Published in European journal of medicinal chemistry (20.11.2018)
Journal Article
N3-시클릭 치환된 티에노우라실 및 그의 용도
DELBECK MARTINA, KOSEMUND DIRK, KALTHOF BERND, SUESSMEIER FRANK, LUSTIG KLEMENS, HAERTER MICHAEL, CANCHO GRANDE YOLANDA
Year of Publication 17.05.2019
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Year of Publication 17.05.2019
Patent
TASK-1 및 TASK-3 채널 억제제를 함유하는 제약 투여 형태, 및 호흡 장애 요법에서의 그의 용도
ANLAHR JOHANNA, DELBECK MARTINA, NICOLAI JANINE, BECK BROICHSITTER MORITZ, ROSENSTEIN BJOERN, GEHRING DORIS, HAHN MICHAEL, ALBUS UDO
Year of Publication 26.08.2019
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Year of Publication 26.08.2019
Patent