Biarylaniline phenethanolamines as potent and selective beta(3) adrenergic receptor agonists
Uehling, DE, Shearer, BG, Donaldson, KH, Chao, EY, Deaton, DN, Adkison, KK, Brown, KK, Cariello, NF, Faison, WL, Lancaster, ME, Lin, J, Hart, R, Milliken, TO, Paulik, MA, Sherman, BW, Sugg, EE, Cowan, C
Published in Journal of medicinal chemistry (04.05.2006)
Published in Journal of medicinal chemistry (04.05.2006)
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Design of Potent, Selective, and Orally Bioavailable Inhibitors of Cysteine Protease Cathepsin K
Tavares, Francis X, Boncek, Virginia, Deaton, David N, Hassell, Anne M, Long, Stacey T, Miller, Aaron B, Payne, Alan A, Miller, Larry R, Shewchuk, Lisa M, Wells-Knecht, Kevin, Willard, Derril H, Wright, Lois L, Zhou, Hui-Qiang
Published in Journal of medicinal chemistry (29.01.2004)
Published in Journal of medicinal chemistry (29.01.2004)
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Novel and potent cyclic cyanamide-based cathepsin K inhibitors
Deaton, David N., Hassell, Anne M., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Shewchuk, Lisa M., Tavares, Francis X., Willard, Derril H., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (01.04.2005)
Published in Bioorganic & medicinal chemistry letters (01.04.2005)
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Potent and Selective Ketoamide-Based Inhibitors of Cysteine Protease, Cathepsin K
Tavares, Francis X, Deaton, David N, Miller, Aaron B, Miller, Larry R, Wright, Lois L, Zhou, Hui-Qiang
Published in Journal of medicinal chemistry (07.10.2004)
Published in Journal of medicinal chemistry (07.10.2004)
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Ketoamide-Based Inhibitors of Cysteine Protease, Cathepsin K: P3 Modifications
Tavares, Francis X, Deaton, David N, Miller, Larry R, Wright, Lois L
Published in Journal of medicinal chemistry (07.10.2004)
Published in Journal of medicinal chemistry (07.10.2004)
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P 2–P 3 conformationally constrained ketoamide-based inhibitors of cathepsin K
Barrett, David G., Boncek, Virginia M., Catalano, John G., Deaton, David N., Hassell, Anne M., Jurgensen, Cynthia H., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Payne, J. Alan, Ray, John A., Samano, Vicente, Shewchuk, Lisa M., Tavares, Francis X., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L., Zhou, Hui-Qiang Q.
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
Published in Bioorganic & medicinal chemistry letters (01.08.2005)
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Potent and selective P 2–P 3 ketoamide inhibitors of cathepsin K with good pharmacokinetic properties via favorable P 1′, P 1, and/or P 3 substitutions
Barrett, David G., Catalano, John G., Deaton, David N., Hassell, Anne M., Long, Stacey T., Miller, Aaron B., Miller, Larry R., Shewchuk, Lisa M., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (04.10.2004)
Published in Bioorganic & medicinal chemistry letters (04.10.2004)
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Acyclic cyanamide-based inhibitors of cathepsin K
Barrett, David G., Deaton, David N., Hassell, Anne M., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Payne, J. Alan, Shewchuk, Lisa M., Willard, Derril H., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (15.06.2005)
Published in Bioorganic & medicinal chemistry letters (15.06.2005)
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Synthesis and evaluation of potent and selective beta(3) adrenergic receptor agonists containing acylsulfonamide, sulfonylsulfonamide, and sulfonylurea carboxylic acid isosteres
Uehling, DE, Donaldson, KH, Deaton, DN, Hyman, CE, Sugg, EE, Barrett, DG, Hughes, RG, Reitter, B, Adkison, KK, Lancaster, ME, Lee, F, Hart, R, Paulik, MA, Sherman, BW, True, T, Cowan, C
Published in Journal of medicinal chemistry (31.01.2002)
Published in Journal of medicinal chemistry (31.01.2002)
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Design of small molecule ketoamide-based inhibitors of cathepsin K
Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Larry R., Payne, J.Alan, Wells-Knecht, Kevin J., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
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A structural screening approach to ketoamide-based inhibitors of cathepsin K
Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Wells-Knecht, Kevin J., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
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Semicarbazone-based inhibitors of cathepsin K, are they prodrugs for aldehyde inhibitors?
Adkison, Kim K., Barrett, David G., Deaton, David N., Gampe, Robert T., Hassell, Anne M., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Payne, J. Alan, Shewchuk, Lisa M., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L.
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
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Orally bioavailable small molecule ketoamide-based inhibitors of cathepsin K
Barrett, David G., Catalano, John G., Deaton, David N., Long, Stacey T., Miller, Larry R., Tavares, Francis X., Wells-Knecht, Kevin J., Wright, Lois L., Zhou, Hui-Qiang Q.
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
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MATRIX METALLOPROTEINASE INHIBITORS CONTAINING A (CARBOXYALKYL)AMINO ZINC LIGAND - MODIFICATION OF THE P1 AND P2' RESIDUES
BROWN, FK, BROWN, PJ, BICKETT, DM, CHAMBERS, CL, DAVIES, HG, DEATON, DN, DREWRY, D, FOLEY, M, MCELROY, AB, GREGSON, M, MCGEEHAN, GM, MYERS, PL, NORTON, D, SALOVICH, JM, SCHOENEN, FJ, WARD, P
Published in Journal of medicinal chemistry (04.03.1994)
Published in Journal of medicinal chemistry (04.03.1994)
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Effect of matrix metalloproteinase inhibitors on tumor growth and spontaneous metastasis
Conway, J G, Trexler, S J, Wakefield, J A, Marron, B E, Emerson, D L, Bickett, D M, Deaton, D N, Garrison, D, Elder, M, McElroy, A, Willmott, N, Dockerty, A J, McGeehan, G M
Published in Clinical & experimental metastasis (01.03.1996)
Published in Clinical & experimental metastasis (01.03.1996)
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STEREOCONTROLLED ONE-POT CONVERSIONS OF ALPHA-ALKOXY ESTERS TO SYN-1,2-DIOL AND ANTI-1,2-DIOL DERIVATIVES
BURKE, SD, DEATON, DN, OLSEN, RJ, ARMISTEAD, DM, BLOUGH, BE
Published in Tetrahedron letters (01.01.1987)
Published in Tetrahedron letters (01.01.1987)
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Studies directed toward the total synthesis of cerorubenic acid-III. 3. A convergent enantioselective approach involving new arrangements for the actuation of ring D cyclization
Paquette, Leo A, Deaton, David N, Endo, Yasuyuki, Poupart, Marc Andre
Published in Journal of organic chemistry (01.07.1993)
Published in Journal of organic chemistry (01.07.1993)
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