UNITE4TB: a new consortium for clinical drug and regimen development for TB
Boeree, M. J., Lange, C., Thwaites, G., Paton, N., de Vrueh, R., Barros, D., Hoelscher, M., on behalf of the UNITE4TB Consortium
Published in The international journal of tuberculosis and lung disease (01.11.2021)
Published in The international journal of tuberculosis and lung disease (01.11.2021)
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Novel hepatotrophic prodrugs of the antiviral nucleoside 9-(2-phosphonylmethoxyethyl)adenine with improved pharmacokinetics and antiviral activity
Biessen, E A, Valentijn, A R, De Vrueh, R L, Van De Bilt, E, Sliedregt, L A, Prince, P, Bijsterbosch, M K, Van Boom, J H, Van Der Marel, G A, Abrahams, P J, Van Berkel, T J
Published in The FASEB journal (01.09.2000)
Published in The FASEB journal (01.09.2000)
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5'-Amino acid esters of antiviral nucleosides, acyclovir, and AZT are absorbed by the intestinal PEPT1 peptide transporter
HAN, H.-K, DE VRUEH, R. L. A, RHIE, J. K, COVITZ, K.-M. Y, SMITH, P. L, LEE, C.-P, OH, D.-M, SADEE, W, AMIDON, G. L
Published in Pharmaceutical research (01.08.1998)
Published in Pharmaceutical research (01.08.1998)
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Preclinical and Clinical In Vitro In Vivo Correlation of an hGH Dextran Microsphere Formulation
VLUGT-WENSINK, K. D. F, DE VRUEH, R, GRESNIGT, M. G, HOOGERBRUGGE, C. M, VAN BUUL-OFFERS, S. C, DE LEEDE, L. G. J, STERKMAN, L. G. W, CROMMELIN, D. J. A, HENNINK, W. E, VERRIJK, R
Published in Pharmaceutical research (01.12.2007)
Published in Pharmaceutical research (01.12.2007)
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Carrier-Mediated Delivery of 9-(2-Phosphonylmethoxyethyl)Adenine to Parenchymal Liver Cells: a Novel Therapeutic Approach for Hepatitis B
DE VRUEH, R. L. A, RUMP, E. T, VAN DE BILT, E, VAN VEGHEL, R, BALZARINI, J, BIESSEN, E. A. L, VAN BERKEL, T. J. C, BIJSTERBOSCH, M. K
Published in Antimicrobial Agents and Chemotherapy (01.03.2000)
Published in Antimicrobial Agents and Chemotherapy (01.03.2000)
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Synthesis of a lipophilic prodrug of 9-(2-phosphonylmethoxyethyl)adenine (PMEA) and its incorporation into a hepatocyte-specific lipidic carrier
DE VRUEH, R. L. A, RUMP, E. T, SLIEDREGT, L. A. J. M, BIESSEN, E. A. L, VAN BERKEL, T. J. C, BIJSTERBOSCH, M. K
Published in Pharmaceutical research (01.08.1999)
Published in Pharmaceutical research (01.08.1999)
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In vivo fate of phosphorothioate antisense oligodeoxynucleotides: predominant uptake by scavenger receptors on endothelial liver cells
Bijsterbosch, Martin K., Manoharan, Muthiah, Rump, Erik T., De Vrueh, Remco L. A., van Veghel, Richard, Tivel, Kathleen L., Biessen, Erik A. L., Bennett, C. Frank, Cook, P. Dan, van Berkel, Theo J. C.
Published in Nucleic acids research (15.08.1997)
Published in Nucleic acids research (15.08.1997)
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Modulation of plasma protein binding and in vivo liver cell uptake of phosphorothioate oligodeoxynucleotides by cholesterol conjugation
Bijsterbosch, M K, Rump, E T, De Vrueh, R L, Dorland, R, van Veghel, R, Tivel, K L, Biessen, E A, van Berkel, T J, Manoharan, M
Published in Nucleic acids research (15.07.2000)
Published in Nucleic acids research (15.07.2000)
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Preparation of Conjugates of Oligodeoxynucleotides and Lipid Structures and Their Interaction with Low-Density Lipoprotein
Rump, Erik T, de Vrueh, Remco L. A, Sliedregt, Leo A. J. M, Biessen, Erik A. L, van Berkel, Theo J. C, Bijsterbosch, Martin K
Published in Bioconjugate chemistry (01.05.1998)
Published in Bioconjugate chemistry (01.05.1998)
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Modification of the plasma clearance and liver uptake of steroid ester-conjugated oligodeoxynucleotides by association with (lactosylated) low-density lipoprotein
Rump, Erik T, de Vrueh, Remco L.A, Manoharan, Muthiah, Waarlo, Ingrid H.E, van Veghel, Richard, Biessen, Erik A.L, van Berkel, Theo J.C, Bijsterbosch, Martin K
Published in Biochemical pharmacology (01.06.2000)
Published in Biochemical pharmacology (01.06.2000)
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