Microspectrofluorimetry to dissect the permeation of ceftazidime in Gram-negative bacteria
Allam, Anas, Maigre, Laure, Vergalli, Julia, Dumont, Estelle, Cinquin, Bertrand, Alves de Sousa, Rodolphe, Pajovic, Jelena, Pinet, Elizabeth, Smith, Nikaia, Herbeuval, Jean-Philippe, Réfrégiers, Matthieu, Artaud, Isabelle, Pagès, Jean-Marie
Published in Scientific reports (20.04.2017)
Published in Scientific reports (20.04.2017)
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Targeting Degradation of EGFR through the Allosteric Site Leads to Cancer Cell Detachment-Promoted Death
Iradyan, Melkon, Iradyan, Nina, Hulin, Philippe, Hambardzumyan, Artur, Gyulkhandanyan, Aram, Alves de Sousa, Rodolphe, Hessani, Assia, Roussakis, Christos, Bollot, Guillaume, Bauvais, Cyril, Sakanyan, Vehary
Published in Cancers (01.08.2019)
Published in Cancers (01.08.2019)
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Activation of EGFR by small compounds through coupling the generation of hydrogen peroxide to stable dimerization of Cu/Zn SOD1
Sakanyan, Vehary, Hulin, Philippe, Alves de Sousa, Rodolphe, Silva, Viviane A O, Hambardzumyan, Artur, Nedellec, Steven, Tomasoni, Christophe, Logé, Cédric, Pineau, Charles, Roussakis, Christos, Fleury, Fabrice, Artaud, Isabelle
Published in Scientific reports (17.02.2016)
Published in Scientific reports (17.02.2016)
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Discovery and Refinement of a New Structural Class of Potent Peptide Deformylase Inhibitors
Boularot, Adrien, Giglione, Carmela, Petit, Sylvain, Duroc, Yann, Alves de Sousa, Rodolphe, Larue, Valéry, Cresteil, Thierry, Dardel, Frédéric, Artaud, Isabelle, Meinnel, Thierry
Published in Journal of medicinal chemistry (11.01.2007)
Published in Journal of medicinal chemistry (11.01.2007)
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Revisiting the nature and pharmacodynamics of tacrolimus metabolites
Mevizou, Rudy, Aouad, Hassan, Sauvage, François-Ludovic, Arnion, Hélène, Pinault, Emilie, Bernard, Jean-Sébastien, Bertho, Gildas, Giraud, Nicolas, Alves de Sousa, Rodolphe, Lopez-Noriega, Adolfo, Di Meo, Florent, Campana, Mélanie, Marquet, Pierre
Published in Pharmacological research (01.11.2024)
Published in Pharmacological research (01.11.2024)
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Antidepressant efficacy of a selective organic cation transporter blocker in a mouse model of depression
Orrico-Sanchez, Alejandro, Chausset-Boissarie, Laetitia, Alves de Sousa, Rodolphe, Coutens, Basile, Rezai Amin, Sara, Vialou, Vincent, Louis, Franck, Hessani, Assia, Dansette, Patrick M, Zornoza, Teodoro, Gruszczynski, Carole, Giros, Bruno, Guiard, Bruno P, Acher, Francine, Pietrancosta, Nicolas, Gautron, Sophie
Published in Molecular psychiatry (01.06.2020)
Published in Molecular psychiatry (01.06.2020)
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Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition
Hayek, Simon, Pietrancosta, Nicolas, Hovhannisyan, Anna A., de Sousa, Rodolphe Alves, Bekaddour, Nassima, Ermellino, Laura, Tramontano, Enzo, Arnould, Stephanie, Sardet, Claude, Dairou, Julien, Diaz, Olivier, Lotteau, Vincent, Nisole, Sebastien, Melikyan, Gagik, Herbeuval, Jean-Philippe, Vidalain, Pierre-Olivier
Published in European journal of medicinal chemistry (15.01.2020)
Published in European journal of medicinal chemistry (15.01.2020)
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New Inhibitors of Iron-Containing Nitrile Hydratases
Bonnet, Didier, Stevens, Julie M., Sousa, Rodolphe Alves de, Sari, Marie-Agnès, Mansuy, Daniel, Artaud, Isabelle
Published in Journal of biochemistry (Tokyo) (01.08.2001)
Published in Journal of biochemistry (Tokyo) (01.08.2001)
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New amphiphilic neamine conjugates bearing a metal binding motif active against MDR E. aerogenes Gram-negative bacteria
Allam, Anas, Maigre, Laure, Alves de Sousa, Rodolphe, Dumont, Estelle, Vergalli, Julia, Pagès, Jean-Marie, Artaud, Isabelle
Published in European journal of medicinal chemistry (15.02.2017)
Published in European journal of medicinal chemistry (15.02.2017)
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Journal Article
New Peptides with Metal Binding Abilities and Their Use as Drug Carriers
Allam, Anas, Maigre, Laure, Alimi, Mickael, Alves de Sousa, Rodolphe, Hessani, Assia, Galardon, Erwan, Pagès, Jean-Marie, Artaud, Isabelle
Published in Bioconjugate chemistry (15.10.2014)
Published in Bioconjugate chemistry (15.10.2014)
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Corrigendum: A unique peptide deformylase platform to rationally design and challenge novel active compounds
Fieulaine, Sonia, Alves de Sousa, Rodolphe, Maigre, Laure, Hamiche, Karim, Alimi, Mickael, Bolla, Jean-Michel, Taleb, Abbass, Denis, Alexis, Pagès, Jean-Marie, Artaud, Isabelle, Meinnel, Thierry, Giglione, Carmela
Published in Scientific reports (11.01.2017)
Published in Scientific reports (11.01.2017)
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Hydroxamic Acids as Potent Inhibitors of FeII and MnII E. coli Methionine Aminopeptidase: Biological Activities and X-ray Structures of Oxazole Hydroxamate-EcMetAP-Mn Complexes
Huguet, Florian, Melet, Armelle, Alves de Sousa, Rodolphe, Lieutaud, Aurélie, Chevalier, Jacqueline, Maigre, Laure, Deschamps, Patrick, Tomas, Alain, Leulliot, Nicolas, Pages, Jean-Marie, Artaud, Isabelle
Published in ChemMedChem (01.06.2012)
Published in ChemMedChem (01.06.2012)
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New peptide deformylase inhibitors and cooperative interaction: a combination to improve antibacterial activity
GOEMAERE, Emilie, MELET, Armelle, MEINNEL, Thierry, DARDEL, Frederic, ARTAUD, Isabelle, PAGES, Jean-Marie, LARUE, Valéry, LIEUTAUD, Aurélie, DE SOUSA, Rodolphe Alves, CHEVALIER, Jacqueline, YIMGA-DJAPA, Liselotte, GIGLIONE, Carmela, HUGUET, Florian, ALIMI, Mickael
Published in Journal of antimicrobial chemotherapy (01.06.2012)
Published in Journal of antimicrobial chemotherapy (01.06.2012)
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Identification of Primary Natural Killer Cell Modulators by Chemical Library Screening with a Luciferase-Based Functional Assay
Hayek, Simon, Bekaddour, Nassima, Besson, Laurie, Alves de Sousa, Rodolphe, Pietrancosta, Nicolas, Viel, Sébastien, Smith, Nikaia, Jacob, Yves, Nisole, Sébastien, Mandal, Rupasri, Wishart, David S., Walzer, Thierry, Herbeuval, Jean-Philippe, Vidalain, Pierre-Olivier
Published in SLAS discovery (01.01.2019)
Published in SLAS discovery (01.01.2019)
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