The cholesterol-derived metabolite dendrogenin A functionally reprograms breast adenocarcinoma and undifferentiated thyroid cancer cells
Bauriaud-Mallet, Mathilde, Vija-Racaru, Lavinia, Brillouet, Séverine, Mallinger, Arnaud, de Medina, Philippe, Rives, Arnaud, Payre, Bruno, Poirot, Marc, Courbon, Fréderic, Silvente-Poirot, Sandrine
Published in The Journal of steroid biochemistry and molecular biology (01.09.2019)
Published in The Journal of steroid biochemistry and molecular biology (01.09.2019)
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Journal Article
Identification and pharmacological characterization of cholesterol-5,6-epoxide hydrolase as a target for tamoxifen and AEBS ligands
de Medina, Philippe, Paillasse, Michael R., Segala, Gregory, Poirot, Marc, Silvente-Poirot, Sandrine, Mangelsdorf, David J.
Published in Proceedings of the National Academy of Sciences - PNAS (27.07.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (27.07.2010)
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Journal Article
HPLC Analysis and Skin Whitening Effects of Umbelliprenin-containing Extracts of Anethum Graveolens , Pimpinella Anisum , and Ferulago Campestris
Taddeo, Vito Alessandro, Epifano, Francesco, Preziuso, Francesca, Fiorito, Serena, Caron, Nicolas, Rives, Arnaud, de Medina, Philippe, Poirot, Marc, Silvente-Poirot, Sandrine, Genovese, Salvatore
Published in Molecules (Basel, Switzerland) (30.01.2019)
Published in Molecules (Basel, Switzerland) (30.01.2019)
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Journal Article
5,6-Epoxy-cholesterols contribute to the anticancer pharmacology of Tamoxifen in breast cancer cells
Segala, Gregory, de Medina, Philippe, Iuliano, Luigi, Zerbinati, Chiara, Paillasse, Michael R., Noguer, Emmanuel, Dalenc, Florence, Payré, Bruno, Jordan, V. Craig, Record, Michel, Silvente-Poirot, Sandrine, Poirot, Marc
Published in Biochemical pharmacology (01.07.2013)
Published in Biochemical pharmacology (01.07.2013)
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Journal Article
Dendrogenin A Synergizes with Cytarabine to Kill Acute Myeloid Leukemia Cells In Vitro and In Vivo
Serhan, Nizar, Mouchel, Pierre-Luc, de Medina, Philippe, Segala, Gregory, Mougel, Aurélie, Saland, Estelle, Rives, Arnaud, Lamaziere, Antonin, Despres, Gaëtan, Sarry, Jean-Emmanuel, Larrue, Clément, Vergez, François, Largeaud, Laetitia, Record, Michel, Récher, Christian, Silvente-Poirot, Sandrine, Poirot, Marc
Published in Cancers (01.07.2020)
Published in Cancers (01.07.2020)
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Journal Article
Signaling through cholesterol esterification: a new pathway for the cholecystokinin 2 receptor involved in cell growth and invasion
Paillasse, Michael R., de Medina, Philippe, Amouroux, Guillaume, Mhamdi, Loubna, Poirot, Marc, Silvente-Poirot, Sandrine
Published in Journal of lipid research (01.11.2009)
Published in Journal of lipid research (01.11.2009)
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Journal Article
Auraptene is an inhibitor of cholesterol esterification and a modulator of estrogen receptors
de Medina, Philippe, Genovese, Salvatore, Paillasse, Michael R, Mazaheri, Mahta, Caze-Subra, Stephanie, Bystricky, Kerstin, Curini, Massimo, Silvente-Poirot, Sandrine, Epifano, Francesco, Poirot, Marc
Published in Molecular pharmacology (01.11.2010)
Published in Molecular pharmacology (01.11.2010)
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Journal Article
The novel steroidal alkaloids dendrogenin A and B promote proliferation of adult neural stem cells
Khalifa, Shaden A.M., de Medina, Philippe, Erlandsson, Anna, El-Seedi, Hesham R., Silvente-Poirot, Sandrine, Poirot, Marc
Published in Biochemical and biophysical research communications (11.04.2014)
Published in Biochemical and biophysical research communications (11.04.2014)
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Journal Article
Importance of cholesterol and oxysterols metabolism in the pharmacology of tamoxifen and other AEBS ligands
de Medina, Philippe, Paillasse, Michael R., Ségala, Gregory, Khallouki, Farid, Brillouet, Severine, Dalenc, Florence, Courbon, Frederic, Record, Michel, Poirot, Marc, Silvente-Poirot, Sandrine
Published in Chemistry and physics of lipids (01.09.2011)
Published in Chemistry and physics of lipids (01.09.2011)
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Journal Article
Microsomal antiestrogen-binding site ligands induce growth control and differentiation of human breast cancer cells through the modulation of cholesterol metabolism
Payré, Bruno, de Medina, Philippe, Boubekeur, Nadia, Mhamdi, Loubna, Bertrand-Michel, Justine, Tercé, François, Fourquaux, Isabelle, Goudounèche, Dominique, Record, Michel, Poirot, Marc, Silvente-Poirot, Sandrine
Published in Molecular cancer therapeutics (01.12.2008)
Published in Molecular cancer therapeutics (01.12.2008)
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Journal Article
27-Hydroxylation of oncosterone by CYP27A1 switches its activity from pro-tumor to anti-tumor
Ayadi, Silia, Friedrichs, Silvia, Soulès, Regis, Pucheu, Laly, Lütjohann, Dieter, Silvente-Poirot, Sandrine, Poirot, Marc, de Medina, Philippe
Published in Journal of lipid research (01.12.2023)
Published in Journal of lipid research (01.12.2023)
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Journal Article
Tamoxifen Is a Potent Inhibitor of Cholesterol Esterification and Prevents the Formation of Foam Cells
de Medina, Philippe, Payré, Bruno L, Bernad, José, Bosser, Isabelle, Pipy, Bernard, Silvente-Poirot, Sandrine, Favre, Gilles, Faye, Jean-Charles, Poirot, Marc
Published in The Journal of pharmacology and experimental therapeutics (01.03.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2004)
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Journal Article
Exosomes account for vesicle-mediated transcellular transport of activatable phospholipases and prostaglandins[S]
Subra, Caroline, Grand, David, Laulagnier, Karine, Stella, Alexandre, Lambeau, Gérard, Paillasse, Michael, De Medina, Philippe, Monsarrat, Bernard, Perret, Bertrand, Silvente-Poirot, Sandrine, Poirot, Marc, Record, Michel
Published in Journal of lipid research (01.08.2010)
Published in Journal of lipid research (01.08.2010)
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Journal Article
Quantification of biologically active O-prenylated and unprenylated phenylpropanoids in dill (Anethum graveolens), anise (Pimpinella anisum), and wild celery (Angelica archangelica)
Taddeo, Vito Alessandro, Genovese, Salvatore, Medina, Philippe de, Palmisano, Roberta, Epifano, Francesco, Fiorito, Serena
Published in Journal of pharmaceutical and biomedical analysis (05.02.2017)
Published in Journal of pharmaceutical and biomedical analysis (05.02.2017)
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Journal Article
Identification of a tumor-promoter cholesterol metabolite in human breast cancers acting through the glucocorticoid receptor
Voisin, Maud, de Medina, Philippe, Mallinger, Arnaud, Dalenc, Florence, Huc-Claustre, Emilie, Leignadier, Julie, Serhan, Nizar, Soules, Régis, Ségala, Grégory, Mougel, Aurélie, Noguer, Emmanuel, Mhamdi, Loubna, Bacquié, Elodie, Iuliano, Luigi, Zerbinati, Chiara, Lacroix-Triki, Magali, Chaltiel, Léonor, Filleron, Thomas, Cavaillès, Vincent, Saati, Talal Al, Rochaix, Philippe, Duprez-Paumier, Raphaelle, Franchet, Camille, Ligat, Laetitia, Lopez, Fréderic, Record, Michel, Poirot, Marc, Silvente-Poirot, Sandrine
Published in Proceedings of the National Academy of Sciences - PNAS (31.10.2017)
Published in Proceedings of the National Academy of Sciences - PNAS (31.10.2017)
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Journal Article
Dendrogenin A drives LXR to trigger lethal autophagy in cancers
Segala, Gregory, David, Marion, de Medina, Philippe, Poirot, Mathias C., Serhan, Nizar, Vergez, François, Mougel, Aurelie, Saland, Estelle, Carayon, Kevin, Leignadier, Julie, Caron, Nicolas, Voisin, Maud, Cherier, Julia, Ligat, Laetitia, Lopez, Frederic, Noguer, Emmanuel, Rives, Arnaud, Payré, Bruno, Saati, Talal al, Lamaziere, Antonin, Despres, Gaëtan, Lobaccaro, Jean-Marc, Baron, Silvere, Demur, Cecile, de Toni, Fabienne, Larrue, Clément, Boutzen, Helena, Thomas, Fabienne, Sarry, Jean-Emmanuel, Tosolini, Marie, Picard, Didier, Record, Michel, Récher, Christian, Poirot, Marc, Silvente-Poirot, Sandrine
Published in Nature communications (04.12.2017)
Published in Nature communications (04.12.2017)
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Journal Article
From tamoxifen to dendrogenin A: The discovery of a mammalian tumor suppressor and cholesterol metabolite
Silvente-Poirot, Sandrine, de Medina, Philippe, Record, Michel, Poirot, Marc
Published in Biochimie (01.11.2016)
Published in Biochimie (01.11.2016)
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