Characterization of a Novel, Non-peptidyl Antagonist of the Human Glucagon Receptor
Cascieri, M A, Koch, G E, Ber, E, Sadowski, S J, Louizides, D, de Laszlo, S E, Hacker, C, Hagmann, W K, MacCoss, M, Chicchi, G G, Vicario, P P
Published in The Journal of biological chemistry (26.03.1999)
Published in The Journal of biological chemistry (26.03.1999)
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N-(3-Phenylsulfonyl-3-piperidinoyl)-phenylalanine derivatives as potent, selective VLA-4 antagonists
Gutteridge, Clare E, de Laszlo, Stephen E, Kamenecka, Theodore M, McCauley, Ermengilda, van Riper, Gail, Mumford, Richard A, Kidambi, Usha, Egger, Linda A, Tong, Sharon, Hagmann, William K
Published in Bioorganic & medicinal chemistry letters (10.03.2003)
Published in Bioorganic & medicinal chemistry letters (10.03.2003)
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Identification of Unique VLA-4 Antagonists from a Combinatorial Library
de Laszlo, Stephen E., Li, Bing, McCauley, Ermengilda, Van Riper, Gail, Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
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The discovery of sulfonylated dipeptides as Potent VLA-4 antagonists
Hagmann, William K, Durette, Philippe L, Lanza, Thomas, Kevin, Nancy Jo, de Laszlo, Stephen E, Kopka, Ihor E, Young, David, Magriotis, Plato A, Li, Bing, Lin, Linus S, Yang, Ginger, Kamenecka, Theodore, Chang, Linda L, Wilson, Jonathan, MacCoss, Malcolm, Mills, Sander G, Van Riper, Gail, McCauley, Ermengilda, Egger, Linda A, Kidambi, Usha, Lyons, Kathryn, Vincent, Stella, Stearns, Ralph, Colletti, Adria, Teffera, Johannes, Tong, Sharon, Fenyk-Melody, Judy, Owens, Karen, Levorse, Dorothy, Kim, Philip, Schmidt, John A, Mumford, Richard A
Published in Bioorganic & medicinal chemistry letters (22.10.2001)
Published in Bioorganic & medicinal chemistry letters (22.10.2001)
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N-(Arylacetyl)-biphenylalanines as Potent VLA-4 Antagonists
Li, Bing, de Laszlo, Stephen E, Kamenecka, Theodore M, Kopka, Ihor E, Durette, Philippe L, Lanza, Jr, Thomas, MacCoss, Malcolm, Tong, Sharon, Mumford, Richard A, McCauley, Ermengilda D, Van Riper, Gail, Schmidt, John A, Hagmann, William K
Published in Bioorganic & medicinal chemistry letters (19.08.2002)
Published in Bioorganic & medicinal chemistry letters (19.08.2002)
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N-Tetrahydrofuroyl-( l)-phenylalanine derivatives as potent VLA-4 antagonists
Yang, Ginger X., Chang, Linda L., Truong, Quang, Doherty, George A., Magriotis, Plato A., de Laszlo, Stephen E., Li, Bing, MacCoss, Malcolm, Kidambi, Usha, Egger, Linda A., McCauley, Ermengilda, Van Riper, Gail, Mumford, Richard A., Schmidt, John A., Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (03.06.2002)
Published in Bioorganic & medicinal chemistry letters (03.06.2002)
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N-Aryl-prolyl-dipeptides as potent antagonists of VLA-4
Kamenecka, Theodore M., Lanza, Jr, Thomas, de Laszlo, Stephen E., Li, Bing, McCauley, Ermengilda D., Van Riper, Gail, Egger, Linda A., Kidambi, Usha, Mumford, Richard A., Tong, Sharon, MacCoss, Malcolm, Schmidt, John A., Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (19.08.2002)
Published in Bioorganic & medicinal chemistry letters (19.08.2002)
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A potent, orally active, balanced affinity angiotensin II AT1 antagonist and AT2 binding inhibitor
de Laszlo, Stephen E, Quagliato, Carol S, Greenlee, William J, Patchett, Arthur A, Chang, Raymond S. L, Lotti, Victor J, Chen, Tsing Bau, Scheck, Stacey A, Faust, Kristi A
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
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Potent, orally absorbed glucagon receptor antagonists
de Laszlo, Stephen E., Hacker, Candice, Li, Bing, Kim, Dooseop, MacCoss, Malcolm, Mantlo, Nathan, Pivnichny, James V., Colwell, Larry, Koch, Gregory E., Cascieri, Margaret A., Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (08.03.1999)
Published in Bioorganic & medicinal chemistry letters (08.03.1999)
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Substituted Imidazoles as Glucagon Receptor Antagonists
Chang, Linda L., Sidler, Kelly L., Cascieri, Margaret A., de Laszlo, Stephen, Koch, Greg, Li, Bing, MacCoss, Malcolm, Mantlo, Nathan, O'Keefe, Stephen, Pang, Margaret, Rolando, Anna, Hagmann, William K.
Published in Bioorganic & medicinal chemistry letters (17.09.2001)
Published in Bioorganic & medicinal chemistry letters (17.09.2001)
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Pyrroles and other heterocycles as inhibitors of P38 kinase
de Laszlo, Stephen E., Visco, Denise, Agarwal, Lily, Chang, Linda, Chin, Jayne, Croft, Gist, Forsyth, Amy, Fletcher, Daniel, Frantz, Betsy, Hacker, Candice, Hanlon, William, Harper, Coral, Kostura, Matthew, Li, Bing, Luell, Sylvie, MacCoss, Malcolm, Mantlo, Nathan, O'Neill, Edward A., Orevillo, Chad, Pang, Margaret, Parsons, Janey, Rolando, Anna, Sahly, Yousif, Sidler, Kelley, Widmer, W.Rick, O'Keefe, Stephen J.
Published in Bioorganic & medicinal chemistry letters (06.10.1998)
Published in Bioorganic & medicinal chemistry letters (06.10.1998)
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Total synthesis of (+)-demethyldysidenin and (-)-demethylisodysidenin, hexachlorinated amino acids from the marine sponge Dysidea herbacea. Assignment of absolute stereochemistry
De Laszlo, Stephen E, Williard, Paul G
Published in Journal of the American Chemical Society (01.01.1985)
Published in Journal of the American Chemical Society (01.01.1985)
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Deprotection of N- tert-butoxycarbonyl (Boc) groups in the presence of tert-butyl esters
Lin, Linus S, Lanza, Thomas, de Laszlo, Stephen E, Truong, Quang, Kamenecka, Theodore, Hagmann, William K
Published in Tetrahedron letters (02.09.2000)
Published in Tetrahedron letters (02.09.2000)
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Amidines as amide bond replacements in VLA-4 antagonists
KAMENECKA, Theodore M, PARK, You-Jung, WEI TANG, COLLETTI, Adria, TEFFERA, Yohannes, STEARNS, Ralph, MACCOSS, Malcolm, SCHMIDT, John A, HAGMANN, William K, LIN, Linus S, DE LASZLO, Stephen, MCCAULEY, Ermengilda D, VAN RIPER, Gail, EGGER, Linda, KIDAMBI, Usha, MUMFORD, Richard A, TONG, Sharon
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Carbohydroxamido-oxazolidines: antibacterial agents that target lipid A biosynthesis
Chen, Meng-Hsin, Steiner, Mark G., de Laszlo, Stephen E., Patchett, Arthur A., Anderson, Matt S., Hyland, Sheryl A., Russell Onishi, H., Silyer, Lynn L., Raetz, Christian R.H.
Published in Bioorganic & medicinal chemistry letters (08.02.1999)
Published in Bioorganic & medicinal chemistry letters (08.02.1999)
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A small molecule alpha4beta1/alpha4beta7 antagonist differentiates between the low-affinity states of alpha4beta1 and alpha4beta7: characterization of divalent cation dependence
Egger, Linda A, Cao, Jin, McCallum, Christine, Kidambi, Usha, Van Riper, Gail, McCauley, Ermengilda, Mumford, Richard A, Lanza, Thomas J, Lin, Linus S, de Laszlo, Stephen E, Young, David N, Yang, Ginger, Dean, Dennis C, Raab, Conrad E, Wallace, Mike A, Jones, Allen N, Hagmann, William K, Schmidt, John A, Pepinsky, R Blake, Scott, Daniel M, Lee, Wen-Cherng, Cornebise, Mark A, Detmers, Patricia A
Published in The Journal of pharmacology and experimental therapeutics (01.09.2003)
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Published in The Journal of pharmacology and experimental therapeutics (01.09.2003)
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A Small Molecule α 4 β 1 /α 4 β 7 Antagonist Differentiates between the Low-Affinity States of α 4 β 1 and α 4 β 7 : Characterization of Divalent Cation Dependence
Egger, Linda A., Cao, Jin, McCallum, Christine, Kidambi, Usha, Van Riper, Gail, McCauley, Ermengilda, Mumford, Richard A., Lanza, Thomas J., Lin, Linus S., de Laszlo, Stephen E., Young, David N., Yang, Ginger, Dean, Dennis C., Raab, Conrad E., Wallace, Mike A., Jones, Allen N., Hagmann, William K., Schmidt, John A., Pepinsky, R. Blake, Scott, Daniel M., Lee, Wen-Cherng, Cornebise, Mark A., Detmers, Patricia A.
Published in The Journal of pharmacology and experimental therapeutics (01.09.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2003)
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