Molecular basis for cooperative binding and synergy of ATP-site and allosteric EGFR inhibitors
Beyett, Tyler S, To, Ciric, Heppner, David E, Rana, Jaimin K, Schmoker, Anna M, Jang, Jaebong, De Clercq, Dries J H, Gomez, Gabriel, Scott, David A, Gray, Nathanael S, Jänne, Pasi A, Eck, Michael J
Published in Nature communications (09.05.2022)
Published in Nature communications (09.05.2022)
Get full text
Journal Article
Discovery of a Highly Potent and Broadly Effective Epidermal Growth Factor Receptor and HER2 Exon 20 Insertion Mutant Inhibitor
Jang, Jaebong, Son, Jieun, Park, Eunyoung, Kosaka, Takayuki, Saxon, Jamie A., De Clercq, Dries J. H., Choi, Hwan Geun, Tanizaki, Junko, Eck, Michael J., Jänne, Pasi A., Gray, Nathanael S.
Published in Angewandte Chemie (International ed.) (03.09.2018)
Published in Angewandte Chemie (International ed.) (03.09.2018)
Get full text
Journal Article
Mutant‐Selective Allosteric EGFR Degraders are Effective Against a Broad Range of Drug‐Resistant Mutations
Jang, Jaebong, To, Ciric, De Clercq, Dries J. H., Park, Eunyoung, Ponthier, Charles M., Shin, Bo Hee, Mushajiang, Mierzhati, Nowak, Radosław P., Fischer, Eric S., Eck, Michael J., Jänne, Pasi A., Gray, Nathanael S.
Published in Angewandte Chemie International Edition (17.08.2020)
Published in Angewandte Chemie International Edition (17.08.2020)
Get full text
Journal Article
Fast micromagnetic simulations on GPU-recent advances made with mumax3
Leliaert, J, Dvornik, M, Mulkers, J, De Clercq, J, Miloševi, M V, Van Waeyenberge, B
Published in Journal of physics. D, Applied physics (21.02.2018)
Published in Journal of physics. D, Applied physics (21.02.2018)
Get full text
Journal Article
Discovery and Optimization of Dibenzodiazepinones as Allosteric Mutant-Selective EGFR Inhibitors
De Clercq, Dries J. H, Heppner, David E, To, Ciric, Jang, Jaebong, Park, Eunyoung, Yun, Cai-Hong, Mushajiang, Mierzhati, Shin, Bo Hee, Gero, Thomas W, Scott, David A, Jänne, Pasi A, Eck, Michael J, Gray, Nathanael S
Published in ACS medicinal chemistry letters (14.11.2019)
Published in ACS medicinal chemistry letters (14.11.2019)
Get full text
Journal Article
Effect of Organic Selenium in the Diet on Sperm Quality of Boars
López, A, Rijsselaere, T, Van Soom, A, Leroy, JLMR, De Clercq, JBP, Bols, PEJ, Maes, D
Published in Reproduction in domestic animals (01.12.2010)
Published in Reproduction in domestic animals (01.12.2010)
Get full text
Journal Article
Chemical Dimerizers in Three-Hybrid Systems for Small Molecule–Target Protein Profiling
De Clercq, Dries J. H, Tavernier, Jan, Lievens, Sam, Van Calenbergh, Serge
Published in ACS chemical biology (19.08.2016)
Published in ACS chemical biology (19.08.2016)
Get full text
Journal Article
Proteome-scale Binary Interactomics in Human Cells
Lievens, Sam, Van der Heyden, José, Masschaele, Delphine, De Ceuninck, Leentje, Petta, Ioanna, Gupta, Surya, De Puysseleyr, Veronic, Vauthier, Virginie, Lemmens, Irma, De Clercq, Dries J.H., Defever, Dieter, Vanderroost, Nele, De Smet, Anne-Sophie, Eyckerman, Sven, Van Calenbergh, Serge, Martens, Lennart, De Bosscher, Karolien, Libert, Claude, Hill, David E., Vidal, Marc, Tavernier, Jan
Published in Molecular & cellular proteomics (01.12.2016)
Published in Molecular & cellular proteomics (01.12.2016)
Get full text
Journal Article
An optimized Agrobacterium-mediated transformation procedure for Phaseolus acutifolius A. Gray
DE CLERCQ, J, ZAMBRE, M, VAN MONTAGU, M, DILLEN, W, ANGENON, G
Published in Plant cell reports (01.11.2002)
Published in Plant cell reports (01.11.2002)
Get full text
Journal Article
Diagnosing COVID-19; towards a feasible COVID-19 rule-out protocol
De Clercq, J, Malfait, T, Malfait, S, Boelens, J, Coorevits, L, Padalko, E, Vandendriessche, S, Verhasselt, B, Morbée, L, Bauters, F, Hertegonne, K, Stevens, D, Vande Weygaerde, Y, Vermaelen, K, Van Biesen, W, Vanommeslaeghe, F, Verbeke, F, Piers, R, Van Den Noortgate, N, Desmet, T, Vermassen, F, Vandekerckhove, L, Van Braeckel, E
Published in Acta clinica belgica (English ed. Online) (01.04.2022)
Published in Acta clinica belgica (English ed. Online) (01.04.2022)
Get more information
Journal Article
Evaluation of epididymis storage temperature and cryopreservation conditions for improved mitochondrial membrane potential, membrane integrity, sperm motility and in vitro fertilization in bovine epididymal sperm
Nichi, M, Rijsselaere, T, Losano, JDA, Angrimani, DSR, Kawai, GKV, Goovaerts, IGF, Van Soom, A, Barnabe, VH, De Clercq, JBP, Bols, PEJ
Published in Reproduction in domestic animals (01.04.2017)
Published in Reproduction in domestic animals (01.04.2017)
Get full text
Journal Article
Single and Dual Targeting of Mutant EGFR with an Allosteric Inhibitor
To, Ciric, Jang, Jaebong, Chen, Ting, Park, Eunyoung, Mushajiang, Mierzhati, De Clercq, Dries J H, Xu, Man, Wang, Stephen, Cameron, Michael D, Heppner, David E, Shin, Bo Hee, Gero, Thomas W, Yang, Annan, Dahlberg, Suzanne E, Wong, Kwok-Kin, Eck, Michael J, Gray, Nathanael S, Jänne, Pasi A
Published in Cancer discovery (01.07.2019)
Published in Cancer discovery (01.07.2019)
Get full text
Journal Article
OP 3.8 – 00066 Characterization of the HIV-1 viral reservoir in subtype B early treated individuals
Struyve, T., Pardons, M., Termote, L., De Clercq, J., Lambrechts, L., Vega, J., Boden, D., Lichterfeld, M., Rutsaert, S., Vandekerckhove, L.
Published in Journal of Virus Eradication (01.12.2022)
Published in Journal of Virus Eradication (01.12.2022)
Get full text
Journal Article
Agrobacterium-mediated transformation of Phaseolus acutifolius A. Gray
Dillen, W, Clercq, J. de, Goossens, A, Montagu, M. van, Angenon, G. (Gent Univ. (Belgium). Flanders Interuniv. Inst. for Biotechnology. Dept. of Genetics. Lab. voor Genetica)
Published in Theoretical and applied genetics (01.02.1997)
Published in Theoretical and applied genetics (01.02.1997)
Get full text
Journal Article
Quantification and Viability Assessment of Isolated Bovine Primordial and Primary Ovarian Follicles Retrieved Through a Standardized Biopsy Pick-Up Procedure
Aerts, JMJ, Martinez-Madrid, B, Flothmann, K, De Clercq, JBP, Van Aelst, S, Bols, PEJ
Published in Reproduction in domestic animals (01.06.2008)
Published in Reproduction in domestic animals (01.06.2008)
Get full text
Journal Article