Substituted Aryl Benzylamines as Potent and Selective Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 3
Vicker, Nigel, Bailey, Helen V, Day, Joanna M, Mahon, Mary F, Smith, Andrew, Tutill, Helena J, Purohit, Atul, Potter, Barry V L
Published in Molecules (Basel, Switzerland) (26.11.2021)
Published in Molecules (Basel, Switzerland) (26.11.2021)
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Journal Article
Design and validation of specific inhibitors of 17β-hydroxysteroid dehydrogenases for therapeutic application in breast and prostate cancer, and in endometriosis
Day, Joanna M, Tutill, Helena J, Purohit, Atul, Reed, Michael J
Published in Endocrine-related cancer (01.09.2008)
Published in Endocrine-related cancer (01.09.2008)
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Journal Article
STX140, but not paclitaxel, inhibits mammary tumour initiation and progression in C3(1)/SV40 T/t-antigen transgenic mice
Meyer-Losic, Florence, Newman, Simon P, Day, Joanna M, Reed, Michael J, Kasprzyk, Philip G, Purohit, Atul, Foster, Paul A
Published in PloS one (06.12.2013)
Published in PloS one (06.12.2013)
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Journal Article
The Development of Steroid Sulfatase Inhibitors for Hormone-Dependent Cancer Therapy
Day, Joanna M., Purohit, Atul, Tutill, Helena J., Foster, Paul A., Woo, L. W. Lawrence, Potter, Barry V. L., Reed, Michael J.
Published in Annals of the New York Academy of Sciences (01.02.2009)
Published in Annals of the New York Academy of Sciences (01.02.2009)
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Journal Article
Alternative Splicing in the Aggrecan G3 Domain Influences Binding Interactions with Tenascin-C and Other Extracellular Matrix Proteins
Day, Joanna M., Olin, Anders I., Murdoch, Alan D., Canfield, Ann, Sasaki, Takako, Timpl, Rupert, Hardingham, Timothy E., Aspberg, Anders
Published in The Journal of biological chemistry (26.03.2004)
Published in The Journal of biological chemistry (26.03.2004)
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Journal Article
STX140 Is Efficacious In vitro and In vivo in Taxane-Resistant Breast Carcinoma Cells
NEWMAN, Simon P, FOSTER, Paul A, REED, Michael J, PUROHIT, Atul, STENGEL, Chloe, DAY, Joanna M, HO, Yaik T, JUDDE, Jean-Gabriel, LASSALLE, Myriam, PREVOST, Gregoire, LEESE, Mathew P, POTTER, Barry V. L
Published in Clinical cancer research (15.01.2008)
Published in Clinical cancer research (15.01.2008)
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Journal Article
Overexpression of 17β-Hydroxysteroid Dehydrogenase Type 1 Increases the Exposure of Endometrial Cancer to 17β-Estradiol
Cornel, Karlijn M. C, Kruitwagen, Roy F. P. M, Delvoux, Bert, Visconti, Laura, Van de Vijver, Koen K, Day, Joanna M, Van Gorp, Toon, Hermans, Rob J. J, Dunselman, Gerard A, Romano, Andrea
Published in The journal of clinical endocrinology and metabolism (01.04.2012)
Published in The journal of clinical endocrinology and metabolism (01.04.2012)
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Journal Article
17β‐hydroxysteroid dehydrogenase Type 1, and not Type 12, is a target for endocrine therapy of hormone‐dependent breast cancer
Day, Joanna M., Foster, Paul A., Tutill, Helena J., Parsons, Michael F.C., Newman, Simon P., Chander, Surinder K., Allan, Gillian M., Lawrence, Harshani R., Vicker, Nigel, Potter, Barry V.L., Reed, Michael J., Purohit, Atul
Published in International journal of cancer (01.05.2008)
Published in International journal of cancer (01.05.2008)
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Journal Article
17 beta -hydroxysteroid dehydrogenase Type 1, and not Type 12, is a target for endocrine therapy of hormone-dependent breast cancer
Day, Joanna M, Foster, Paul A, Tutill, Helena J, Parsons, Michael F C, Newman, Simon P, Chander, Surinder K, Allan, Gillian M, Lawrence, Harshani R, Vicker, Nigel, Potter, Barry V L, Reed, Michael J, Purohit, Atul
Published in International journal of cancer (01.05.2008)
Published in International journal of cancer (01.05.2008)
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Journal Article
Order within disorder: Aggrecan chondroitin sulphate-attachment region provides new structural insights into protein sequences classified as disordered
Jowitt, Thomas A., Murdoch, Alan D., Baldock, Clair, Berry, Richard, Day, Joanna M., Hardingham, Timothy E.
Published in Proteins, structure, function, and bioinformatics (01.12.2010)
Published in Proteins, structure, function, and bioinformatics (01.12.2010)
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Journal Article
STX2171, a 17β-hydroxysteroid dehydrogenase type 3 inhibitor, is efficacious in vivo in a novel hormone-dependent prostate cancer model
Day, Joanna M, Foster, Paul A, Tutill, Helena J, Schmidlin, Fabien, Sharland, Christopher M, Hargrave, Jonathan D, Vicker, Nigel, Potter, Barry V L, Reed, Michael J, Purohit, Atul
Published in Endocrine-related cancer (01.02.2013)
Published in Endocrine-related cancer (01.02.2013)
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Journal Article
Modification of Estrone at the 6, 16, and 17 Positions: Novel Potent Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 1
Allan, Gillian M, Lawrence, Harshani R, Cornet, Josephine, Bubert, Christian, Fischer, Delphine S, Vicker, Nigel, Smith, Andrew, Tutill, Helena J, Purohit, Atul, Day, Joanna M, Mahon, Mary F, Reed, Michael J, Potter, Barry V. L
Published in Journal of medicinal chemistry (23.02.2006)
Published in Journal of medicinal chemistry (23.02.2006)
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Journal Article
Novel inhibitors of 17β-hydroxysteroid dehydrogenase type 1: Templates for design
Allan, Gillian M., Vicker, Nigel, Lawrence, Harshani R., Tutill, Helena J., Day, Joanna M., Huchet, Marion, Ferrandis, Eric, Reed, Michael J., Purohit, Atul, Potter, Barry V.L.
Published in Bioorganic & medicinal chemistry (15.04.2008)
Published in Bioorganic & medicinal chemistry (15.04.2008)
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Journal Article
The role of 17β-hydroxysteroid dehydrogenases in modulating the activity of 2-methoxyestradiol in breast cancer cells
NEWMAN, Simon P, IRESON, Christopher R, TUTILL, Helena J, DAY, Joanna M, PARSONS, Michael F. C, LEESE, Mathew P, POTTER, Barry V. L, REED, Michael J, PUROHIT, Atul
Published in Cancer research (Chicago, Ill.) (2006)
Published in Cancer research (Chicago, Ill.) (2006)
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Journal Article
The design of novel 17β-hydroxysteroid dehydrogenase type 3 inhibitors
Vicker, Nigel, Sharland, Christopher M., Heaton, Wesley B., Gonzalez, Ana M. Ramos, Bailey, Helen V., Smith, Andrew, Springall, Jeremy S., Day, Joanna M., Tutill, Helena J., Reed, Michael J., Purohit, Atul, Potter, Barry V.L.
Published in Molecular and cellular endocrinology (25.03.2009)
Published in Molecular and cellular endocrinology (25.03.2009)
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Journal Article
Development of hormone-dependent prostate cancer models for the evaluation of inhibitors of 17β-hydroxysteroid dehydrogenase Type 3
Day, Joanna M., Tutill, Helena J., Foster, Paul A., Bailey, Helen V., Heaton, Wesley B., Sharland, Christopher M., Vicker, Nigel, Potter, Barry V.L., Purohit, Atul, Reed, Michael J.
Published in Molecular and cellular endocrinology (25.03.2009)
Published in Molecular and cellular endocrinology (25.03.2009)
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Journal Article
Focused libraries of 16-substituted estrone derivatives and modified e-ring steroids: inhibitors of 17beta-hydroxysteroid dehydrogenase type 1
Vicker, Nigel, Lawrence, Harshani R, Allan, Gillian M, Bubert, Christian, Smith, Andrew, Tutill, Helena J, Purohit, Atul, Day, Joanna M, Mahon, Mary F, Reed, Michael J, Potter, Barry V L
Published in ChemMedChem (01.04.2006)
Published in ChemMedChem (01.04.2006)
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Journal Article
Cytokines in human breast cyst fluid
Parish, David C., Ghilchik, Margaret W., Day, Joanna M., Eaton, James, Purohit, Atul, Reed, Michael J.
Published in The Journal of steroid biochemistry and molecular biology (01.05.2007)
Published in The Journal of steroid biochemistry and molecular biology (01.05.2007)
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Journal Article
The effects of 2-substituted oestrogen sulphamates on the growth of prostate and ovarian cancer cells
Day, Joanna M., Newman, Simon P., Comninos, Alexander, Solomon, Claire, Purohit, Atul, Leese, Matthew P., Potter, Barry V.L., Reed, Michael J.
Published in Journal of steroid biochemistry and molecular biology (01.02.2003)
Published in Journal of steroid biochemistry and molecular biology (01.02.2003)
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