Search Results - "DAX, SCOTT" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloid Receptor Antagonist

Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloid Receptor Antagonist

by Swanson, Devin M, Dubin, Adrienne E, Shah, Chandra, Nasser, Nadia, Chang, Leon, Dax, Scott L, Jetter, Michele, Breitenbucher, J. Guy, Liu, Changlu, Mazur, Curt, Lord, Brian, Gonzales, Lisa, Hoey, Kenway, Rizzolio, Michele, Bogenstaetter, Michael, Codd, Ellen E, Lee, Doo H, Zhang, Sui-Po, Chaplan, Sandra R, Carruthers, Nicholas I
Published in Journal of medicinal chemistry (24.03.2005)

Get full text

Journal Article

JNJ-20788560 [9-(8-Azabicyclo[3.2.1]oct-3-ylidene)-9H-xanthene-3-carboxylic Acid Diethylamide], a Selective Delta Opioid Receptor Agonist, Is a Potent and Efficacious Antihyperalgesic Agent That Does Not Produce Respiratory Depression, Pharmacologic Tolerance, or Physical Dependence

JNJ-20788560 [9-(8-Azabicyclo[3.2.1]oct-3-ylidene)-9H-xanthene-3-carboxylic Acid Diethylamide], a Selective Delta Opioid Receptor Agonist, Is a Potent and Efficacious Antihyperalgesic Agent That Does Not Produce Respiratory Depression, Pharmacologic Tolerance, or Physical Dependence

by Codd, Ellen E, Carson, John R, Colburn, Raymond W, Stone, Dennis J, Van Besien, Christopher R, Zhang, Sui-Po, Wade, Paul R, Gallantine, Elizabeth L, Meert, Theo F, Molino, Lory, Pullan, Shirley, Razler, Christine M, Dax, Scott L, Flores, Christopher M
Published in The Journal of pharmacology and experimental therapeutics (01.04.2009)

Get full text

Journal Article

Iodoacetic Acid is an Efficient Reagent for the Synthesis of Amino Acid Derived 2-Aminobenzimidazoles

Iodoacetic Acid is an Efficient Reagent for the Synthesis of Amino Acid Derived 2-Aminobenzimidazoles

by Krasikovs, Andrejs, Ozola, Vita, Dax, Scott L., Suna, Edgars
Published in Synthesis (Stuttgart) (01.03.2013)

Get more information

Journal Article

Benzo[d]imidazole Transient Receptor Potential Vanilloid 1 Antagonists for the Treatment of Pain: Discovery of trans-2-(2-{2-[2-(4-Trifluoromethyl-phenyl)-vinyl]‑1H‑benzimidazol-5-yl}-phenyl)-propan-2-ol (Mavatrep)

Benzo[d]imidazole Transient Receptor Potential Vanilloid 1 Antagonists for the Treatment of Pain: Discovery of trans-2-(2-{2-[2-(4-Trifluoromethyl-phenyl)-vinyl]‑1H‑benzimidazol-5-yl}-phenyl)-propan-2-ol (Mavatrep)

by Parsons, William H, Calvo, Raul R, Cheung, Wing, Lee, Yu-Kai, Patel, Sharmila, Liu, Jian, Youngman, Mark A, Dax, Scott L, Stone, Dennis, Qin, Ning, Hutchinson, Tasha, Lubin, Mary Lou, Zhang, Sui-Po, Finley, Michael, Liu, Yi, Brandt, Michael R, Flores, Christopher M, Player, Mark R
Published in Journal of medicinal chemistry (14.05.2015)

Get full text

Journal Article

The design and synthesis of novel, phosphonate-containing transient receptor potential melastatin 8 (TRPM8) antagonists

The design and synthesis of novel, phosphonate-containing transient receptor potential melastatin 8 (TRPM8) antagonists

by Matthews, Jay M., Qin, Ning, Colburn, Raymond W., Dax, Scott L., Hawkins, Mike, McNally, James J., Reany, Laura, Youngman, Mark A., Baker, Judith, Hutchinson, Tasha, Liu, Yi, Lubin, Mary Lou, Neeper, Michael, Brandt, Michael R., Stone, Dennis J., Flores, Christopher M.
Published in Bioorganic & medicinal chemistry letters (15.04.2012)

Get full text

Journal Article

Arylglycine derivatives as potent transient receptor potential melastatin 8 (TRPM8) antagonists

Arylglycine derivatives as potent transient receptor potential melastatin 8 (TRPM8) antagonists

by Zhu, Bin, Xia, Mingde, Xu, Xiaoqing, Ludovici, Donald W., Tennakoon, Manomi, Youngman, Mark A., Matthews, Jay M., Dax, Scott L., Colburn, Raymond W., Qin, Ning, Hutchinson, Tasha L., Lubin, Mary Lou, Brandt, Michael R., Stone, Dennis J., Flores, Christopher M., Macielag, Mark J.
Published in Bioorganic & medicinal chemistry letters (01.04.2013)

Get full text

Journal Article

Heteroaryl β-tetralin ureas as novel antagonists of human TRPV1

Heteroaryl β-tetralin ureas as novel antagonists of human TRPV1

by Jetter, Michele C., Youngman, Mark A., McNally, James J., McDonnell, Mark E., Zhang, Sui-Po, Dubin, Adrienne E., Nasser, Nadia, Codd, Ellen E., Flores, Christopher M., Dax, Scott L.
Published in Bioorganic & medicinal chemistry (15.11.2007)

Get full text

Journal Article

Diabetogenic Effect of a Series of Tricyclic Delta Opioid Agonists Structurally Related to Cyproheptadine

Diabetogenic Effect of a Series of Tricyclic Delta Opioid Agonists Structurally Related to Cyproheptadine

by Codd, Ellen E., Baker, Judith, Brandt, Michael R., Bryant, Stewart, Cai, Chaozhong, Carson, John R., Chevalier, Kristen M., Colburn, Raymond W., Coogan, Timothy P., Dax, Scott L., DeCorte, Bart, Kemmerer, Michael, LeGrand, Edmund K., Lenhard, James M., Leone, Angelique M., Lin, Ling, Mabus, John R., McDonnell, Mark E., McMillian, Michael K., McNally, James J., Stone, Dennis J., Wang, Charles Y., Zhang, Sui-Po, Flores, Christopher M.
Published in Toxicological sciences (01.10.2010)

Get full text

Journal Article

티아졸린 항통각과민제로 통증을 치료하는 방법

티아졸린 항통각과민제로 통증을 치료하는 방법

by DAX SCOTT
Year of Publication 14.10.2021

Get full text

Patent

N-Pyridin-3-yl- and N-quinolin-3-yl-benzamides: Modulators of Human Vanilloid Receptor 1 (TRPV1)

N-Pyridin-3-yl- and N-quinolin-3-yl-benzamides: Modulators of Human Vanilloid Receptor 1 (TRPV1)

by Jetter, Michele C., McNally, James J., Youngman, Mark A., McDonnell, Mark E., Dubin, Adrienne E., Nasser, Nadia, Zhang, Sui-Po, Codd, Ellen E., Colburn, Ray W., Stone, Dennis R., Brandt, Michael R., Flores, Christopher M., Dax, Scott L.
Published in Bioorganic & medicinal chemistry letters (15.04.2008)

Get full text

Journal Article

N-Isoquinolin-5-yl- N′-aralkyl-urea and -amide antagonists of human vanilloid receptor 1

N-Isoquinolin-5-yl- N′-aralkyl-urea and -amide antagonists of human vanilloid receptor 1

by Jetter, Michele C., Youngman, Mark A., McNally, James J., Zhang, Sui-Po, Dubin, Adrienne E., Nasser, Nadia, Dax, Scott L.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)

Get full text

Journal Article

N, N-Dialkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, potent, selective δ opioid agonists

N, N-Dialkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, potent, selective δ opioid agonists

by CARSON, John R, COATS, Steven J, CODD, Ellen E, DAX, Scott L, JUNG LEE, MARTINEZ, Rebecca P, NEILSON, Lou Anne, PITIS, Philip M, ZHANG, Sui-Po
Published in Bioorganic & medicinal chemistry letters (03.05.2004)

Get full text

Journal Article

7-Hydroxynaphthalen-1-yl-urea and -amide antagonists of human vanilloid receptor 1

7-Hydroxynaphthalen-1-yl-urea and -amide antagonists of human vanilloid receptor 1

by McDonnell, Mark E., Zhang, Sui-Po, Nasser, Nadia, Dubin, Adrienne E., Dax, Scott L.
Published in Bioorganic & medicinal chemistry letters (2004)

Get full text

Journal Article

티아졸린 항통각과민제의 제조 방법 및 다형체

티아졸린 항통각과민제의 제조 방법 및 다형체

by DAX SCOTT L
Year of Publication 17.01.2022

Get full text

Patent

Parallel methods for the preparation and SAR exploration of N-ethyl-4-[(8-alkyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-aryl-methyl]-benzamides, powerful mu and delta opioid agonists

Parallel methods for the preparation and SAR exploration of N-ethyl-4-[(8-alkyl-8-aza-bicyclo[3.2.1]oct-3-ylidene)-aryl-methyl]-benzamides, powerful mu and delta opioid agonists

by Coats, Steven J., Schulz, Mark J., Carson, John R., Codd, Ellen E., Hlasta, Dennis J., Pitis, Philip M., Stone, Dennis J., Zhang, Sui-Po, Colburn, Ray W., Dax, Scott L.
Published in Bioorganic & medicinal chemistry letters (15.11.2004)

Get full text

Journal Article

Synthesis and in vitro evaluation of a novel iodinated resiniferatoxin derivative that is an agonist at the human vanilloid VR1 receptor

Synthesis and in vitro evaluation of a novel iodinated resiniferatoxin derivative that is an agonist at the human vanilloid VR1 receptor

by MCDONNELL, Mark E, ZHANG, Sui-Po, DUBIN, Adrienne E, DAX, Scott L
Published in Bioorganic & medicinal chemistry letters (22.04.2002)

Get full text

Journal Article

Explorer51 - Indoor Mapping, Discovery, and Navigation for an Autonomous Mobile Robot

Explorer51 - Indoor Mapping, Discovery, and Navigation for an Autonomous Mobile Robot

by Argush, Gabriel, Holincheck, William, Krynitsky, Jessica, McGuire, Brian, Scott, Dax, Tolleson, Charlie, Behl, Madhur
Published in 2020 Systems and Information Engineering Design Symposium (SIEDS) (01.04.2020)

Get full text

Conference Proceeding

Novel non-peptidic neuropeptide Y Y2 receptor antagonists

Novel non-peptidic neuropeptide Y Y2 receptor antagonists

by JABLONOWSKI, Jill A, WENYING CHAI, CARRUTHERS, Nicholas I, XIAOBING LI, RUDOLPH, Dale A, MURRAY, William V, YOUNGMAN, Mark A, DAX, Scott L, NEPOMUCENO, Diane, BONAVENTURE, Pascal, LOVENBERG, Timothy W
Published in Bioorganic & medicinal chemistry letters (08.03.2004)

Get full text

Journal Article

Aminopyrazoles with high affinity for the human neuropeptide Y5 receptor

Aminopyrazoles with high affinity for the human neuropeptide Y5 receptor

by Kordik, Cheryl P, Luo, Chi, Zanoni, Brian C, Dax, Scott L, McNally, James J, Lovenberg, Timothy W, Wilson, Sandy J, Reitz, Allen B
Published in Bioorganic & medicinal chemistry letters (03.09.2001)

Get full text

Journal Article

N-Alkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, μ and δ opioid agonists: a μ address

N-Alkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]-benzamides, μ and δ opioid agonists: a μ address

by CARSON, John R, COATS, Steven J, ZHANG, Sui-Po, CODD, Ellen E, DAX, Scott L, JUNG LEE, MARTINEZ, Rebecca P, MCKOWN, Linda A, NEILSON, Lou Anne, PITIS, Philip M, WU, Wu-Nan
Published in Bioorganic & medicinal chemistry letters (03.05.2004)

Get full text

Journal Article

1
2
3
4
5
6
7
8
9
10
11
Next
[20]