GPR91 senses extracellular succinate released from inflammatory macrophages and exacerbates rheumatoid arthritis
Littlewood-Evans, Amanda, Sarret, Sophie, Apfel, Verena, Loesle, Perrine, Dawson, Janet, Zhang, Juan, Muller, Alban, Tigani, Bruno, Kneuer, Rainer, Patel, Saijel, Valeaux, Stephanie, Gommermann, Nina, Rubic-Schneider, Tina, Junt, Tobias, Carballido, José M
Published in The Journal of experimental medicine (22.08.2016)
Published in The Journal of experimental medicine (22.08.2016)
Get full text
Journal Article
Discovery of LOU064 (Remibrutinib), a Potent and Highly Selective Covalent Inhibitor of Bruton’s Tyrosine Kinase
Angst, Daniela, Gessier, François, Janser, Philipp, Vulpetti, Anna, Wälchli, Rudolf, Beerli, Christian, Littlewood-Evans, Amanda, Dawson, Janet, Nuesslein-Hildesheim, Barbara, Wieczorek, Grazyna, Gutmann, Sascha, Scheufler, Clemens, Hinniger, Alexandra, Zimmerlin, Alfred, Funhoff, Enrico G, Pulz, Robert, Cenni, Bruno
Published in Journal of medicinal chemistry (28.05.2020)
Published in Journal of medicinal chemistry (28.05.2020)
Get full text
Journal Article
Pharmacological inhibition of RORγt suppresses the Th17 pathway and alleviates arthritis in vivo
Guendisch, Ulf, Weiss, Jessica, Ecoeur, Florence, Riker, Julia Christina, Kaupmann, Klemens, Kallen, Joerg, Hintermann, Samuel, Orain, David, Dawson, Janet, Billich, Andreas, Guntermann, Christine
Published in PloS one (20.11.2017)
Published in PloS one (20.11.2017)
Get full text
Journal Article
A natural ligand for the orphan receptor GPR15 modulates lymphocyte recruitment to epithelia
Suply, Thomas, Hannedouche, Sébastien, Carte, Nathalie, Li, Jianping, Grosshans, Bianka, Schaefer, Michael, Raad, Layla, Beck, Valérie, Vidal, Solange, Hiou-Feige, Agnès, Beluch, Noémie, Barbieri, Samuel, Wirsching, Johann, Lageyre, Nadine, Hillger, Frank, Debon, Corinne, Dawson, Janet, Smith, Philip, Lannoy, Vincent, Detheux, Michel, Bitsch, Francis, Falchetto, Rocco, Bouwmeester, Tewis, Porter, Jeffrey, Baumgarten, Birgit, Mansfield, Keith, Carballido, José M, Seuwen, Klaus, Bassilana, Frédéric
Published in Science signaling (12.09.2017)
Published in Science signaling (12.09.2017)
Get more information
Journal Article
Degenerative joint disease induced by repeated intra-articular injections of monosodium urate crystals in rats as investigated by translational imaging
Accart, Nathalie, Dawson, Janet, Obrecht, Michael, Lambert, Christian, Flueckiger, Manuela, Kreider, Julie, Hatakeyama, Shinji, Richards, Peter J., Beckmann, Nicolau
Published in Scientific reports (07.01.2022)
Published in Scientific reports (07.01.2022)
Get full text
Journal Article
Pathophysiological Consequences of a Break in S1P1-Dependent Homeostasis of Vascular Permeability Revealed by S1P1 Competitive Antagonism
Bigaud, Marc, Dincer, Zuhal, Bollbuck, Birgit, Dawson, Janet, Beckmann, Nicolau, Beerli, Christian, Fishli-Cavelti, Gina, Nahler, Michaela, Angst, Daniela, Janser, Philipp, Otto, Heike, Rosner, Elisabeth, Hersperger, Rene, Bruns, Christian, Quancard, Jean
Published in PloS one (22.12.2016)
Published in PloS one (22.12.2016)
Get full text
Journal Article
Transient targeting of phosphoinositide 3-kinase acts as a roadblock in mast cells' route to allergy
Collmann, Emilie, PhD, Bohnacker, Thomas, PhD, Marone, Romina, PhD, Dawson, Janet, PhD, Rehberg, Markus, PhD, Stringer, Rowan, PhD, Krombach, Fritz, PhD, Burkhart, Christoph, PhD, Hirsch, Emilio, PhD, Hollingworth, Gregory J., PhD, Thomas, Matthew, PhD, Wymann, Matthias P., PhD
Published in Journal of allergy and clinical immunology (01.10.2013)
Published in Journal of allergy and clinical immunology (01.10.2013)
Get full text
Journal Article
Choice behavior of the generalist pentatomid predator Podisus maculiventris when offered lepidopteran larvae infected with an entomopathogenic fungus
Avery, Pasco B., George, Justin, Markle, Larry, Martini, Xavier, Rowley, Amy L., Meagher, Robert L., Barger, Rachel E., Duren, Emily B., Dawson, Janet S., Cave, Ronald D.
Published in BioControl (Dordrecht, Netherlands) (01.04.2022)
Published in BioControl (Dordrecht, Netherlands) (01.04.2022)
Get full text
Journal Article
Fluorescent Nanoprobes as a Biomarker for Increased Vascular Permeability: Implications in Diagnosis and Treatment of Cancer and Inflammation
Sandanaraj, Britto S, Gremlich, Hans-Ulrich, Kneuer, Rainer, Dawson, Janet, Wacha, Stefan
Published in Bioconjugate chemistry (20.01.2010)
Published in Bioconjugate chemistry (20.01.2010)
Get full text
Journal Article
Development of Selective, Orally Active GPR4 Antagonists with Modulatory Effects on Nociception, Inflammation, and Angiogenesis
Velcicky, Juraj, Miltz, Wolfgang, Oberhauser, Berndt, Orain, David, Vaupel, Andrea, Weigand, Klaus, Dawson King, Janet, Littlewood-Evans, Amanda, Nash, Mark, Feifel, Roland, Loetscher, Pius
Published in Journal of medicinal chemistry (11.05.2017)
Published in Journal of medicinal chemistry (11.05.2017)
Get full text
Journal Article
Inhibition of the Inositol Kinase Itpkb Augments Calcium Signaling in Lymphocytes and Reveals a Novel Strategy to Treat Autoimmune Disease
Miller, Andrew T, Dahlberg, Carol, Sandberg, Mark L, Wen, Ben G, Beisner, Daniel R, Hoerter, John A H, Parker, Albert, Schmedt, Christian, Stinson, Monique, Avis, Jacqueline, Cienfuegos, Cynthia, McPate, Mark, Tranter, Pamela, Gosling, Martin, Groot-Kormelink, Paul J, Dawson, Janet, Pan, Shifeng, Tian, Shin-Shay, Seidel, H Martin, Cooke, Michael P
Published in PloS one (29.06.2015)
Published in PloS one (29.06.2015)
Get full text
Journal Article
Retinoic-acid-orphan-receptor-C inhibition suppresses Th17 cells and induces thymic aberrations
Guntermann, Christine, Piaia, Alessandro, Hamel, Marie-Laure, Theil, Diethilde, Rubic-Schneider, Tina, Del Rio-Espinola, Alberto, Dong, Linda, Billich, Andreas, Kaupmann, Klemens, Dawson, Janet, Hoegenauer, Klemens, Orain, David, Hintermann, Samuel, Stringer, Rowan, Patel, Dhavalkumar D, Doelemeyer, Arno, Deurinck, Mark, Schümann, Jens
Published in JCI insight (09.03.2017)
Published in JCI insight (09.03.2017)
Get full text
Journal Article
Nonhematopoietic IRAK1 drives arthritis via neutrophil chemoattractants
Hoyler, Thomas, Bannert, Bettina, André, Cédric, Beck, Damian, Boulay, Thomas, Buffet, David, Caesar, Nadja, Calzascia, Thomas, Dawson, Janet, Kyburz, Diego, Hennze, Robert, Huppertz, Christine, Littlewood-Evans, Amanda, Loetscher, Pius, Mertz, Kirsten D., Niwa, Satoru, Robert, Gautier, Rush, James S., Ruzzante, Giulia, Sarret, Sophie, Stein, Thomas, Touil, Ismahane, Wieczorek, Grazyna, Zipfel, Geraldine, Hawtin, Stuart, Junt, Tobias
Published in JCI insight (08.07.2022)
Published in JCI insight (08.07.2022)
Get full text
Journal Article
Preclinical pharmacology of lumiracoxib: a novel selective inhibitor of cyclooxygenase‐2
Esser, Ronald, Berry, Carol, Du, Zhengming, Dawson, Janet, Fox, Alyson, Fujimoto, Roger A, Haston, William, Kimble, Earl F, Koehler, Julie, Peppard, Jane, Quadros, Elizabeth, Quintavalla, Joseph, Toscano, Karen, Urban, Laszlo, Duzer, John, Zhang, Xiaoli, Zhou, Siyuan, Marshall, Paul J
Published in British journal of pharmacology (01.02.2005)
Published in British journal of pharmacology (01.02.2005)
Get full text
Journal Article
Serum Amyloid A (apoSAA) Expression Is Up-Regulated in Rheumatoid Arthritis and Induces Transcription of Matrix Metalloproteinases
Vallon, Rudiger, Freuler, Felix, Desta-Tsedu, Netsanet, Robeva, Anna, Dawson, Janet, Wenner, Peter, Engelhardt, Petra, Boes, Ludwig, Schnyder, Jorg, Tschopp, Claude, Urfer, Roman, Baumann, Gotz
Published in The Journal of immunology (1950) (15.02.2001)
Published in The Journal of immunology (1950) (15.02.2001)
Get full text
Journal Article
Hemoglobinase Activity of the Lysine Gingipain Protease (Kgp) of Porphyromonas gingivalis W83
Lewis, J P, Dawson, J A, Hannis, J C, Muddiman, D, Macrina, F L
Published in Journal of Bacteriology (01.08.1999)
Published in Journal of Bacteriology (01.08.1999)
Get full text
Journal Article
Anti-hyperalgesic activity of the cox-2 inhibitor lumiracoxib in a model of bone cancer pain in the rat
Fox, Alyson, Medhurst, Stephen, Courade, Jean-Philippe, Glatt, Marcus, Dawson, Janet, Urban, Laszlo, Bevan, Stuart, Gonzalez, Isabel
Published in Pain (Amsterdam) (2004)
Published in Pain (Amsterdam) (2004)
Get full text
Journal Article
Effects of dietary quebracho tannin on nutrient utilisation and tissue metabolism in sheep and rats
Dawson, J.M, Buttery, P.J, Jenkins, D, Wood, C.D, Gill, M
Published in Journal of the science of food and agriculture (01.08.1999)
Published in Journal of the science of food and agriculture (01.08.1999)
Get full text
Journal Article