The cancer epigenome: Concepts, challenges, and therapeutic opportunities
Dawson, Mark A.
Published in Science (American Association for the Advancement of Science) (17.03.2017)
Published in Science (American Association for the Advancement of Science) (17.03.2017)
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Targeting the epigenetic regulation of antitumour immunity
Hogg, Simon J, Beavis, Paul A, Dawson, Mark A, Johnstone, Ricky W
Published in Nature reviews. Drug discovery (01.11.2020)
Published in Nature reviews. Drug discovery (01.11.2020)
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Non-genetic mechanisms of therapeutic resistance in cancer
Marine, Jean-Christophe, Dawson, Sarah-Jane, Dawson, Mark A
Published in Nature reviews. Cancer (01.12.2020)
Published in Nature reviews. Cancer (01.12.2020)
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Ibrutinib plus Venetoclax for the Treatment of Mantle-Cell Lymphoma
Tam, Constantine S, Anderson, Mary Ann, Pott, Christiane, Agarwal, Rishu, Handunnetti, Sasanka, Hicks, Rodney J, Burbury, Kate, Turner, Gillian, Di Iulio, Juliana, Bressel, Mathias, Westerman, David, Lade, Stephen, Dreyling, Martin, Dawson, Sarah-Jane, Dawson, Mark A, Seymour, John F, Roberts, Andrew W
Published in The New England journal of medicine (29.03.2018)
Published in The New England journal of medicine (29.03.2018)
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An Evolutionarily Conserved Function of Polycomb Silences the MHC Class I Antigen Presentation Pathway and Enables Immune Evasion in Cancer
Burr, Marian L., Sparbier, Christina E., Chan, Kah Lok, Chan, Yih-Chih, Kersbergen, Ariena, Lam, Enid Y.N., Azidis-Yates, Elizabeth, Vassiliadis, Dane, Bell, Charles C., Gilan, Omer, Jackson, Susan, Tan, Lavinia, Wong, Stephen Q., Hollizeck, Sebastian, Michalak, Ewa M., Siddle, Hannah V., McCabe, Michael T., Prinjha, Rab K., Guerra, Glen R., Solomon, Benjamin J., Sandhu, Shahneen, Dawson, Sarah-Jane, Beavis, Paul A., Tothill, Richard W., Cullinane, Carleen, Lehner, Paul J., Sutherland, Kate D., Dawson, Mark A.
Published in Cancer cell (14.10.2019)
Published in Cancer cell (14.10.2019)
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Epigenetic silencing by the HUSH complex mediates position-effect variegation in human cells
Tchasovnikarova, Iva A., Timms, Richard T., Matheson, Nicholas J., Wals, Kim, Antrobus, Robin, Göttgens, Berthold, Dougan, Gordon, Dawson, Mark A., Lehner, Paul J.
Published in Science (American Association for the Advancement of Science) (26.06.2015)
Published in Science (American Association for the Advancement of Science) (26.06.2015)
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Selective targeting of BD1 and BD2 of the BET proteins in cancer and immunoinflammation
Gilan, Omer, Rioja, Inmaculada, Knezevic, Kathy, Bell, Matthew J, Yeung, Miriam M, Harker, Nicola R, Lam, Enid Y N, Chung, Chun-Wa, Bamborough, Paul, Petretich, Massimo, Urh, Marjeta, Atkinson, Stephen J, Bassil, Anna K, Roberts, Emma J, Vassiliadis, Dane, Burr, Marian L, Preston, Alex G S, Wellaway, Christopher, Werner, Thilo, Gray, James R, Michon, Anne-Marie, Gobbetti, Thomas, Kumar, Vinod, Soden, Peter E, Haynes, Andrea, Vappiani, Johanna, Tough, David F, Taylor, Simon, Dawson, Sarah-Jane, Bantscheff, Marcus, Lindon, Matthew, Drewes, Gerard, Demont, Emmanuel H, Daniels, Danette L, Grandi, Paola, Prinjha, Rab K, Dawson, Mark A
Published in Science (American Association for the Advancement of Science) (24.04.2020)
Published in Science (American Association for the Advancement of Science) (24.04.2020)
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TET2 and TET3 regulate GlcNAcylation and H3K4 methylation through OGT and SET1/COMPASS
Deplus, Rachel, Delatte, Benjamin, Schwinn, Marie K, Defrance, Matthieu, Méndez, Jacqui, Murphy, Nancy, Dawson, Mark A, Volkmar, Michael, Putmans, Pascale, Calonne, Emilie, Shih, Alan H, Levine, Ross L, Bernard, Olivier, Mercher, Thomas, Solary, Eric, Urh, Marjeta, Daniels, Danette L, Fuks, François
Published in The EMBO journal (06.03.2013)
Published in The EMBO journal (06.03.2013)
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Detection of cell-free microbial DNA using a contaminant-controlled analysis framework
Zozaya-Valdés, Enrique, Wong, Stephen Q, Raleigh, Jeanette, Hatzimihalis, Athena, Ftouni, Sarah, Papenfuss, Anthony T, Sandhu, Shahneen, Dawson, Mark A, Dawson, Sarah-Jane
Published in Genome Biology (23.06.2021)
Published in Genome Biology (23.06.2021)
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Click chemistry enables preclinical evaluation of targeted epigenetic therapies
Tyler, Dean S., Vappiani, Johanna, Cañeque, Tatiana, Lam, Enid Y. N., Ward, Aoife, Gilan, Omer, Chan, Yih-Chih, Hienzsch, Antje, Rutkowska, Anna, Werner, Thilo, Wagner, Anne J., Lugo, Dave, Gregory, Richard, Molina, Cesar Ramirez, Garton, Neil, Wellaway, Christopher R., Jackson, Susan, MacPherson, Laura, Figueiredo, Margarida, Stolzenburg, Sabine, Bell, Charles C., House, Colin, Dawson, Sarah-Jane, Hawkins, Edwin D., Drewes, Gerard, Prinjha, Rab K., Rodriguez, Raphaël, Grandi, Paola, Dawson, Mark A.
Published in Science (American Association for the Advancement of Science) (30.06.2017)
Published in Science (American Association for the Advancement of Science) (30.06.2017)
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A combination strategy targeting enhancer plasticity exerts synergistic lethality against BETi-resistant leukemia cells
Guo, Lei, Li, Jia, Zeng, Hongxiang, Guzman, Anna G, Li, Tingting, Lee, Minjung, Zhou, Yubin, Goodell, Margaret A, Stephan, Clifford, Davies, Peter J A, Dawson, Mark A, Sun, Deqiang, Huang, Yun
Published in Nature communications (06.02.2020)
Published in Nature communications (06.02.2020)
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Heterochromatin protein 1 alpha (HP1α) undergoes a monomer to dimer transition that opens and compacts live cell genome architecture
Lou, Jieqiong, Deng, Qiji, Zhang, Xiaomeng, Bell, Charles C, Das, Andrew B, Bediaga, Naiara G, Zlatic, Courtney O, Johanson, Timothy M, Allan, Rhys S, Griffin, Michael D W, Paradkar, PrasadN, Harvey, Kieran F, Dawson, Mark A, Hinde, Elizabeth
Published in Nucleic acids research (28.08.2024)
Published in Nucleic acids research (28.08.2024)
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Molecular disease monitoring using circulating tumor DNA in myelodysplastic syndromes
Yeh, Paul, Dickinson, Michael, Ftouni, Sarah, Hunter, Tane, Sinha, Devbarna, Wong, Stephen Q., Agarwal, Rishu, Vedururu, Ravikiran, Doig, Kenneth, Fong, Chun Yew, Blombery, Piers, Westerman, David, Dawson, Mark A., Dawson, Sarah-Jane
Published in Blood (23.03.2017)
Published in Blood (23.03.2017)
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Dual Targeting of Bromodomain and Extraterminal Domain Proteins, and WNT or MAPK Signaling, Inhibits c-MYC Expression and Proliferation of Colorectal Cancer Cells
Tögel, Lars, Nightingale, Rebecca, Chueh, Anderly C, Jayachandran, Aparna, Tran, Hoanh, Phesse, Toby, Wu, Rui, Sieber, Oliver M, Arango, Diego, Dhillon, Amardeep S, Dawson, Mark A, Diez-Dacal, Beatriz, Gahman, Timothy C, Filippakopoulos, Panagis, Shiau, Andrew K, Mariadason, John M
Published in Molecular cancer therapeutics (01.06.2016)
Published in Molecular cancer therapeutics (01.06.2016)
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Circulating tumour DNA reflects treatment response and clonal evolution in chronic lymphocytic leukaemia
Yeh, Paul, Hunter, Tane, Sinha, Devbarna, Ftouni, Sarah, Wallach, Elise, Jiang, Damian, Chan, Yih-Chih, Wong, Stephen Q, Silva, Maria Joao, Vedururu, Ravikiran, Doig, Kenneth, Lam, Enid, Arnau, Gisela Mir, Semple, Timothy, Wall, Meaghan, Zivanovic, Andjelija, Agarwal, Rishu, Petrone, Pasquale, Jones, Kate, Westerman, David, Blombery, Piers, Seymour, John F, Papenfuss, Anthony T, Dawson, Mark A, Tam, Constantine S, Dawson, Sarah-Jane
Published in Nature communications (17.03.2017)
Published in Nature communications (17.03.2017)
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