Identification and profiling of 3,5-dimethyl-isoxazole-4-carboxylic acid [2-methyl-4-((2S,3′S)-2-methyl-[1,3′]bipyrrolidinyl-1′-yl)phenyl] amide as histamine H3 receptor antagonist for the treatment of depression
Gao, Zhongli, Hurst, William J., Czechtizky, Werngard, Hall, Daniel, Moindrot, Nicolas, Nagorny, Raisa, Pichat, Philippe, Stefany, David, Hendrix, James A., George, Pascal G.
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
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Journal Article
Identification and profiling of 3,5-dimethyl-isoxazole-4-carboxylic acid [2-methyl-4-((2S,3 ' S)-2-methyl-[1,3 ']bipyrrolidinyl-1 '-yl)phenyl] amide as histamine H-3 receptor antagonist for the treatment of depression
Gao, Zhongli, Hurst, William J., Czechtizky, Werngard, Hall, Daniel, Moindrot, Nicolas, Nagorny, Raisa, Pichat, Philippe, Stefany, David, Hendrix, James A., George, Pascal G.
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
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Journal Article
Identification and profiling of 3,5-dimethyl-isoxazole-4-carboxylic acid [2-methyl-4-((2S,3a2S)-2-methyl-[1,3a2]bipyrrolidinyl-1a2-yl)phe nyl] amide as histamine H3 receptor antagonist for the treatment of depression
Gao, Zhongli, Hurst, William, Czechtizky, Werngard, Hall, Daniel, Moindrot, Nicolas, Nagorny, Raisa, Pichat, Philippe, Stefany, David, Hendrix, James, George, Pascal
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
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Journal Article
The discovery of thienopyridine analogues as potent IκB kinase β inhibitors. Part II
Wu, Jiang-Ping, Fleck, Roman, Brickwood, Janice, Capolino, Alison, Catron, Katrina, Chen, Zhidong, Cywin, Charles, Emeigh, Jonathan, Foerst, Melissa, Ginn, John, Hrapchak, Matt, Hickey, Eugene, Hao, Ming-Hong, Kashem, Mohammed, Li, Jun, Liu, Weimin, Morwick, Tina, Nelson, Richard, Marshall, Daniel, Martin, Leslie, Nemoto, Peter, Potocki, Ian, Liuzzi, Michel, Peet, Gregory W., Scouten, Erika, Stefany, David, Turner, Michael, Weldon, Steve, Zimmitti, Clare, Spero, Denise, Kelly, Terence A.
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
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Journal Article
Understanding DP receptor antagonism using a CoMSIA approach
Mu, Lan, Aguiar, Joacy, Ardati, Ali, Cao, Bin, Gardner, Charles J., Gillespy, Tim, Harris, Keith, Lim, Sungtaek, Marcus, Robert, Morize, Isabelle, Parkar, Ashfaq, Stefany, David, Li, Yi, Vaz, Roy J., Cirovic, Dragan A.
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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Journal Article
Identification and profiling of 3,5-dimethyl-isoxazole-4-carboxylic acid [2-methyl-4-((2S,3'S)-2-methyl-[1,3']bipyrrolidinyl-1'-yl)phenyl] amide as histamine H(3) receptor antagonist for the treatment of depression
Gao, Zhongli, Hurst, William J, Czechtizky, Werngard, Hall, Daniel, Moindrot, Nicolas, Nagorny, Raisa, Pichat, Philippe, Stefany, David, Hendrix, James A, George, Pascal G
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
Get full text
Journal Article
The discovery of thienopyridine analogues as potent I[kappa]B kinase beta inhibitors. Part II
Wu, Jiang-Ping, Fleck, Roman, Brickwood, Janice, Capolino, Alison, Catron, Katrina, Chen, Zhidong, Cywin, Charles, Emeigh, Jonathan, Foerst, Melissa, Ginn, John, Hrapchak, Matt, Hickey, Eugene, Hao, Ming-Hong, Kashem, Mohammed, Li, Jun, Liu, Weimin, Morwick, Tina, Nelson, Richard, Marshall, Daniel, Martin, Leslie, Nemoto, Peter, Potocki, Ian, Liuzzi, Michel, Peet, Gregory W, Scouten, Erika, Stefany, David, Turner, Michael, Weldon, Steve, Zimmitti, Clare, Spero, Denise, Kelly, Terence A
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Get full text
Journal Article