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Published in Journal of medicinal chemistry (10.10.2013)
Published in Journal of medicinal chemistry (10.10.2013)
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Pharmacological inhibition of Stearoyl-CoA Desaturase 1 improves insulin sensitivity in insulin-resistant rat models
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Published in Journal of medicinal chemistry (23.05.2019)
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Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis
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Published in Journal of medicinal chemistry (14.02.2019)
Published in Journal of medicinal chemistry (14.02.2019)
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Year of Publication 21.11.2023
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Year of Publication 21.11.2023
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The Discovery of Tadalafil: A Novel and Highly Selective PDE5 Inhibitor. 2: 2,3,6,7,12,12a-hexahydropyrazino[1‘,2‘:1,6]pyrido[3,4-b]indole-1,4-dione Analogues
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Published in Journal of medicinal chemistry (09.10.2003)
Published in Journal of medicinal chemistry (09.10.2003)
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DENIS ALEXIS, BLOM PETRA MARCELLA, LAUGEOIS MAXIME, LE TIRAN ARNAUD, DAUGAN ALAIN, HOUSSEMAN CHRISTOPHER GAETAN, DUMOULIN AUDREY, CHRISTENSEN KENNETH, BOTEZ IULIANA, LAMOTTE YANN, FAUCHER NICOLAS
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Year of Publication 10.01.2023
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The Discovery of Tadalafil: A Novel and Highly Selective PDE5 Inhibitor. 1: 5,6,11,11a-Tetrahydro-1H-imidazo[1‘,5‘:1,6]pyrido[3,4-b]indole-1,3(2H)-dione Analogues
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Published in Journal of medicinal chemistry (09.10.2003)
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Deng, Hongfeng, Zhou, Jingye, Sundersingh, Flora, Messer, Jeffrey A, Somers, Donald O, Ajakane, Myriam, Arico-Muendel, Christopher C, Beljean, Arthur, Belyanskaya, Svetlana L, Bingham, Ryan, Blazensky, Emily, Boullay, Anne-Benedicte, Boursier, Eric, Chai, Jing, Carter, Paul, Chung, Chun-Wa, Daugan, Alain, Ding, Yun, Herry, Kenny, Hobbs, Clare, Humphries, Eric, Kollmann, Christopher, Nguyen, Van Loc, Nicodeme, Edwige, Smith, Sarah E, Dodic, Nerina, Ancellin, Nicolas
Published in ACS medicinal chemistry letters (14.04.2016)
Published in ACS medicinal chemistry letters (14.04.2016)
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Identification of 6-amino-1H-pyrazolo[3,4-d]pyrimidines with in vivo efficacy against visceral leishmaniasis
Thomas, Michael G, De Rycker, Manu, Ajakane, Myriam, Crouch, Sabrinia D, Campbell, Lorna, Daugan, Alain, Fra, Gloria, Guerrero, César, Mackenzie, Claire J, MacLean, Lorna, Manthri, Sujatha, Martin, Franck, Norval, Suzanne, Osuna-Cabello, Maria, Riley, Jennifer, Shishikura, Yoko, Miguel-Siles, Juan, Simeons, Frederick R C, Stojanovski, Laste, Thomas, John, Thompson, Stephen, Velasco, Raul F, Fiandor, Jose M, Wyatt, Paul G, Read, Kevin D, Gilbert, Ian H, Miles, Timothy J
Published in MedChemComm (01.10.2020)
Published in MedChemComm (01.10.2020)
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NICOLAS S GEORGE, DAUGAN ALAIN CLAUDE-MARIE, NICOLAS ERIC FAUCHER, NIALL ANDREW ANDERSON, JAE U JEONG, BRYAN W KING, DAVID DUFF WISNOSKI, FREDERIC G DONCHE, CLARK A SEHON, GEMMA VICTORIA WHITE, PHILIP ANTHONY HARRIS, DEEPAK BANDYOPADHYAY, PATRICK M EIDAM
Year of Publication 16.09.2021
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Year of Publication 16.09.2021
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HETEROCYCLIC AMIDES AS KINASE INHIBITORS
NICOLAS S GEORGE, DAUGAN ALAIN CLAUDE-MARIE, NICOLAS ERIC FAUCHER, NIALL ANDREW ANDERSON, JAE U JEONG, BRYAN W KING, DAVID DUFF WISNOSKI, FREDERIC G DONCHE, CLARK A SEHON, GEMMA VICTORIA WHITE, PHILIP ANTHONY HARRIS, DEEPAK BANDYOPADHYAY, PATRICK M EIDAM
Year of Publication 10.09.2020
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Year of Publication 10.09.2020
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Published in RSC medicinal chemistry (21.10.2020)
Published in RSC medicinal chemistry (21.10.2020)
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Identification of 6-amino-1H-pyrazolo[3,4-d]pyrimidines with in vivo efficacy against visceral leishmaniasis† †Electronic supplementary information (ESI) available. See DOI: 10.1039/d0md00203h
Thomas, Michael G., De Rycker, Manu, Ajakane, Myriam, Crouch, Sabrinia D., Campbell, Lorna, Daugan, Alain, Fra, Gloria, Guerrero, César, Mackenzie, Claire J., MacLean, Lorna, Manthri, Sujatha, Martin, Franck, Norval, Suzanne, Osuna-Cabello, Maria, Riley, Jennifer, Shishikura, Yoko, Miguel-Siles, Juan, Simeons, Frederick R. C., Stojanovski, Laste, Thomas, John, Thompson, Stephen, Velasco, Raul F., Fiandor, Jose M., Wyatt, Paul G., Read, Kevin D., Gilbert, Ian H., Miles, Timothy J.
Published in RSC medicinal chemistry (06.08.2020)
Published in RSC medicinal chemistry (06.08.2020)
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Year of Publication 18.05.2018
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Year of Publication 18.05.2018
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Year of Publication 12.01.2018
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The Discovery of Tadalafil: A Novel and Highly Selective PDE5 Inhibitor. 1: 5,6,11,11a-Tetrahydro-1 H -imidazo[1‘,5‘:1,6]pyrido[3,4- b ]indole-1,3(2 H )-dione Analogues
Daugan, Alain, Grondin, Pascal, Ruault, Cécile, Le Monnier de Gouville, Anne-Charlotte, Coste, Hervé, Kirilovsky, Jorge, Hyafil, François, Labaudinière, Richard
Published in Journal of medicinal chemistry (01.10.2003)
Published in Journal of medicinal chemistry (01.10.2003)
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Year of Publication 25.07.2024
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Year of Publication 25.07.2024
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