First‐in‐human study of JNJ‐63709178, a CD123/CD3 targeting antibody, in relapsed/refractory acute myeloid leukemia
Boyiadzis, Michael, Desai, Pinkal, Daskalakis, Nikki, Donnellan, William, Ferrante, Lucille, Goldberg, Jenna D., Grunwald, Michael R., Guttke, Christina, Li, Xiang, Perez‐Simon, Jose Antonio, Salamero, Olga, Tucker, Trevor, Xu, Xiaoying, Yang, Jay, Pemmaraju, Naveen, Alonso‐Dominguez, Juan Manuel
Published in Clinical and translational science (01.03.2023)
Published in Clinical and translational science (01.03.2023)
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First‐in‐human study of JNJ‐67571244, a CD33 × CD3 bispecific antibody, in relapsed/refractory acute myeloid leukemia and myelodysplastic syndrome
Narayan, Rupa, Piérola, Ana Alfonso, Donnellan, William B., Yordi, Antonieta Molero, Abdul‐Hay, Maher, Platzbecker, Uwe, Subklewe, Marion, Kadia, Tapan Mahendra, Alonso‐Domínguez, Juan Manuel, McCloskey, James, Bradford, Kathryn, Curtis, Martin, Daskalakis, Nikki, Guttke, Christina, Safer, Karim, Hiebert, Brett, Murphy, Joseph, Li, Xiang, Duchin, Ken, Esteban, Daniel
Published in Clinical and translational science (01.03.2024)
Published in Clinical and translational science (01.03.2024)
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Clopidogrel pharmacodynamics and pharmacokinetics in the fed and fasted state: a randomized crossover study of healthy men
Hurbin, Fabrice, Boulenc, Xavier, Daskalakis, Nikki, Farenc, Christine, Taylor, Theresa, Bonneau, Damien, Lacreta, Frank, Cheng, Sue, Sultan, Eric
Published in Journal of clinical pharmacology (01.10.2012)
Published in Journal of clinical pharmacology (01.10.2012)
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Preclinical Efficacy of the Menin-KMT2A Inhibitor JNJ-75276617 in Combination with Venetoclax and Azacitidine in AML
Kwon, Min Chul, Verhulst, Tinne, Goffin, Dries, Marien, Ann, Verbist, Bie, Guttke, Christina, Thuring, Jan Willem, Ferrante, Lucille, Daskalakis, Nikki, Pietsch, E. Christine, Elsayed, Yusri, Packman, Kathryn, Philippar, Ulrike
Published in Blood (02.11.2023)
Published in Blood (02.11.2023)
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A First-in-Human Phase 1 Study of the Menin-KMT2A (MLL1) Inhibitor JNJ-75276617 in Adult Patients with Relapsed/Refractory Acute Leukemia Harboring KMT2A or NPM1 Alterations
Jabbour, Elias, Searle, Emma, Abdul-Hay, Maher, Abedin, Sameem, Aldoss, Ibrahim, Alfonso Piérola, Ana, Alonso-Dominguez, Juan Manuel, Chevallier, Patrice, Cost, Carrye, Daskalakis, Nikki, Dillon, Richard, Dunavin, Neil, Esteve, Jordi, Fathi, Amir T., Fedele, Pasquale L., Ferrante, Lucille, Garciaz, Sylvain, Guttke, Christina, Gyan, Emmanuel, Hiebert, Brett, Kwon, Min Chul, Miller, Jonathan, Ng, Teng Fong, Packman, Kathryn, Philippar, Ulrike, Pigneux, Arnaud, Recher, Christian, Salamero, Olga, Sanga, Madhu, Stone, Richard M, Tan, Peter, Thuring, Jan Willem, Tucker, Trevor, Vyas, Paresh
Published in Blood (02.11.2023)
Published in Blood (02.11.2023)
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Preclinical efficacy of the potent, selective menin-KMT2A inhibitor JNJ-75276617 (bleximenib) in KMT2A- and NPM1-altered leukemias
Kwon, Min Chul, Thuring, Jan Willem, Querolle, Olivier, Dai, Xuedong, Verhulst, Tinne, Pande, Vineet, Marien, Ann, Goffin, Dries, Wenge, Daniela V., Yue, Hong, Cutler, Jevon A., Jin, Cyrus, Perner, Florian, Hogeling, Shanna M., Shaffer, Paul L., Jacobs, Frank, Vinken, Petra, Cai, Wei, Keersmaekers, Vikki, Eyassu, Filmon, Bhogal, Balpreet, Verstraeten, Karin, El Ashkar, Sara, Perry, Jennifer A., Jayaguru, Prathiba, Barreyro, Laura, Kuchnio, Anna, Darville, Nicolas, Krosky, Daniel, Urbanietz, Gregor, Verbist, Bie, Edwards, James P., Cowley, Glenn S., Kirkpatrick, Robert, Steele, Ruth, Ferrante, Lucille, Guttke, Christina, Daskalakis, Nikki, Pietsch, E. Christine, Wilson, David M., Attar, Ricardo, Elsayed, Yusri, Fischer, Eric S., Schuringa, Jan Jacob, Armstrong, Scott A., Packman, Kathryn, Philippar, Ulrike
Published in Blood (12.09.2024)
Published in Blood (12.09.2024)
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Pharmacological Characterization of JNJ-75276617, a Menin-KMT2A Inhibitor, As Targeted Treatment for KMT2A-Altered and NPM1-Mutant Acute Leukemia
Kwon, Min Chul, Querolle, Olivier, Dai, Xuedong, Thuring, Jan Willem, Verhulst, Tinne, Marien, Ann, Goffin, Dries, Cai, Wei, Keersmaekers, Vikki, Eyassu, Filmon, Verstraeten, Karin, El Ashkar, Sara, Hogeling, Shanna M, Jacob, Frank, Vinken, Petra, Darville, Nicolas, Pande, Vineet, Krosky, Daniel, Urbanietz, Gregor, Verbist, Bie, Ferrante, Lucille A., Drenberg, Christina Diane, Wilson, David, Attar, Ricardo M., Schuringa, Jan Jacob, Daskalakis, Nikki, Packman, Kathryn, Pietsch, Christine, Elsayed, Yusri, Philippar, Ulrike
Published in Blood (15.11.2022)
Published in Blood (15.11.2022)
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Abstract 1256: JNJ-74856665, a novel DHODH inhibitor, mediates potent anti-leukemic activity and differentiation in vitro and in vivo
Pietsch, Christine, Kuduk, Scott, Zhang, Xiaochun, Bush, Tammy, Kazmi, Faraz, Jacoby, Edgar, Zhang, Zhuming, DeRatt, Lindsey, Wang, Weixue, Patrick, Aaron, Steele, Andrew, Pastore, Friedericke, Greway, Tony, Daskalakis, Nikki, Bradford, Kathryn, Packman, Kathryn, Bignan, Gilles, Edwards, James, Attar, Ricardo, Elsayed, Yusri, Bussolari, Jacqueline, Philippar, Ulrike
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Mutation in the TRPC6 Cation Channel Causes Familial Focal Segmental Glomerulosclerosis
Winn, Michelle P, Conlon, Peter J, Lynn, Kelvin L, Farrington, Merry Kay, Creazzo, Tony, Hawkins, April F, Daskalakis, Nikki, Kwan, Shu Ying, Ebersviller, Seth, Burchette, James L, Pericak-Vance, Margaret A, Howell, David N, Vance, Jeffery M, Rosenberg, Paul B
Published in Science (American Association for the Advancement of Science) (17.06.2005)
Published in Science (American Association for the Advancement of Science) (17.06.2005)
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SAR650984, a CD38 Monoclonal Antibody In Patients With Selected CD38+ Hematological Malignancies- Data From a Dose-Escalation Phase I Study
Martin, Thomas G, Strickland, Stephen A., Glenn, Martha, Zheng, Wei, Daskalakis, Nikki, Mikhael, Joseph R.
Published in Blood (15.11.2013)
Published in Blood (15.11.2013)
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Abstract 563: A prospective biomarker study to demonstrate high MET expression and gene amplification in a subset of patients with advanced gastric cancer
Han-Kwang, Yang, Takeuchi, Hiroya, Kong, Seong-Ho, Lee, Hyuk-Joon, Shamiyeh, Elias, Daskalakis, Nikki, Goulaouic, Hélène, Castell, Christelle, Ozoux, Marie-Laure, Lim, Ju O., Wu, Kaida
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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조합 요법
PACKMAN KATHRYN ELIZABETH, DASKALAKIS NIKKI, ALI AHMED SUMIA, LI MING, XU YANPING, THURING JOHANNES WILHELMUS J, DENG XIANGJUN, FANG LICHAO, DAI XUEDONG, KWON MIN CHUL, PANDE VINEET, PIETSCH EVA CHRISTINE, LIU YINGTAO, GUTTKE CHRISTINA DIANE, VERHULST TINNE ANN J, QUEROLLE OLIVIER ALEXIS GEORGES, FU LIQIANG, NG ALICIA TEE FUAY, SUN YU, FERRANTE LUCILLE ANGELA, PHILIPPAR ULRIKE, BHOGAL BALPREET, LIU LIANZHU, DARVILLE NICOLAS FREDDY J, CAI WEI
Year of Publication 15.01.2024
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Year of Publication 15.01.2024
Patent
조합 요법
PANDE VINEET, PIETSCH EVA CHRISTINE, LIU YINGTAO, GUTTKE CHRISTINA DIANE, VERHULST TINNE ANN J, QUEROLLE OLIVIER ALEXIS GEORGES, PACKMAN KATHRYN ELIZABETH, DASKALAKIS NIKKI, FU LIQIANG, LI MING, XU YANPING, NG ALICIA TEE FUAY, SUN YU, FERRANTE LUCILLE ANGELA, THURING JOHANNES WILHELMUS J, DENG XIANGJUN, PHILIPPAR ULRIKE, BHOGAL BALPREET, FANG LICHAO, LIU LIANZHU, DAI XUEDONG, DARVILLE NICOLAS FREDDY J, KWON MIN CHUL, CAI WEI
Year of Publication 15.01.2024
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Year of Publication 15.01.2024
Patent
Abstract LB-294: Determination of JAK2 V617F allele burden in a phase II study of patients with myelofibrosis treated with SAR302503 using a sensitive and robust allele-specific qPCR assay
Liu, Feng, Talpaz, Moshe, Pardanani, Animesh, Jamieson, Catriona, Gabrail, Nashat, Tefferi, Ayalew, Lei, Tianlei, Greco, Rita, Adrian, Francisco, Daskalakis, Nikki, Lebedinsky, Claudia, Cohen, Pamela, Bergstrom, Donald
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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COMBINATION THERAPIES
Guttke, Christina Diane, Deng, Xiangjun, Ali-Ahmed, Sumia, Cai, Wei, Ng, Alicia Tee Fuay, Xu, Yanping, Li, Ming, Pietsch, Eva Christine, Thuring, Johannes Wilhelmus J, Querolle, Olivier Alexis Georges, Kwon, Min Chul, Liu, Yingtao, Dai, Xuedong, Packman, Kathryn Elizabeth, Fang, Lichao, Fu, Liqiang, Sun, Yu, Ferrante, Lucille Angela, Bhogal, Balpreet, Darville, Nicolas Freddy J, Liu, Lianzhu, Daskalakis, Nikki, Pande, Vineet, Philippar, Ulrike, Verhulst, Tinne Ann J
Year of Publication 08.08.2024
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Year of Publication 08.08.2024
Patent
COMBINATIONS COMPRISING A MENIN-MLL INHIBITOR AND AT LEAST ONE OTHER THERAPEUTIC AGENT
DASKALAKIS, Nikki, DARVILLE, Nicolas Freddy J, DAI, Xuedong, NG, Alicia Tee Fuay, DENG, Xiangjun, KWON, Min Chul, PIETSCH, Eva Christine, SCHEPENS, Wim Bert Griet, LIANG, Chao, DYUBANKOVA, Natalia Nikolaevna, JOUFFROY, Matthieu Dominique, ALI-AHMED, Sumia, FERRANTE, Lucille Angela, GUTTKE, Christina Diane, HULPIA, Fabian, ZHANG, Zhigao, LEPRI, Susan, PACKMAN, Kathryn Elizabeth, PANDE, Vineet, EDWARDS, James Patrick, CAI, Wei, QUEROLLE, Olivier Alexis Georges, SUN, Zhen, DEMIN, Samuël Dominique, THURING, Johannes Wilhelmus J, PHILIPPAR, Ulrike, LI, Ming
Year of Publication 06.06.2024
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Year of Publication 06.06.2024
Patent
COMBINATIONS COMPRISING A MENIN-MLL INHIBITOR AND A BCL-2 INHIBITOR
DASKALAKIS, Nikki, DARVILLE, Nicolas Freddy J, DAI, Xuedong, NG, Alicia Tee Fuay, DENG, Xiangjun, KWON, Min Chul, PIETSCH, Eva Christine, SCHEPENS, Wim Bert Griet, LIANG, Chao, DYUBANKOVA, Natalia Nikolaevna, JOUFFROY, Matthieu Dominique, ALI-AHMED, Sumia, FERRANTE, Lucille Angela, GUTTKE, Christina Diane, HULPIA, Fabian, ZHANG, Zhigao, LEPRI, Susan, PACKMAN, Kathryn Elizabeth, PANDE, Vineet, EDWARDS, James Patrick, CAI, Wei, QUEROLLE, Olivier Alexis Georges, SUN, Zhen, DEMIN, Samuël Dominique, THURING, Johannes Wilhelmus J, PHILIPPAR, Ulrike, LI, Ming
Year of Publication 06.06.2024
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Year of Publication 06.06.2024
Patent