Deletion of the MAD2L1 spindle assembly checkpoint gene is tolerated in mouse models of acute T-cell lymphoma and hepatocellular carcinoma
Foijer, Floris, Albacker, Lee A, Bakker, Bjorn, Spierings, Diana C, Yue, Ying, Xie, Stephanie Z, Davis, Stephanie, Lutum-Jehle, Annegret, Takemoto, Darin, Hare, Brian, Furey, Brinley, Bronson, Roderick T, Lansdorp, Peter M, Bradley, Allan, Sorger, Peter K
Published in eLife (20.03.2017)
Published in eLife (20.03.2017)
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Hepatitis C Virus Variants with Decreased Sensitivity to Direct-Acting Antivirals (DAAs) Were Rarely Observed in DAA-Naive Patients prior to Treatment
Bartels, Doug J, Sullivan, James C, Zhang, Eileen Z, Tigges, Ann M, Dorrian, Jennifer L, De Meyer, Sandra, Takemoto, Darin, Dondero, Elizabeth, Kwong, Ann D, Picchio, Gaston, Kieffer, Tara L
Published in Journal of Virology (01.02.2013)
Published in Journal of Virology (01.02.2013)
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Potentiation of tumor responses to DNA damaging therapy by the selective ATR inhibitor VX-970
Hall, Amy B, Newsome, Dave, Wang, Yuxin, Boucher, Diane M, Eustace, Brenda, Gu, Yong, Hare, Brian, Johnson, Mac A, Milton, Sean, Murphy, Cheryl E, Takemoto, Darin, Tolman, Crystal, Wood, Mark, Charlton, Peter, Charrier, Jean-Damien, Furey, Brinley, Golec, Julian, Reaper, Philip M, Pollard, John R
Published in Oncotarget (30.07.2014)
Published in Oncotarget (30.07.2014)
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Abstract PR02: Aneuploidy as a driver of liver cancer
Albacker, Lee A., Foijer, Floris, Yue, Ying, Takemoto, Darin, Davis, Stehpanie, Bronson, Rodney T., Sorger, Peter K.
Published in Cancer research (Chicago, Ill.) (15.11.2015)
Published in Cancer research (Chicago, Ill.) (15.11.2015)
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Abstract 3711: Pre-clinical combinations of ATR and PARP inhibitors: Defining target patient populations and dose schedule
Pollard, John, Reaper, Phil, Peek, Adele, Hughes, Stuart, Djeha, Hakim, Cummings, Steven, Larbi, Karen, Penney, Marina, Sullivan, Jim, Takemoto, Darin, DeFranco, Chris
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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PTERIDINONE COMPOUNDS AND USES THEREOF
GU WENXIN, MARINA PENNEY, LEDFORD BRIAN, MALTAIS FRANCOIS, DAVID DEININGER, NATHAN D WAAL, MARK WILLEM LEDEBOER, LI PAN, DENG HONGBO, LAUFFER DAVID J, GUY BEMIS, RUSSELL R HOOVER, MAC ARTHUR JOHNSON JR, DARIN TAKEMOTO, WANG TIANSHENG, MICHAEL BOYD, WARREN DORSCH
Year of Publication 22.08.2023
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Year of Publication 22.08.2023
Patent
ANTIPROLIFERATIVE COMPOUNDS AND USES THEREOF
STEVEN RONKIN, TANG QING, CLARKE MICHAEL, MARINA PENNEY, NATHAN D WAAL, LI PAN, DENG HONGBO, DONG HUIJUN, PHILIP COLLIER, LAUFFER DAVID J, GUY BEMIS, RUSSELL R HOOVER, HENRY YU, MAC ARTHUR JOHNSON JR, SHASHANK KUKAMI, DARIN TAKEMOTO, WANG TIANSHENG, MICHAEL BOYD, KISHAN CHANDUPATLA, WARREN DORSCH
Year of Publication 21.07.2023
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Year of Publication 21.07.2023
Patent
Abstract 1644: VX-970, the first-in-class inhibitor of the DNA damage repair enzyme ATR
Pollard, John, Reaper, Philip, Jones, Julie, Barnes, Christopher, Gladwell, Scott, Hughes, Stuart, Peak, Adele, Djeha, Hakim, Hall, Amy, Newsome, David, Wang, Yuxin, Boucher, Diane, Eustace, Brenda, Gu, Yong, Hare, Brian, Johnson, Mac, Milton, Sean, Murphy, Cheryl, Takemoto, Darin, Tolman, Crystal, Wood, Mark, Furey, Brinley, Penney, Marina, Li, Howard, Defranco, Christopher, Asmal, Mohammed, Fields, Scott
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Abstract LB-299: Comprehensive preclinical evaluation of VE-822, the first ATR-targeted drug candidate: a novel approach to transforming the efficacy of DNA damaging agents
Boucher, Diane, Charlton, Peter, Charrier, Jean-Damien, Furey, Brinley, Gu, Yong, Hall, Amy, Hare, Brian, Li, Howard, Milton, Sean, Murphy, Cheryl, Reaper, Philip, Takemoto, Darin, Udagawa, Taturo, Wang, Yuxin, Wood, Mark, Pollard, John
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Abstract 5491: Evaluation of the first potent and highly selective inhibitor of ATR kinase: An approach to selectively sensitize cancer cells to genotoxic drugs
Pollard, John R., Caron, Paul, Charlton, Peter, Charrier, Jean-Damien, Golec, Julian, Griffiths, Matthew, Hall, Amy, Hare, Brian, Long, Joanna, MacCormick, Somhairle, Milton, Sean, Murcko, Mark, Murphy, Cheryl, Peek, Adele, Reaper, Philip, Takemoto, Darin
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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METHODS OF CANCER TREATMENT USING AN ATR INHIBITOR
PENNEY, Marina, SULLIVAN, James, REAPER, Philip Michael, GEHO, David, TAKEMOTO, Darin, POLLARD, John Robert
Year of Publication 09.02.2022
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Year of Publication 09.02.2022
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METHODS OF CANCER TREATMENT USING AN ATR INHIBITOR
SULLIVAN, James, REAPER, Philip Michael, GEHO, David, PENNEY, Marina S, TAKEMOTO, Darin, POLLARD, John Robert
Year of Publication 01.07.2021
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Year of Publication 01.07.2021
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PTERIDINONE COMPOUNDS AND USES THEREOF
Takemoto, Darin, Li, Pan, Gu, Wenxin, Bemis, Guy, Dorsch, Warren, Boyd, Michael, Deng, Hongbo, Wang, Tiansheng, Ledeboer, Mark Willem, Penney, Marina, Ledford, Brian, LAUFFER, David, Maltais, Francois, Deininger, David, Waal, Nathan D, Hoover, Russell R, Johnson, JR., Mac Arthur
Year of Publication 05.10.2023
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Year of Publication 05.10.2023
Patent
METHODS OF CANCER TREATMENT USING AN ATR INHIBITOR
PENNEY, Marina, SULLIVAN, James, REAPER, Philip Michael, GEHO, David, TAKEMOTO, Darin, POLLARD, John Robert
Year of Publication 04.11.2020
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Year of Publication 04.11.2020
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ANTIPROLIFERATION COMPOUNDS AND USES THEREOF
WANG, Tiansheng, LAUFFER, David J, JOHNSON, Mac, Arthur, JR, WAAL, Nathan, D, YU, Henry, HOOVER, Russell, R, KULKARNI, Shashank, COLLIER, Philip, BEMIS, Guy, TAKEMOTO, Darin, DONG, Huijun, CHANDUPATLA, Kishan, CLARK, Michael, PENNEY, Marina, LI, Pan, DENG, Hongbo, RONKIN, Steven, DORSCH, Warren, BOYD, Michael, TANG, Qing
Year of Publication 05.06.2024
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Year of Publication 05.06.2024
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METHODS OF CANCER TREATMENT USING AN ATR INHIBITOR
PENNEY, Marina, SULLIVAN, James, REAPER, Philip Michael, GEHO, David, TAKEMOTO, Darin, POLLARD, John Robert
Year of Publication 29.07.2020
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Year of Publication 29.07.2020
Patent
Methods of cancer treatment using an ATR inhibitor
PENNEY, Marina, SULLIVAN, James, REAPER, Philip Michael, GEHO, David, TAKEMOTO, Darin, POLLARD, John Robert
Year of Publication 09.07.2020
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Year of Publication 09.07.2020
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ANTIPROLIFERATION COMPOUNDS AND USES THEREOF
HUIJUN DONG, STEVEN RONKIN, TIANSHENG WANG, DAVID J LAUFFER, MICHAEL CLARK, HONGBO DENG, MARINA PENNEY, Pan LI, NATHAN D WAAL, Qing TANG, PHILIP COLLIER, KULKARNI, SHASHANK, GUY BEMIS, RUSSELL R HOOVER, HENRY YU, MAC ARTHUR JOHNSON JR, DARIN TAKEMOTO, MICHAEL BOYD, KISHAN CHANDUPATLA, WARREN DORSCH
Year of Publication 31.01.2024
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Year of Publication 31.01.2024
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