Structure guided design of a series of sphingosine kinase (SphK) inhibitors
Gustin, Darin J., Li, Yihong, Brown, Matthew L., Min, Xiaoshan, Schmitt, Mike J., Wanska, Malgorzata, Wang, Xiaodong, Connors, Richard, Johnstone, Sheere, Cardozo, Mario, Cheng, Alan C., Jeffries, Shawn, Franks, Brendon, Li, Shyun, Shen, Shanling, Wong, Mariwil, Wesche, Holger, Xu, Guifen, Carlson, Timothy J., Plant, Matthew, Morgenstern, Kurt, Rex, Karen, Schmitt, Joanna, Coxon, Angela, Walker, Nigel, Kayser, Frank, Wang, Zhulun
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
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Structure-Based Design of Novel Inhibitors of the MDM2–p53 Interaction
Rew, Yosup, Sun, Daqing, Gonzalez-Lopez De Turiso, Felix, Bartberger, Michael D, Beck, Hilary P, Canon, Jude, Chen, Ada, Chow, David, Deignan, Jeffrey, Fox, Brian M, Gustin, Darin, Huang, Xin, Jiang, Min, Jiao, Xianyun, Jin, Lixia, Kayser, Frank, Kopecky, David J, Li, Yihong, Lo, Mei-Chu, Long, Alexander M, Michelsen, Klaus, Oliner, Jonathan D, Osgood, Tao, Ragains, Mark, Saiki, Anne Y, Schneider, Steve, Toteva, Maria, Yakowec, Peter, Yan, Xuelei, Ye, Qiuping, Yu, Dongyin, Zhao, Xiaoning, Zhou, Jing, Medina, Julio C, Olson, Steven H
Published in Journal of medicinal chemistry (14.06.2012)
Published in Journal of medicinal chemistry (14.06.2012)
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Journal Article
Sphingosine kinase activity is not required for tumor cell viability
Rex, Karen, Jeffries, Shawn, Brown, Matthew L, Carlson, Timothy, Coxon, Angela, Fajardo, Flordeliza, Frank, Brendon, Gustin, Darin, Kamb, Alexander, Kassner, Paul D, Li, Shyun, Li, Yihong, Morgenstern, Kurt, Plant, Matthew, Quon, Kim, Ruefli-Brasse, Astrid, Schmidt, Joanna, Swearingen, Elissa, Walker, Nigel, Wang, Zhulun, Watson, J E Vivienne, Wickramasinghe, Dineli, Wong, Mariwil, Xu, Guifen, Wesche, Holger
Published in PloS one (05.07.2013)
Published in PloS one (05.07.2013)
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Journal Article
Identification of potent, noncovalent fatty acid amide hydrolase (FAAH) inhibitors
Gustin, Darin J., Ma, Zhihua, Min, Xiaoshan, Li, Yihong, Hedberg, Christine, Guimaraes, Cris, Porter, Amy C., Lindstrom, Michelle, Lester-Zeiner, Dianna, Xu, Guifen, Carlson, Timothy J., Xiao, Shouhua, Meleza, Cesar, Connors, Richard, Wang, Zhulun, Kayser, Frank
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
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Journal Article
Discovery of potent and specific CXCR3 antagonists
Chen, Xiaoqi, Mihalic, Jeff, Deignan, Jeff, Gustin, Darin J., Duquette, Jason, Du, Xiaohui, Chan, Johann, Fu, Zice, Johnson, Michael, Li, An-Rong, Henne, Kirk, Sullivan, Tim, Lemon, Bryan, Ma, Ji, Miao, Shichang, Tonn, George, Collins, Tassie, Medina, Julio C.
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
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Journal Article
Imidazo-pyrazine derivatives as potent CXCR3 antagonists
Du, Xiaohui, Gustin, Darin J., Chen, Xiaoqi, Duquette, Jason, McGee, Lawrence R., Wang, Zhulun, Ebsworth, Karen, Henne, Kirk, Lemon, Bryan, Ma, Ji, Miao, Shichang, Sabalan, Emmanuel, Sullivan, Timothy J., Tonn, George, Collins, Tassie L., Medina, Julio C.
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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Journal Article
Optimization of the heterocyclic core of the quinazolinone-derived CXCR3 antagonists
Li, An-Rong, Johnson, Michael G., Liu, Jiwen, Chen, Xiaoqi, Du, Xiaohui, Mihalic, Jeffrey T., Deignan, Jeffrey, Gustin, Darin J., Duquette, Jason, Fu, Zice, Zhu, Liusheng, Marcus, Andrew P., Bergeron, Phillipe, McGee, Lawrence R., Danao, Jay, Lemon, Bryan, Carabeo, Teresa, Sullivan, Timothy, Ma, Ji, Tang, Liang, Tonn, George, Collins, Tassie L., Medina, Julio C.
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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Journal Article
Nonpeptidic, Noncovalent Inhibitors of the Cysteine Protease Cathepsin S
Thurmond, Robin L, Beavers, Mary Pat, Cai, Hui, Meduna, Steven P, Gustin, Darin J, Sun, Siquan, Almond, Harold J, Karlsson, Lars, Edwards, James P
Published in Journal of medicinal chemistry (23.09.2004)
Published in Journal of medicinal chemistry (23.09.2004)
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Journal Article
Discovery and SAR studies of a novel series of noncovalent cathepsin S inhibitors
Gustin, Darin J., Sehon, Clark A., Wei, Jianmei, Cai, Hui, Meduna, Steven P., Khatuya, Haripada, Sun, Siquan, Gu, Yin, Jiang, Wen, Thurmond, Robin L., Karlsson, Lars, Edwards, James P.
Published in Bioorganic & medicinal chemistry letters (15.03.2005)
Published in Bioorganic & medicinal chemistry letters (15.03.2005)
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Experimental Evidence for Chair-Like Transition States in Aldol Reactions of Methyl Ketone Lithium Enolates: Stereoselective Synthesis and Utilization of a Deuterium-Labeled Enolate as a Probe of Reaction Stereochemistry
Liu, Christopher M, Smith, William J, Gustin, Darin J, Roush, William R
Published in Journal of the American Chemical Society (27.04.2005)
Published in Journal of the American Chemical Society (27.04.2005)
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Journal Article
Total Synthesis of Olivomycin A
Roush, William R, Hartz, Richard A, Gustin, Darin J
Published in Journal of the American Chemical Society (10.03.1999)
Published in Journal of the American Chemical Society (10.03.1999)
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Journal Article
The SAR of 4-substituted (6,6-bicyclic) piperidine cathepsin S inhibitors
Grice, Cheryl A., Tays, Kevin, Khatuya, Haripada, Gustin, Darin J., Butler, Christopher R., Wei, Jianmei, Sehon, Clark A., Sun, Siquan, Gu, Yin, Jiang, Wen, Thurmond, Robin L., Karlsson, Lars, Edwards, James P.
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
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Journal Article
An NMR Method for Assigning Relative Stereochemistry to β-Hydroxy Ketones Deriving from Aldol Reactions of Methyl Ketones
Roush, William R, Bannister, Thomas D, Wendt, Michael D, VanNieuwenhze, Michael S, Gustin, Darin J, Dilley, Garrett J, Lane, Gregory C, Scheidt, Karl A, Smith, William J
Published in Journal of organic chemistry (14.06.2002)
Published in Journal of organic chemistry (14.06.2002)
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Journal Article
Studies on the Synthesis of Aureolic Acid Antibiotics: Acyloin Glycosidation Studies
Roush, William R, Briner, Karin, Kesler, Brenda S, Murphy, Megan, Gustin, Darin J
Published in Journal of organic chemistry (06.09.1996)
Published in Journal of organic chemistry (06.09.1996)
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Journal Article
Total Synthesis of Olivomycin A J. Am. Chem. Soc. 1999, 121, 1990−1991
Roush, William R, Hartz, Richard A, Gustin, Darin J
Published in Journal of the American Chemical Society (28.04.1999)
Published in Journal of the American Chemical Society (28.04.1999)
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Journal Article
Synthesis of the C(3)C(15) segment of rutamycin B via a C(8)C(9) fragment assembly aldol reaction: Metal dependence of the aldehyde and enolate diastereofacial selectivities
Gustin, Darin J, VanNieuwenhze, Michael S, Roush, William R
Published in Tetrahedron letters (15.05.1995)
Published in Tetrahedron letters (15.05.1995)
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Journal Article
Abstract LB-39: Sphingosine kinase activity is not required for tumor cell viability
Wesche, Holger, Brown, Matthew L., Carlson, Timothy J., Coxon, Angela, Frank, Brendon, Gustin, Darin J., Jeffries, Shawn, Li, Shyun, Li, Yihong, Morgenstern, Kurt, Plant, Matthew, Rex, Karen, Schmidt, Joanna, Shen, Shanling, Walker, Nigel, Wickramasinghe, Dineli, Xu, Guifen
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Journal Article
Design, Synthesis, and in Vitro Evaluation of Dipeptide-Based Antibody Minor Groove Binder Conjugates
Jeffrey, Scott C, Torgov, Michael Y, Andreyka, Jamie B, Boddington, Laura, Cerveny, Charles G, Denny, William A, Gordon, Kristine A, Gustin, Darin, Haugen, Jennifer, Kline, Toni, Nguyen, Minh T, Senter, Peter D
Published in Journal of medicinal chemistry (10.03.2005)
Published in Journal of medicinal chemistry (10.03.2005)
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