Search Results - "DANILA BRANCA" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Series of Novel and Highly Potent Cyclic Peptide PCSK9 Inhibitors Derived from an mRNA Display Screen and Optimized via Structure-Based Design

Series of Novel and Highly Potent Cyclic Peptide PCSK9 Inhibitors Derived from an mRNA Display Screen and Optimized via Structure-Based Design

by Alleyne, Candice, Amin, Rupesh P, Bhatt, Bhavana, Bianchi, Elisabetta, Blain, J. Craig, Boyer, Nicolas, Branca, Danila, Embrey, Mark W, Ha, Sookhee N, Jette, Kelli, Johns, Douglas G, Kerekes, Angela D, Koeplinger, Kenneth A, LaPlaca, Derek, Li, Nianyu, Murphy, Beth, Orth, Peter, Ricardo, Alonso, Salowe, Scott, Seyb, Kathleen, Shahripour, Aurash, Stringer, Joseph R, Sun, Yili, Tracy, Rodger, Wu, Chengwei, Xiong, Yusheng, Youm, Hyewon, Zokian, Hratch J, Tucker, Thomas J
Published in Journal of medicinal chemistry (25.11.2020)

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A Series of Novel, Highly Potent, and Orally Bioavailable Next-Generation Tricyclic Peptide PCSK9 Inhibitors

A Series of Novel, Highly Potent, and Orally Bioavailable Next-Generation Tricyclic Peptide PCSK9 Inhibitors

by Tucker, Thomas J, Embrey, Mark W, Alleyne, Candice, Amin, Rupesh P, Bass, Alan, Bhatt, Bhavana, Bianchi, Elisabetta, Branca, Danila, Bueters, Tjerk, Buist, Nicole, Ha, Sookhee N, Hafey, Mike, He, Huaibing, Higgins, John, Johns, Douglas G, Kerekes, Angela D, Koeplinger, Kenneth A, Kuethe, Jeffrey T, Li, Nianyu, Murphy, BethAnn, Orth, Peter, Salowe, Scott, Shahripour, Aurash, Tracy, Rodger, Wang, Weixun, Wu, Chengwei, Xiong, Yusheng, Zokian, Hratch J, Wood, Harold B, Walji, Abbas
Published in Journal of medicinal chemistry (25.11.2021)

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Journal Article

Orally Bioavailable Macrocyclic Peptide That Inhibits Binding of PCSK9 to the Low Density Lipoprotein Receptor

Orally Bioavailable Macrocyclic Peptide That Inhibits Binding of PCSK9 to the Low Density Lipoprotein Receptor

by Johns, Douglas G, Campeau, Louis-Charles, Banka, Puja, Bautmans, An, Bueters, Tjerk, Bianchi, Elisabetta, Branca, Danila, Bulger, Paul G, Crevecoeur, Inne, Ding, Fa-Xiang, Garbaccio, Robert M, Guetschow, Erik D, Guo, Yan, Ha, Sookhee N, Johnston, Jennifer M, Josien, Hubert, Kauh, Eunkyung A, Koeplinger, Kenneth A, Kuethe, Jeffrey T, Lai, Eseng, Lanning, Christine L, Lee, Anita Y H, Li, Li, Nair, Anilkumar G, O'Neill, Edward A, Stoch, S Aubrey, Thaisrivongs, David A, Tucker, Thomas J, Vachal, Petr, van Dyck, Kristien, Vanhoutte, Frederic P, Volckaert, Bram, Wolford, Dennis G, Xu, Andy, Zhao, Tian, Zhou, Dan, Zhou, Susan, Zhu, Xiaohong, Zokian, Hratch J, Walji, Abbas, Wood, Harold B
Published in Circulation (New York, N.Y.) (11.07.2023)

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Journal Article

PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR AND THEIR USE TO TREAT INFLAMMATORY DISEASES

PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR AND THEIR USE TO TREAT INFLAMMATORY DISEASES

by RAFFAELE INGENITO, RAYMOND PATCH, GREGORY THOMAS BOURNE, ROBERTO COSTANTE, SUN CHENGZAO, ASHOK BHANDARI, ELISABETTA BIANCHI, BRIAN TROY FREDERICK, SANDEEP SOMANI, DANILA BRANCA
Year of Publication 03.10.2023

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Patent

Identification of substituted pyrazolo[1,5-a]quinazolin-5(4H)-one as potent poly(ADP-ribose)polymerase-1 (PARP-1) inhibitors

Identification of substituted pyrazolo[1,5-a]quinazolin-5(4H)-one as potent poly(ADP-ribose)polymerase-1 (PARP-1) inhibitors

by Orvieto, Federica, Branca, Danila, Giomini, Claudia, Jones, Philip, Koch, Uwe, Ontoria, Jesus M., Palumbi, Maria Cecilia, Rowley, Michael, Toniatti, Carlo, Muraglia, Ester
Published in Bioorganic & medicinal chemistry letters (01.08.2009)

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Journal Article

2-Trifluoroacetylthiophene oxadiazoles as potent and selective class II human histone deacetylase inhibitors

2-Trifluoroacetylthiophene oxadiazoles as potent and selective class II human histone deacetylase inhibitors

by MURAGLIA, Ester, ALTAMURA, Sergio, JONES, Philip, BRANCA, Danila, CECCHETTI, Ottavia, FERRIGNO, Federica, ORSALE, Maria Vittoria, PALUMBI, Maria Cecilia, ROWLEY, Michael, SCARPELLI, Rita, STEINKÜHLER, Christian
Published in Bioorganic & medicinal chemistry (01.12.2008)

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Discovery of N-[(1-aryl-1H-indazol-5-yl)methyl]amides derivatives as smoothened antagonists for inhibition of the hedgehog pathway

Discovery of N-[(1-aryl-1H-indazol-5-yl)methyl]amides derivatives as smoothened antagonists for inhibition of the hedgehog pathway

by Dessole, Gabriella, Branca, Danila, Ferrigno, Federica, Kinzel, Olaf, Muraglia, Ester, Palumbi, Maria Cecilia, Rowley, Michael, Serafini, Sergio, Steinkühler, Christian, Jones, Philip
Published in Bioorganic & medicinal chemistry letters (01.08.2009)

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Journal Article

Identification and SAR of novel pyrrolo[1,2- a]pyrazin-1(2 H)-one derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1)

Identification and SAR of novel pyrrolo[1,2- a]pyrazin-1(2 H)-one derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1)

by Pescatore, Giovanna, Branca, Danila, Fiore, Fabrizio, Kinzel, Olaf, Bufi, Laura Llauger, Muraglia, Ester, Orvieto, Federica, Rowley, Michael, Toniatti, Carlo, Torrisi, Caterina, Jones, Philip
Published in Bioorganic & medicinal chemistry letters (01.02.2010)

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Journal Article

N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxamides as highly potent smoothened antagonists

N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxamides as highly potent smoothened antagonists

by Muraglia, Ester, Ontoria, Jesus M., Branca, Danila, Dessole, Gabriella, Bresciani, Alberto, Fonsi, Massimiliano, Giuliano, Claudio, Llauger Bufi, Laura, Monteagudo, Edith, Palumbi, Maria Cecilia, Torrisi, Caterina, Rowley, Michael, Steinkühler, Christian, Jones, Philip
Published in Bioorganic & medicinal chemistry letters (15.09.2011)

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Journal Article

Identification of aminoethyl pyrrolo dihydroisoquinolinones as novel poly(ADP-ribose) polymerase-1 inhibitors

Identification of aminoethyl pyrrolo dihydroisoquinolinones as novel poly(ADP-ribose) polymerase-1 inhibitors

by Branca, Danila, Cerretani, Mauro, Jones, Philip, Koch, Uwe, Orvieto, Federica, Palumbi, Maria Cecilia, Rowley, Michael, Toniatti, Carlo, Muraglia, Ester
Published in Bioorganic & medicinal chemistry letters (01.08.2009)

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Journal Article

Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazin-3(2 H)-ones as potent poly(ADP–ribose) polymerase-1 (PARP-1) inhibitors active in BRCA deficient cells

Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazin-3(2 H)-ones as potent poly(ADP–ribose) polymerase-1 (PARP-1) inhibitors active in BRCA deficient cells

by Ferrigno, Federica, Branca, Danila, Kinzel, Olaf, Lillini, Samuele, Llauger Bufi, Laura, Monteagudo, Edith, Muraglia, Ester, Rowley, Michael, Schultz-Fademrecht, Carsten, Toniatti, Carlo, Torrisi, Caterina, Jones, Philip
Published in Bioorganic & medicinal chemistry letters (01.02.2010)

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Journal Article

N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxa mide s as highly potent smoothened antagonists

N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxa mide s as highly potent smoothened antagonists

by Muraglia, Ester, Ontoria, Jesus M, Branca, Danila, Dessole, Gabriella, Bresciani, Alberto, Fonsi, Massimiliano, Giuliano, Claudio, Bufi, Laura Llauger, Monteagudo, Edith, Palumbi, Maria Cecilia, Torrisi, Caterina, Rowley, Michael, Steinkuehler, Christian, Jones, Philip
Published in Bioorganic & medicinal chemistry letters (15.09.2011)

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Journal Article

Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazi n -3(2H)-ones as potent poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors active in BRCA deficient cells

Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazi n -3(2H)-ones as potent poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors active in BRCA deficient cells

by Ferrigno, Federica, Branca, Danila, Kinzel, Olaf, Lillini, Samuele, Bufi, Laura Llauger, Monteagudo, Edith, Muraglia, Ester, Rowley, Michael, Schultz-Fademrecht, Carsten, Toniatti, Carlo, Torrisi, Caterina, Jones, Philip
Published in Bioorganic & medicinal chemistry letters (01.02.2010)

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Journal Article

POLYCYCLIC PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR

POLYCYCLIC PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR

by BIANCHI, Elisabetta, NEELAMKAVIL, Santhosh Francis, BRANCA, Danila, COSTANTE, Roberto, SUN, Chengzao, INGENITO, Raffaele, SOMANI, Sandeep, ZHANG, Jing, BARROS, Stephanie A
Year of Publication 25.07.2024

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Patent

LIPIDATED PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR

LIPIDATED PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR

by NEELAMKAVIL, Santhosh Francis, BRANCA, Danila, COSTANTE, Roberto, GUO, Boying, SUN, Chengzao, MARCOUX, David, SOMANI, Sandeep, THIEU, Tho, ZHANG, Jing, BARROS, Stephanie A
Year of Publication 25.07.2024

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Patent

Peptide inhibitors of interleukin-23 receptor and their use to treat inflammatory diseases

Peptide inhibitors of interleukin-23 receptor and their use to treat inflammatory diseases

by Frederick, Brian Troy, Bhandari, Ashok, Barros, Stephanie, Bianchi, Elisabetta, Somani, Sandeep, Branca, Danila, Patch, Raymond, Ingenito, Raffaele, Sun, Chengzao, Costante, Roberto
Year of Publication 25.06.2024

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Patent

PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR AND THEIR USE TO TREAT INFLAMMATORY DISEASES

PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR AND THEIR USE TO TREAT INFLAMMATORY DISEASES

by FREDERICK, Brian Troy, BIANCHI, Elisabetta, BRANCA, Danila, BOURNE, Gregory Thomas, PATCH, Raymond, COSTANTE, Roberto, SUN, Chengzao, INGENITO, Raffaele, SOMANI, Sandeep, BHANDARI, Ashok
Year of Publication 09.05.2024

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Patent

PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR

PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR

by HENDRICK, Charles, RINALDI, Antonia, FREDERICK, Brian Troy, BRANCA, Danila, PATCH, Raymond J, BOURNE, Gregory Thomas, SUN, Chengzao, INGENITO, Raffaele, SOMANI, Sandeep, LOLLOBRIGIDA, Martina, BIANCHI, Elisabetta, COSTANTINI, Willy, NEELAMKAVIL, Santhosh Francis, COSTANTE, Roberto, BARROS, Stephanie A, ZHANG, Jing, BHANDARI, Ashok
Year of Publication 29.08.2024

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Patent

Peptide Inhibitors of Interleukin-23 Receptor

Peptide Inhibitors of Interleukin-23 Receptor

by Frederick, Brian Troy, SUN, Chengzao, Zhang, Jing, Somani, Sandeep, Hendrick, Charles, Guo, Boying, Neelamkavil, Santhosh Francis, Thieu, Tho, Bhandari, Ashok, Branca, Danila, Marcoux, David, Bourne, Gregory Thomas, BARROS, Stephanie A, Costante, Roberto
Year of Publication 22.08.2024

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Patent

PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR

PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR

by HENDRICK, Charles, RINALDI, Antonia, FREDERICK, Brian Troy, BRANCA, Danila, PATCH, Raymond J, BOURNE, Gregory Thomas, SUN, Chengzao, INGENITO, Raffaele, SOMANI, Sandeep, LOLLOBRIGIDA, Martina, BIANCHI, Elisabetta, COSTANTINI, Willy, NEELAMKAVIL, Santhosh Francis, COSTANTE, Roberto, BARROS, Stephanie A, ZHANG, Jing, BHANDARI, Ashok
Year of Publication 25.07.2024

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