Search Results - "DANIEL-HENRI, CAIGNARD" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Effect of 6-Benzoyl-benzothiazol-2-one scaffold on the pharmacological profile of α-alkoxyphenylpropionic acid derived PPAR agonists

by Hurtevent, Aurélie, Le Naour, Morgan, Leclerc, Veronique, Carato, Pascal, Melnyk, Patricia, Hennuyer, Nathalie, Staels, Bart, Beucher-Gaudin, Monique, Caignard, Daniel-Henri, Dacquet, Catherine, Lebegue, Nicolas
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)

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Journal Article

Synthesis of Omeprazole Analogues and Evaluation of These as Potential Inhibitors of the Multidrug Efflux Pump NorA of Staphylococcus aureus

Synthesis of Omeprazole Analogues and Evaluation of These as Potential Inhibitors of the Multidrug Efflux Pump NorA of Staphylococcus aureus

by VIDAILLAC, Celine, GUILLON, Jean, ARPIN, Corinne, FORFAR-BARES, Isabelle, BOUBAKAR, B, GRELLET, Jean, MOREAU, Stephane, CAIGNARD, Daniel-Henri, JARRY, Christian, QUENTIN, Claudine
Published in Antimicrobial Agents and Chemotherapy (01.03.2007)

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Journal Article

Novel conformationally constrained analogues of agomelatine as new melatoninergic ligands

Novel conformationally constrained analogues of agomelatine as new melatoninergic ligands

by Rami, Marouan, Landagaray, Elodie, Ettaoussi, Mohamed, Boukhalfa, Koussayla, Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Published in Molecules (Basel, Switzerland) (24.12.2012)

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Journal Article

New radioligands for describing the molecular pharmacology of MT1 and MT2 melatonin receptors

New radioligands for describing the molecular pharmacology of MT1 and MT2 melatonin receptors

by Legros, Céline, Matthey, Ulrich, Grelak, Teresa, Pedragona-Moreau, Sandrine, Hassler, Werner, Yous, Saïd, Thomas, Emmanuel, Suzenet, Franck, Folleas, Benoît, Lefoulon, François, Berthelot, Pascal, Caignard, Daniel-Henri, Guillaumet, Gérald, Delagrange, Philippe, Brayer, Jean-Louis, Nosjean, Olivier, Boutin, Jean A
Published in International journal of molecular sciences (25.04.2013)

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Journal Article

Synthesis and biological evaluation of benzimidazole derivatives as potent AMP-activated protein kinase activators

Synthesis and biological evaluation of benzimidazole derivatives as potent AMP-activated protein kinase activators

by Charton, Julie, Girault-Mizzi, Sophie, Debreu-Fontaine, Marie-Ange, Foufelle, Fabienne, Hainault, Isabelle, Bizot-Espiard, Jean-Guy, Caignard, Daniel-Henri, Sergheraert, Christian
Published in Bioorganic & medicinal chemistry (01.07.2006)

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Journal Article

Effect of Oxime Ether Incorporation in Acyl Indole Derivatives on PPAR Subtype Selectivity

Effect of Oxime Ether Incorporation in Acyl Indole Derivatives on PPAR Subtype Selectivity

by Le Naour, Morgan, Leclerc, Veronique, Farce, Amaury, Caignard, Daniel-Henri, Hennuyer, Nathalie, Staels, Bart, Audinot-Bouchez, Valérie, Boutin, Jean-Albert, Lonchampt, Michel, Dacquet, Catherine, Ktorza, Alain, Berthelot, Pascal, Lebegue, Nicolas
Published in ChemMedChem (01.12.2012)

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Journal Article

Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1‑Benzyl-2-acylaminomethyl-tetrahydroquinolines

Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1‑Benzyl-2-acylaminomethyl-tetrahydroquinolines

by Spadoni, Gilberto, Bedini, Annalida, Lucarini, Simone, Mari, Michele, Caignard, Daniel-Henri, Boutin, Jean A, Delagrange, Philippe, Lucini, Valeria, Scaglione, Francesco, Lodola, Alessio, Zanardi, Franca, Pala, Daniele, Mor, Marco, Rivara, Silvia
Published in Journal of medicinal chemistry (24.09.2015)

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Journal Article

Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT1/MT2) and serotoninergic (5-HT2C) dual ligands

Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT1/MT2) and serotoninergic (5-HT2C) dual ligands

by Duroux, Romain, Rami, Marouan, Landagaray, Elodie, Ettaoussi, Mohamed, Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Yous, Saïd
Published in European journal of medicinal chemistry (01.12.2017)

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Journal Article

Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands

Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands

by Rivara, Silvia, Scalvini, Laura, Lodola, Alessio, Mor, Marco, Caignard, Daniel-Henri, Delagrange, Philippe, Collina, Simona, Lucini, Valeria, Scaglione, Francesco, Furiassi, Lucia, Mari, Michele, Lucarini, Simone, Bedini, Annalida, Spadoni, Gilberto
Published in Journal of medicinal chemistry (26.04.2018)

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Journal Article

Novel antitumor artemisinin derivatives targeting G1 phase of the cell cycle

Novel antitumor artemisinin derivatives targeting G1 phase of the cell cycle

by Li, Ying, Shan, Feng, Wu, Jin-Ming, Wu, Guang-Shao, Ding, Jian, Xiao, Dong, Yang, Wei-Yi, Atassi, Ghanem, Léonce, Stéphane, Caignard, Daniel-Henri, Renard, Pierre
Published in Bioorganic & medicinal chemistry letters (08.01.2001)

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Journal Article

Novel N‑Acetyl Bioisosteres of Melatonin: Melatonergic Receptor Pharmacology, Physicochemical Studies, and Phenotypic Assessment of Their Neurogenic Potential

Novel N‑Acetyl Bioisosteres of Melatonin: Melatonergic Receptor Pharmacology, Physicochemical Studies, and Phenotypic Assessment of Their Neurogenic Potential

by de la Fuente Revenga, Mario, Fernández-Sáez, Nerea, Herrera-Arozamena, Clara, Morales-García, José A, Alonso-Gil, Sandra, Pérez-Castillo, Ana, Caignard, Daniel-Henri, Rivara, Silvia, Rodríguez-Franco, María Isabel
Published in Journal of medicinal chemistry (25.06.2015)

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Journal Article

Synthesis of 2-arylfuro[3,2-b]pyridines: Effect of the C2-aryl group on melatoninergic activity

Synthesis of 2-arylfuro[3,2-b]pyridines: Effect of the C2-aryl group on melatoninergic activity

by Couhert, Audrey, Delagrange, Philippe, Caignard, Daniel-Henri, Chartier, Agnès, Suzenet, Franck, Guillaumet, Gérald
Published in European journal of medicinal chemistry (15.02.2016)

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Journal Article

Synthesis and pharmacological evaluation of imidazoline sites I1 and I2 selective ligands

Synthesis and pharmacological evaluation of imidazoline sites I1 and I2 selective ligands

by Anastassiadou, Maria, Danoun, Saı̈da, Crane, Louis, Baziard-Mouysset, Geneviève, Payard, Marc, Caignard, Daniel-Henri, Rettori, Marie-Claire, Renard, Pierre
Published in Bioorganic & medicinal chemistry (01.03.2001)

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Journal Article

Anti-diabetic activity of fused PPARγ-SIRT1 ligands with limited body-weight gain by mimicking calorie restriction and decreasing SGK1 expression

Anti-diabetic activity of fused PPARγ-SIRT1 ligands with limited body-weight gain by mimicking calorie restriction and decreasing SGK1 expression

by Pirat, Celine, Dacquet, Catherine, Leclerc, Veronique, Hennuyer, Nathalie, Beucher-Gaudin, Monique, Zanirato, Ghislaine, Géant, Anne, Staels, Bart, Ktorza, Alain, Farce, Amaury, Caignard, Daniel-Henri, Berthelot, Pascal, Lebegue, Nicolas
Published in European journal of medicinal chemistry (08.09.2017)

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Journal Article

New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation

New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation

by Landagaray, Elodie, Ettaoussi, Mohamed, Rami, Marouan, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Berthelot, Pascal, Yous, Saïd
Published in European journal of medicinal chemistry (15.02.2017)

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Journal Article

Synthesis of Aromatic Analogs of 8(S)-HETE and Their Biological Evaluation as Activators of the PPAR Nuclear Receptors

Synthesis of Aromatic Analogs of 8(S)-HETE and Their Biological Evaluation as Activators of the PPAR Nuclear Receptors

by Caijo, Frédéric, Mosset, Paul, Grée, René, Audinot-Bouchez, Valérie, Boutin, Jean, Renard, Pierre, Caignard, Daniel-Henri, Dacquet, Catherine
Published in European Journal of Organic Chemistry (01.05.2006)

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Book Review Journal Article

New melatonin (MT1/MT2) ligands: Design and synthesis of (8,9-dihydro-7H-furo[3,2-f]chromen-1-yl) derivatives

New melatonin (MT1/MT2) ligands: Design and synthesis of (8,9-dihydro-7H-furo[3,2-f]chromen-1-yl) derivatives

by Landagaray, Elodie, Ettaoussi, Mohamed, Leclerc, Véronique, Traoré, Balla, Perez, Valérie, Nosjean, Olivier, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Published in Bioorganic & medicinal chemistry (01.02.2014)

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Journal Article

Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives

Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives

by Landagaray, Elodie, Ettaoussi, Mohamed, Duroux, Romain, Boutin, Jean A., Caignard, Daniel-Henri, Delagrange, Philippe, Melnyk, Patricia, Berthelot, Pascal, Yous, Saïd
Published in European journal of medicinal chemistry (15.02.2016)

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Journal Article

New Fluorinated 1,2,4-Benzothiadiazine 1,1-Dioxides: Discovery of an Orally Active Cognitive Enhancer Acting through Potentiation of the 2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors

New Fluorinated 1,2,4-Benzothiadiazine 1,1-Dioxides: Discovery of an Orally Active Cognitive Enhancer Acting through Potentiation of the 2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors

by Francotte, Pierre, Goffin, Eric, Fraikin, Pierre, Lestage, Pierre, Van Heugen, Jean-Claude, Gillotin, Florian, Danober, Laurence, Thomas, Jean-Yves, Chiap, Patrice, Caignard, Daniel-Henri, Pirotte, Bernard, de Tullio, Pascal
Published in Journal of medicinal chemistry (25.02.2010)

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Journal Article Web Resource

Development of Thiophenic Analogues of Benzothiadiazine Dioxides as New Powerful Potentiators of 2‑Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid (AMPA) Receptors

Development of Thiophenic Analogues of Benzothiadiazine Dioxides as New Powerful Potentiators of 2‑Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid (AMPA) Receptors

by Francotte, Pierre, Goffin, Eric, Fraikin, Pierre, Graindorge, E, Lestage, Pierre, Danober, Laurence, Challal, Sylvie, Rogez, Nathalie, Nosjean, Olivier, Caignard, Daniel-Henri, Pirotte, Bernard, de Tullio, Pascal
Published in Journal of medicinal chemistry (24.10.2013)

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Journal Article Web Resource

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