Synthesis of the Pentacyclic Skeleton of the Indole Alkaloid Arboflorine
Leal, Raul A, Beaudry, Danial R, Alzghari, Saeed K, Sarpong, Richmond
Published in Organic letters (19.10.2012)
Published in Organic letters (19.10.2012)
Get full text
Journal Article
Fit-for-purpose synthesis of dual leucine zipper kinase (DLK) inhibitor GNE-834
Xu, Jie, Carrera, Diane E., Beaudry, Danial, Siu, Michael, Huestis, Malcolm P., Liu, Wendy, Angelaud, Rémy, Gosselin, Francis
Published in Tetrahedron letters (22.10.2020)
Published in Tetrahedron letters (22.10.2020)
Get full text
Journal Article
Magnesium Ethoxide Promoted Conversion of Nitriles to Amidines and Its Application in 5,6-Dihydroimidazobenzoxazepine Synthesis
Dalziel, Michael E, Deichert, Julie A, Carrera, Diane E, Beaudry, Danial, Han, Chong, Zhang, Haiming, Angelaud, Remy
Published in Organic letters (04.05.2018)
Published in Organic letters (04.05.2018)
Get full text
Journal Article
Development of a Practical and Greener Process for the Dual Leucine Zipper Kinase Inhibitor GDC-0134 Comprising Two S N Ar Reactions, Oxidation and Suzuki Coupling
Hoffmann-Emery, Fabienne, Niedermann, Katrin, Rege, Pankaj D., Konrath, Manuel, Lautz, Christian, Kraft, Anne Katrin, Steiner, Carine, Bliss, Fritz, Hell, André, Fischer, Rolf, Carrera, Diane E., Beaudry, Danial, Angelaud, Remy, Malhotra, Sushant, Gosselin, Francis
Published in Organic process research & development (18.02.2022)
Published in Organic process research & development (18.02.2022)
Get full text
Journal Article
Development of a Practical and Greener Process for the Dual Leucine Zipper Kinase Inhibitor GDC-0134 Comprising Two SNAr Reactions, Oxidation and Suzuki Coupling
Hoffmann-Emery, Fabienne, Niedermann, Katrin, Rege, Pankaj D, Konrath, Manuel, Lautz, Christian, Kraft, Anne Katrin, Steiner, Carine, Bliss, Fritz, Hell, André, Fischer, Rolf, Carrera, Diane E, Beaudry, Danial, Angelaud, Remy, Malhotra, Sushant, Gosselin, Francis
Published in Organic process research & development (18.02.2022)
Published in Organic process research & development (18.02.2022)
Get full text
Journal Article
Development of an Efficient Manufacturing Process for Reversible Bruton’s Tyrosine Kinase Inhibitor GDC-0853
Zhang, Haiming, Cravillion, Theresa, Lim, Ngiap-Kie, Tian, Qingping, Beaudry, Danial, Defreese, Jessica L, Fettes, Alec, James, Philippe, Linder, David, Malhotra, Sushant, Han, Chong, Angelaud, Remy, Gosselin, Francis
Published in Organic process research & development (17.08.2018)
Published in Organic process research & development (17.08.2018)
Get full text
Journal Article
Manufacture of the PI3K β‑Sparing Inhibitor Taselisib. Part 2: Development of a Highly Efficient and Regioselective Late-Stage Process
St-Jean, Frédéric, Remarchuk, Travis, Angelaud, Rémy, Carrera, Diane E, Beaudry, Danial, Malhotra, Sushant, McClory, Andrew, Kumar, Archana, Ohlenbusch, Gerd, Schuster, Andreas M, Gosselin, Francis
Published in Organic process research & development (17.05.2019)
Published in Organic process research & development (17.05.2019)
Get full text
Journal Article
PROCESS FOR PREPARING BTK INHIBITORS
TIAN QINGPING, ALEXANDER GMEHLING, SUSHANT MALHOTRA, DANIAL BEAUDRY, THERESA CRAVILLION, ZHANG HAIMING, LIM NGIAP-KIE, ALEC FETTES, FRANCIS GOSSELIN, STEFAN BACHMANN
Year of Publication 18.03.2021
Get full text
Year of Publication 18.03.2021
Patent
PROCESS FOR PREPARING BTK INHIBITORS
MALHOTRA, SUSHANT, GOSSELIN, FRANCIS, LIM, NGIAP-KIE, BACHMANN, STEPHAN, CRAVILLION, THERESA, TIAN, QINGPING, ZHANG, HAIMING, BEAUDRY, DANIAL, GMEHLING, ALEXANDER, FETTES, ALEC
Year of Publication 19.09.2023
Get full text
Year of Publication 19.09.2023
Patent
PROCESS FOR PREPARING BTK INHIBITORS
BACHMANN, Stephan, CRAVILLION, Theresa, ZHANG, Haiming, GMEHLING, Alexander, FETTES, Alec, BEAUDRY, Danial, MALHOTRA, Sushant, GOSSELIN, Francis, LIM, Ngiap-Kie, TIAN, Qingping
Year of Publication 10.08.2023
Get full text
Year of Publication 10.08.2023
Patent
Process for preparing BTK inhibitors
Beaudry, Danial, Fettes, Alec, Cravillion, Theresa, Malhotra, Sushant, Tian, Qingping, Gosselin, Francis, Lim, Ngiap-Kie, Gmehling, Alexander, Zhang, Haiming, Bachmann, Stephan
Year of Publication 30.05.2023
Get full text
Year of Publication 30.05.2023
Patent
INTERMEDIATES FOR THE SYNTHESIS OF BENZOXAZEPIN COMPOUNDS
ANGELAUD, Remy, CARRERA, Diane, E, BEAUDRY, Danial, R, ST-JEAN, Frederic, MALHOTRA, Sushant, REMARCHUK, Travis
Year of Publication 07.07.2021
Get full text
Year of Publication 07.07.2021
Patent
PROCESS FOR PREPARING BTK INHIBITORS
MALHOTRA, SUSHANT, GOSSELIN, FRANCIS, LIM, NGIAP-KIE, BACHMANN, STEPHAN, CRAVILLION, THERESA, TIAN, QINGPING, ZHANG, HAIMING, BEAUDRY, DANIAL, GMEHLING, ALEXANDER, FETTES, ALEC
Year of Publication 27.12.2021
Get full text
Year of Publication 27.12.2021
Patent
PROCESS FOR PREPARING BTK INHIBITORS
Beaudry, Danial, Fettes, Alec, Cravillion, Theresa, Malhotra, Sushant, Tian, Qingping, Gosselin, Francis, Lim, Ngiap-Kie, Gmehling, Alexander, Zhang, Haiming, Bachmann, Stephan
Year of Publication 24.12.2021
Get full text
Year of Publication 24.12.2021
Patent
PROCESS FOR PREPARING BTK INHIBITORS
CRAVILLION Theresa, MALHOTRA Sushant, GOSSELIN Francis, LIM Ngiap-Kie, BACHMANN Stephan, TIAN Qingping, FETTES Alec, BEAUDRY Danial, ZHANG Haiming, GMEHLING Alexander
Year of Publication 30.11.2021
Get full text
Year of Publication 30.11.2021
Patent
PROCESS FOR PREPARING BTK INHIBITORS
BACHMANN, Stephan, CRAVILLION, Theresa, ZHANG, Haiming, GMEHLING, Alexander, FETTES, Alec, BEAUDRY, Danial, MALHOTRA, Sushant, GOSSELIN, Francis, LIM, Ngiap-Kie, TIAN, Qingping
Year of Publication 18.08.2021
Get full text
Year of Publication 18.08.2021
Patent
PROCESS FOR PREPARING BTK INHIBITORS
BACHMANN, Stephan, CRAVILLION, Theresa, ZHANG, Haiming, GMEHLING, Alexander, FETTES, Alec, BEAUDRY, Danial, MALHOTRA, Sushant, GOSSELIN, Francis, LIM, Ngiap-Kie, TIAN, Qingping
Year of Publication 28.07.2021
Get full text
Year of Publication 28.07.2021
Patent
PROCESS FOR PREPARING BTK INHIBITORS
BACHMANN, Stephan, CRAVILLION, Theresa, ZHANG, Haiming, GMEHLING, Alexander, FETTES, Alec, BEAUDRY, Danial, MALHOTRA, Sushant, GOSSELIN, Francis, LIM, Ngiap-Kie, TIAN, Qingping
Year of Publication 26.05.2021
Get full text
Year of Publication 26.05.2021
Patent