Small-molecule agonists for the glucagon-like peptide 1 receptor
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Published in Proceedings of the National Academy of Sciences - PNAS (16.01.2007)
Published in Proceedings of the National Academy of Sciences - PNAS (16.01.2007)
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Optimization of Alkylidene Hydrazide Based Human Glucagon Receptor Antagonists. Discovery of the Highly Potent and Orally Available 3-Cyano-4-hydroxybenzoic Acid [1-(2,3,5,6-Tetramethylbenzyl)-1H-indol-4-ylmethylene]hydrazide
Madsen, Peter, Ling, Anthony, Plewe, Michael, Sams, Christian K, Knudsen, Lotte B, Sidelmann, Ulla G, Ynddal, Lars, Brand, Christian L, Andersen, Birgitte, Murphy, Douglas, Teng, Min, Truesdale, Larry, Kiel, Dan, May, John, Kuki, Atsuo, Shi, Shenghua, Johnson, Michael D, Teston, Kimberly Ann, Feng, Jun, Lakis, James, Anderes, Kenna, Gregor, Vlad, Lau, Jesper
Published in Journal of medicinal chemistry (19.12.2002)
Published in Journal of medicinal chemistry (19.12.2002)
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Small molecule ago-allosteric modulators of the human glucagon-like peptide-1 (hGLP-1) receptor
Teng, Min, Johnson, Michael D., Thomas, Christine, Kiel, Dan, Lakis, James N., Kercher, Tim, Aytes, Shelley, Kostrowicki, Jarek, Bhumralkar, Dilip, Truesdale, Larry, May, John, Sidelman, Ulla, Kodra, Janos T., Jørgensen, Anker Steen, Olesen, Preben Houlberg, de Jong, Johannes Cornelis, Madsen, Peter, Behrens, Carsten, Pettersson, Ingrid, Knudsen, Lotte Bjerre, Holst, Jens J., Lau, Jesper
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
Published in Bioorganic & medicinal chemistry letters (01.10.2007)
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New β-Alanine Derivatives Are Orally Available Glucagon Receptor Antagonists
Lau, Jesper, Behrens, Carsten, Sidelmann, Ulla G, Knudsen, Lotte B, Lundt, Behrend, Sams, Christian, Ynddal, Lars, Brand, Christian L, Pridal, Lone, Ling, Anthony, Kiel, Dan, Plewe, Michael, Shi, Shengua, Madsen, Peter
Published in Journal of medicinal chemistry (11.01.2007)
Published in Journal of medicinal chemistry (11.01.2007)
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Identification of Alkylidene Hydrazides as Glucagon Receptor Antagonists
Ling, Anthony, Hong, Yufeng, Gonzalez, Javier, Gregor, Vlad, Polinsky, Alex, Kuki, Atsuo, Shi, Shenghua, Teston, Kimberly, Murphy, Douglas, Porter, John, Kiel, Dan, Lakis, James, Anderes, Kenna, May, John, Knudsen, Lotte Bjerre, Lau, Jesper
Published in Journal of medicinal chemistry (13.09.2001)
Published in Journal of medicinal chemistry (13.09.2001)
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Human glucagon receptor antagonists based on alkylidene hydrazides
Ling, Anthony, Plewe, Michael, Gonzalez, Javier, Madsen, Peter, Sams, Christian K., Lau, Jesper, Gregor, Vlad, Murphy, Doug, Teston, Kimberly, Kuki, Atsuo, Shi, Shenghua, Truesdale, Larry, Kiel, Dan, May, John, Lakis, James, Anderes, Kenna, Iatsimirskaia, Eugenia, Sidelmann, Ulla G., Knudsen, Lotte B., Brand, Christian L., Polinsky, Alex
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
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Reduced beta-adrenergic receptor activation decreases G-protein expression and beta-adrenergic receptor kinase activity in porcine heart
Ping, P, Gelzer-Bell, R, Roth, D A, Kiel, D, Insel, P A, Hammond, H K
Published in The Journal of clinical investigation (01.03.1995)
Published in The Journal of clinical investigation (01.03.1995)
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Cloning of GRK2 cDNA from S49 murine lymphoma cells
Hughes, R J, Anderson, K L, Kiel, D, Insel, P A
Published in The American journal of physiology (01.03.1996)
Published in The American journal of physiology (01.03.1996)
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CROSS-REACTIVE DETERMINANTS AND METHODS FOR THEIR IDENTIFICATION
HARLAND RICHARD, PLOCHER THOMAS, JOHNSON TODD, KIEL DAN, CAMPOS MANUEL, HARBISON TRENT
Year of Publication 20.01.2011
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Year of Publication 20.01.2011
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Metodo para identificar polipeptidos que comprenden un determinante antigenico de reaccion cruzada que comprende las etapas de obtener un anticuerpo de un animal expuesto secuencialmente a dos desafios con dos polipeptidos con determinantes antigenicos de una misma especie, pero distinto serotipo
PLOCHER, THOMAS, KIEL, DAN, CAMPOS, MANUEL, HARLAND, RICHARD, HARBISON, TRENT, JOHNSON, TODD
Year of Publication 01.07.2011
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Year of Publication 01.07.2011
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NICHTPEPTIDISCHE ANTAGONISTEN DES GLP-1 REZEPTORS UND VERWENDUNGSMETHODEN
CHOU, TSO-SHENG, BYCHOWSKI, A, LING, L, KUKI, ATSUO, KIEL, DAN, HONG, YUFENG, DHANOA, S, TRUESDALE, KENNETH, GONZALEZ, JAVIER, GREGOR, EDWARD, RAJAPAKSE, JAGATH, TENG, MIN, JOHNSON, DAVID
Year of Publication 23.06.2005
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Year of Publication 23.06.2005
Patent
Non-peptide GLP-1 agonists
Teng, Min, Truesdale, Larry Kenneth, Bhumralkar, Dilip, Kiel, Dan, Johnson, Michael D, Thomas, Christine, Jorgensen, Anker Steen, Madsen, Peter, Olesen, Preben Houlberg, Knudsen, Liselotte Bjerre, Petterson, Ingrid Vivika, de Jong, Johannes Cornelis, Behrens, Carsten, Kodra, Janos Tibor, Lau, Jesper
Year of Publication 09.08.2005
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Year of Publication 09.08.2005
Patent
Non-peptide GLP-1 agonists
MADSEN PETER, OLESEN PREBEN HOULBERG, KNUDSEN LISELOTTE BJERRE, DE JONG JOHANNES CORNELIS, KIEL DAN, JOHNSON MICHAEL D, TENG MIN, BHUMRALKAR DILIP, THOMAS CHRISTINE, BEHRENS CARSTEN, KODRA JANOS TIBOR, LAU JESPER, TRUESDALE LARRY KENNETH, JORGENSEN ANKER STEEN, PETTERSON INGRID VIVIKA
Year of Publication 09.08.2005
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Year of Publication 09.08.2005
Patent
ANTAGONISTAS NAO-PEPTIDICOS DO RECEPTOR DE GLP-1 E METODOS DE UTILIZACAO
DHANOA, DALJIT, S, GREGOR, VLAD, EDWARD, CHOU, TSO-SHENG, BYCHOWSKI, RICHARD, A, JOHNSON, MICHAEL, DAVID, TRUESDALE, LARRY, KENNETH, RAJAPAKSE, RANJAN, JAGATH, LING, ANTHONY, L, KUKI, ATSUO, KIEL, DAN, GONZALEZ, JAVIER, TENG, MIN, YUFENG HONG
Year of Publication 31.05.2005
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Year of Publication 31.05.2005
Patent
NICHTPEPTIDISCHE ANTAGONISTEN DES GLP-1 REZEPTORS UND VERWENDUNGSMETHODEN
DHANOA, DALJIT, S, GREGOR, VLAD, EDWARD, CHOU, TSO-SHENG, BYCHOWSKI, RICHARD, A, JOHNSON, MICHAEL, DAVID, TRUESDALE, LARRY, KENNETH, RAJAPAKSE, RANJAN, JAGATH, LING, ANTHONY, L, KUKI, ATSUO, KIEL, DAN, HONG, YUFENG, GONZALEZ, JAVIER, TENG, MIN
Year of Publication 15.02.2005
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Year of Publication 15.02.2005
Patent
NON-PEPTIDE ANTAGONISTS OF GLP-1 RECEPTOR AND METHODS OF USE
DHANOA, DALJIT, S, GREGOR, VLAD, EDWARD, CHOU, TSO-SHENG, BYCHOWSKI, RICHARD, A, JOHNSON, MICHAEL, DAVID, TRUESDALE, LARRY, KENNETH, RAJAPAKSE, RANJAN, JAGATH, LING, ANTHONY, L, KUKI, ATSUO, KIEL, DAN, HONG, YUFENG, GONZALEZ, JAVIER, TENG, MIN
Year of Publication 02.02.2005
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Year of Publication 02.02.2005
Patent