Developability Assessment of Engineered Monoclonal Antibody Variants with a Complex Self-Association Behavior Using Complementary Analytical and in Silico Tools
Shan, Lu, Mody, Neil, Sormani, Pietro, Rosenthal, Kim L., Damschroder, Melissa M., Esfandiary, Reza
Published in Molecular pharmaceutics (03.12.2018)
Published in Molecular pharmaceutics (03.12.2018)
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Experimentally guided computational antibody affinity maturation with de novo docking, modelling and rational design
Cannon, Daniel A, Shan, Lu, Du, Qun, Shirinian, Lena, Rickert, Keith W, Rosenthal, Kim L, Korade, 3rd, Martin, van Vlerken-Ysla, Lilian E, Buchanan, Andrew, Vaughan, Tristan J, Damschroder, Melissa M, Popovic, Bojana
Published in PLoS computational biology (01.05.2019)
Published in PLoS computational biology (01.05.2019)
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Upregulation of annexin A1 protein expression in the intratumoral vasculature of human non-small-cell lung carcinoma and rodent tumor models
Allen, Kevin L, Cann, Jennifer, Zhao, Weiguang, Peterson, Norman, Lazzaro, Michelle, Zhong, Haihong, Wu, Herren, Dall'Acqua, William F, Borrok, M Jack, Damschroder, Melissa M, Tsui, Ping, Li, Qing
Published in PloS one (04.06.2020)
Published in PloS one (04.06.2020)
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MEDI-563, a humanized anti–IL-5 receptor α mAb with enhanced antibody-dependent cell-mediated cytotoxicity function
Kolbeck, Roland, PhD, Kozhich, Alexander, PhD, Koike, Masamichi, PhD, Peng, Li, PhD, Andersson, Cecilia K., PhD, Damschroder, Melissa M., BA, Reed, Jennifer L., PhD, Woods, Robert, MS, Dall'Acqua, William W., PhD, Stephens, Geoffrey L., PhD, Erjefalt, Jonas S., PhD, Bjermer, Leif, MD, Humbles, Alison A., PhD, Gossage, David, MD, Wu, Herren, PhD, Kiener, Peter A., PhD, Spitalny, George L., PhD, Mackay, Charles R., PhD, Molfino, Nestor A., MD, Coyle, Anthony J., PhD
Published in Journal of allergy and clinical immunology (01.06.2010)
Published in Journal of allergy and clinical immunology (01.06.2010)
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Journal Article
Correction: Upregulation of annexin A1 protein expression in the intratumoral vasculature of human non-small-cell lung carcinoma and rodent tumor models
Allen, Kevin L, Cann, Jennifer, Zhao, Weiguang, Peterson, Norman, Lazzaro, Michelle, Zhong, Haihong, Wu, Herren, Dall'Acqua, William F, Borrok, M Jack, Damschroder, Melissa M, Tsui, Ping, Li, Qing
Published in PloS one (17.05.2021)
Published in PloS one (17.05.2021)
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Molecular basis for antagonistic activity of anifrolumab, an anti-interferon-α receptor 1 antibody
Peng, Li, Oganesyan, Vaheh, Wu, Herren, Dall'Acqua, William F, Damschroder, Melissa M
Published in mAbs (04.03.2015)
Published in mAbs (04.03.2015)
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Mechanisms of Neutralization of a Human Anti-α-toxin Antibody
Oganesyan, Vaheh, Peng, Li, Damschroder, Melissa M., Cheng, Li, Sadowska, Agnieszka, Tkaczyk, Christine, Sellman, Bret R., Wu, Herren, Dall'Acqua, William F.
Published in The Journal of biological chemistry (24.10.2014)
Published in The Journal of biological chemistry (24.10.2014)
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Inhibition of CD73 AMP hydrolysis by a therapeutic antibody with a dual, non-competitive mechanism of action
Geoghegan, James C, Diedrich, Gundo, Lu, Xiaojun, Rosenthal, Kim, Sachsenmeier, Kris F, Wu, Herren, Dall'Acqua, William F, Damschroder, Melissa M
Published in mAbs (02.04.2016)
Published in mAbs (02.04.2016)
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Generation and Characterization of an IgG4 Monomeric Fc Platform
Shan, Lu, Colazet, Magali, Rosenthal, Kim L, Yu, Xiang-Qing, Bee, Jared S, Ferguson, Andrew, Damschroder, Melissa M, Wu, Herren, Dall'Acqua, William F, Tsui, Ping, Oganesyan, Vaheh
Published in PloS one (01.08.2016)
Published in PloS one (01.08.2016)
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Antitumor activity of AZD0754, a dnTGFβRII-armored, STEAP2-targeted CAR-T cell therapy, in prostate cancer
Zanvit, Peter, van Dyk, Dewald, Fazenbaker, Christine, McGlinchey, Kelly, Luo, Weichuan, Pezold, Jessica M, Meekin, John, Chang, Chien-Ying, Carrasco, Rosa A, Breen, Shannon, Cheung, Crystal Sao-Fong, Endlich-Frazier, Ariel, Clark, Benjamin, Chu, Nina J, Vantellini, Alessio, Martin, Philip L, Hoover, Clare E, Riley, Kenesha, Sweet, Steve M, Chain, David, Kim, Yeoun Jin, Tu, Eric, Harder, Nathalie, Phipps, Sandrina, Damschroder, Melissa, Gilbreth, Ryan N, Cobbold, Mark, Moody, Gordon, Bosco, Emily E
Published in The Journal of clinical investigation (15.11.2023)
Published in The Journal of clinical investigation (15.11.2023)
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Mitigation of reversible self-association and viscosity in a human IgG1 monoclonal antibody by rational, structure-guided Fv engineering
Geoghegan, James C, Fleming, Ryan, Damschroder, Melissa, Bishop, Steven M, Sathish, Hasige A, Esfandiary, Reza
Published in mAbs (03.07.2016)
Published in mAbs (03.07.2016)
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Blocking endothelial lipase with monoclonal antibody MEDI5884 durably increases high density lipoprotein in nonhuman primates and in a phase 1 trial
Le Lay, John E, Du, Qun, Mehta, Minal B, Bhagroo, Nicholas, Hummer, B Timothy, Falloon, Judith, Carlson, Glenn, Rosenbaum, Anton I, Jin, ChaoYu, Kimko, Holly, Tsai, Lan-Feng, Novick, Steven, Cook, Bill, Han, David, Han, Chang Yeop, Vaisar, Tomas, Chait, Alan, Karathanasis, Sotirios K, Rhodes, Christopher J, Hirshberg, Boaz, Damschroder, Melissa M, Hsia, Judith, Grimsby, Joseph S
Published in Science translational medicine (21.04.2021)
Published in Science translational medicine (21.04.2021)
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Journal Article
Toward enhancement of antibody thermostability and affinity by computational design in the absence of antigen
Hutchinson, Mark, Ruffolo, Jeffrey A., Haskins, Nantaporn, Iannotti, Michael, Vozza, Giuliana, Pham, Tony, Mehzabeen, Nurjahan, Shandilya, Harini, Rickert, Keith, Croasdale-Wood, Rebecca, Damschroder, Melissa, Fu, Ying, Dippel, Andrew, Gray, Jeffrey J., Kaplan, Gilad
Published in mAbs (31.12.2024)
Published in mAbs (31.12.2024)
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Journal Article
Long-acting antibody ligand mimetics for HER4-selective agonism
Shan, Lu, Cook, Kimberly M, Haskins, Nantaporn, Omar, Bilal, Jiang, Yu, Garcia, Andrew, Koksal, Adem, Oganesyan, Vaheh, Rosenthal, Kim, Wu, Herren, Dall'Acqua, William F, Damschroder, Melissa M
Published in Scientific reports (14.10.2020)
Published in Scientific reports (14.10.2020)
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Bi-epitope SPR surfaces: a solution to develop robust immunoassays
Peng, Li, Damschroder, Melissa M, Wu, Herren, Dall'Acqua, William F
Published in PloS one (05.11.2014)
Published in PloS one (05.11.2014)
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A Monoclonal Antibody to ADAM17 Inhibits Tumor Growth by Inhibiting EGFR and Non-EGFR-Mediated Pathways
Rios-Doria, Jonathan, Sabol, Darrin, Chesebrough, Jon, Stewart, Dave, Xu, Linda, Tammali, Ravinder, Cheng, Li, Du, Qun, Schifferli, Kevin, Rothstein, Ray, Leow, Ching Ching, Heidbrink-Thompson, Jenny, Jin, Xiaofang, Gao, Changshou, Friedman, Jay, Wilkinson, Brandy, Damschroder, Melissa, Pierce, Andrew J, Hollingsworth, Robert E, Tice, David A, Michelotti, Emil F
Published in Molecular cancer therapeutics (01.07.2015)
Published in Molecular cancer therapeutics (01.07.2015)
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Discovery and characterization of potent IL-21 neutralizing antibodies via a novel alternating antigen immunization and humanization strategy
Varkey, Reena, Du, Qun, Karnell, Jodi L, Xiao, Xiaodong, Casey, Kerry A, Woods, Rob, Rosenthal, Kim, Wilson, Susan, Dall'Acqua, William F, Wu, Herren, Herbst, Ronald, Ettinger, Rachel, Damschroder, Melissa
Published in PloS one (25.01.2019)
Published in PloS one (25.01.2019)
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