6-Methyl-2,4-Disubstituted Pyridazin-3(2H)-ones: A Novel Class of Small-Molecule Agonists for Formyl Peptide Receptors
Cilibrizzi, Agostino, Quinn, Mark T, Kirpotina, Liliya N, Schepetkin, Igor A, Holderness, Jeff, Ye, Richard D, Rabiet, Marie-Josephe, Biancalani, Claudio, Cesari, Nicoletta, Graziano, Alessia, Vergelli, Claudia, Pieretti, Stefano, Dal Piaz, Vittorio, Giovannoni, Maria Paola
Published in Journal of medicinal chemistry (27.08.2009)
Published in Journal of medicinal chemistry (27.08.2009)
Get full text
Journal Article
Further studies on 2-arylacetamide pyridazin-3(2H)-ones: Design, synthesis and evaluation of 4,6-disubstituted analogs as formyl peptide receptors (FPRs) agonists
Giovannoni, Maria Paola, Schepetkin, Igor A., Cilibrizzi, Agostino, Crocetti, Letizia, Khlebnikov, Andrei I., Dahlgren, Claes, Graziano, Alessia, Dal Piaz, Vittorio, Kirpotina, Liliya N., Zerbinati, Serena, Vergelli, Claudia, Quinn, Mark T.
Published in European journal of medicinal chemistry (01.06.2013)
Published in European journal of medicinal chemistry (01.06.2013)
Get full text
Journal Article
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase
Crocetti, Letizia, Giovannoni, Maria Paola, Schepetkin, Igor A., Quinn, Mark T., Khlebnikov, Andrei I., Cilibrizzi, Agostino, Piaz, Vittorio Dal, Graziano, Alessia, Vergelli, Claudia
Published in Bioorganic & medicinal chemistry (01.08.2011)
Published in Bioorganic & medicinal chemistry (01.08.2011)
Get full text
Journal Article
Local anti-inflammatory effect and behavioral studies on new PDE4 inhibitors
Pieretti, Stefano, Dominici, Luigi, Di Giannuario, Amalia, Cesari, Nicoletta, Dal Piaz, Vittorio
Published in Life sciences (1973) (17.07.2006)
Published in Life sciences (1973) (17.07.2006)
Get full text
Journal Article
Functionalized pyrazoles and pyrazolo[3,4- d]pyridazinones: Synthesis and evaluation of their phosphodiesterase 4 inhibitory activity
Biagini, Pierfrancesco, Biancalani, Claudio, Graziano, Alessia, Cesari, Nicoletta, Giovannoni, Maria Paola, Cilibrizzi, Agostino, Piaz, Vittorio Dal, Vergelli, Claudia, Crocetti, Letizia, Delcanale, Maurizio, Armani, Elisabetta, Rizzi, Andrea, Puccini, Paola, Gallo, Paola Maria, Spinabelli, Daniele, Caruso, Paola
Published in Bioorganic & medicinal chemistry (15.05.2010)
Published in Bioorganic & medicinal chemistry (15.05.2010)
Get full text
Journal Article
Continental gabbros in the Dent Blanche Tectonic System (Western Alps): from the pre-Alpine crustal structure of the Adriatic palaeomargin to the geometry of an alleged subduction interface
Manzotti, Paola, Ballèvre, Michel, Dal Piaz, Giorgio Vittorio
Published in Journal of metamorphic geology (01.05.2017)
Published in Journal of metamorphic geology (01.05.2017)
Get full text
Journal Article
Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A1 adenosine receptor ligands
GIOVANNONI, Maria Paola, VERGELLI, Claudia, GAVALDA, Amadeu, CILIBRIZZI, Agostino, CROCETTI, Letizia, BIANCALANI, Claudio, GRAZIANO, Alessia, DAL PIAZ, Vittorio, LOZA, Maria Isabel, CADAVID, Maria Isabel, DIAZ, José Luis
Published in Bioorganic & medicinal chemistry (15.11.2010)
Published in Bioorganic & medicinal chemistry (15.11.2010)
Get full text
Journal Article
Phosphodiesterase 4 inhibitors, structurally unrelated to Rolipram, as promising agents for the treatment of asthma and other pathologies
Dal Piaz, Vittorio, Giovannoni, Maria Paola
Published in European Journal of Medicinal Chemistry (01.05.2000)
Published in European Journal of Medicinal Chemistry (01.05.2000)
Get full text
Book Review
Journal Article
4-Amino-5-vinyl-3(2 H)-pyridazinones and analogues as potent antinociceptive agents: Synthesis, SARs, and preliminary studies on the mechanism of action
Vergelli, Claudia, Giovannoni, Maria Paola, Pieretti, Stefano, Giannuario, Amalia Di, Piaz, Vittorio Dal, Biagini, Pierfrancesco, Biancalani, Claudio, Graziano, Alessia, Cesari, Nicoletta
Published in Bioorganic & medicinal chemistry (15.08.2007)
Published in Bioorganic & medicinal chemistry (15.08.2007)
Get full text
Journal Article
Synthesis of pyrrolo[2,3-d]pyridazinones as potent, subtype selective PDE4 inhibitors
Giovannoni, Maria P., Cesari, Nicoletta, Graziano, Alessia, Vergelli, Claudia, Biancalani, Claudio, Biagini, Pierfrancesco, Piaz, Vittorio Dal
Published in Journal of enzyme inhibition and medicinal chemistry (01.06.2007)
Published in Journal of enzyme inhibition and medicinal chemistry (01.06.2007)
Get full text
Journal Article
New pyrazolo[1′,5′:1,6]pyrimido[4,5- d]pyridazin-4(3 H)-ones as potent and selective PDE5 inhibitors
Feixas, Joan, Giovannoni, Maria Paola, Vergelli, Claudia, Gavaldà, Amadeu, Cesari, Nicoletta, Graziano, Alessia, Piaz, Vittorio Dal
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Get full text
Journal Article
Phenylpiperazinylalkylamino Substituted Pyridazinones as Potent α1 Adrenoceptor Antagonists
Barlocco, Daniela, Cignarella, Giorgio, Piaz, Vittorio Dal, Giovannoni, M. Paola, De Benedetti, Pier G, Fanelli, Francesca, Montesano, Federica, Poggesi, Elena, Leonardi, Amedeo
Published in Journal of medicinal chemistry (19.07.2001)
Published in Journal of medicinal chemistry (19.07.2001)
Get full text
Journal Article
4-Amino-3(2 H)-pyridazinones bearing arylpiperazinylalkyl groups and related compounds: synthesis and antinociceptive activity
Piaz, Vittorio Dal, Vergelli, Claudia, Giovannoni, Maria Paola, Scheideler, Mark A, Petrone, Giuseppe, Zaratin, Paola
Published in Farmaco (Società chimica italiana : 1989) (01.11.2003)
Published in Farmaco (Società chimica italiana : 1989) (01.11.2003)
Get full text
Journal Article
Le lettere di Felice Giordano a Quintino Sella. Parte seconda (7.1859-3.5.1875) - The Correspondence between Felice Giordano and Quintino Sella. Second Part (7.1859-3.5.1875)
Giorgio Vittorio Dal Piaz, Roberto Scoth
Published in Rivista di storia dell'Università di Torino (01.04.2022)
Get full text
Published in Rivista di storia dell'Università di Torino (01.04.2022)
Journal Article
Isoxazolo-[3,4-d]-pyridazin-7-(6H)-one as a Potential Substrate for New Aldose Reductase Inhibitors
Costantino, Luca, Rastelli, Giulio, Gamberini, M. Cristina, Giovannoni, M. Paola, Dal Piaz, Vittorio, Vianello, Paola, Barlocco, Daniela
Published in Journal of medicinal chemistry (03.06.1999)
Published in Journal of medicinal chemistry (03.06.1999)
Get full text
Journal Article
5,6-Diphenylpyridazine Derivatives as Acyl-CoA:Cholesterol Acyltransferase Inhibitors
Giovannoni, Maria Paola, Piaz, Vittorio Dal, Kwon, Byoung-Mog, Kim, Mi-Kyung, Kim, Young-Kook, Toma, Lucio, Barlocco, Daniela, Bernini, Franco, Canavesi, Monica
Published in Journal of medicinal chemistry (22.11.2001)
Published in Journal of medicinal chemistry (22.11.2001)
Get full text
Journal Article
Heterocyclic-fused 3(2H)-pyridazinones as potent and selective PDE IV inhibitors: Further structure-activity relationships and molecular modelling studies
Piaz, Vittorio Dal, Giovannoni, Maria Paola, Castellana, Carla, Palacios, José Maria, Beleta, Jorge, Doménech, Teresa, Segarra, Victor
Published in European journal of medicinal chemistry (01.10.1998)
Published in European journal of medicinal chemistry (01.10.1998)
Get full text
Journal Article