Identification of highly selective and potent orexin receptor 1 antagonists derived from a dual orexin receptor 1/2 antagonist based on the structural framework of pyrazoylethylbenzamide
Futamura, Aya, Nozawa, Dai, Araki, Yuko, Tamura, Yunoshin, Tokura, Seiken, Kawamoto, Hiroshi, Tokumaru, Yuichi, Kakihara, Sora, Aoki, Takeshi, Ohtake, Norikazu
Published in Bioorganic & medicinal chemistry (15.10.2017)
Published in Bioorganic & medicinal chemistry (15.10.2017)
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Structure–activity relationships of novel piperazines as antagonists for the melanocortin-4 receptor
Nozawa, Dai, Okubo, Taketoshi, Ishii, Takaaki, Kakinuma, Hiroyuki, Chaki, Shigeyuki, Okuyama, Shigeru, Nakazato, Atsuro
Published in Bioorganic & medicinal chemistry (01.03.2007)
Published in Bioorganic & medicinal chemistry (01.03.2007)
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Synthesis of Diphenylmethyl Analogues and Their Affinity for the Melanocortin-4 Receptor and the Serotonin Transporter
Nozawa, Dai, Okubo, Taketoshi, Ishii, Takaaki, Chaki, Shigeyuki, Okuyama, Shigeru, Nakazato, Atsuro
Published in Chemical & pharmaceutical bulletin (01.07.2007)
Published in Chemical & pharmaceutical bulletin (01.07.2007)
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A Novel Potent and Selective Histamine H 3 Receptor Antagonist Enerisant: In Vitro Profiles, In Vivo Receptor Occupancy, and Wake-Promoting and Procognitive Effects in Rodents
Hino, Noriko, Marumo, Toshiyuki, Kotani, Makiko, Shimazaki, Toshiharu, Kaku-Fukumoto, Ayaka, Hikichi, Hirohiko, Karasawa, Jun-Ichi, Tomishima, Yasumitsu, Komiyama, Hiroko, Tatsuda, Emi, Nozawa, Dai, Nakamura, Toshio, Chaki, Shigeyuki
Published in The Journal of pharmacology and experimental therapeutics (01.11.2020)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2020)
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Discovery of ORN0829, a potent dual orexin 1/2 receptor antagonist for the treatment of insomnia
Futamura, Aya, Suzuki, Ryo, Tamura, Yunoshin, Kawamoto, Hiroshi, Ohmichi, Mari, Hino, Noriko, Tokumaru, Yuichi, Kirinuki, Sora, Hiyoshi, Tetsuaki, Aoki, Takeshi, Kambe, Daiji, Nozawa, Dai
Published in Bioorganic & medicinal chemistry (01.07.2020)
Published in Bioorganic & medicinal chemistry (01.07.2020)
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Discovery of novel indole derivatives as potent and selective inhibitors of proMMP-9 activation
Nishikawa-Shimono, Rie, Kuwabara, Motoi, Fujisaki, Sho, Matsuda, Daisuke, Endo, Mayumi, Kamitani, Masafumi, Futamura, Aya, Nomura, Yusaku, Yamaguchi-Sasaki, Toru, Yabuuchi, Tetsuya, Yamaguchi, Chitose, Tanaka-Yamamoto, Nozomi, Satake, Shunya, Abe-Sato, Kumi, Funayama, Kosuke, Sakata, Mayumi, Takahashi, Shinji, Hirano, Koga, Fukunaga, Takuya, Uozumi, Yoriko, Kato, Sayaka, Tamura, Yunoshin, Nakamori, Tomoaki, Mima, Masashi, Mishima-Tsumagari, Chiemi, Nozawa, Dai, Imai, Yudai, Asami, Taiji
Published in Bioorganic & medicinal chemistry letters (01.01.2024)
Published in Bioorganic & medicinal chemistry letters (01.01.2024)
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Synthesis of sulfobacin A and B, new sulfonolipids isolated from Chryseobacterium sp
Takikawa, Hirosato, Muto, Shin-etsu, Nozawa, Dai, Kayo, Akihiro, Mori, Kenji
Published in Tetrahedron letters (17.09.1998)
Published in Tetrahedron letters (17.09.1998)
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Discovery and in vitro and in vivo profiles of N-ethyl-N-[2-[3-(5-fluoro-2-pyridinyl)-1H-pyrazol-1-yl]ethyl]-2-(2H-1,2,3-triazol-2-yl)-benzamide as a novel class of dual orexin receptor antagonist
Suzuki, Ryo, Nozawa, Dai, Futamura, Aya, Nishikawa-Shimono, Rie, Abe, Masahito, Hattori, Nobutaka, Ohta, Hiroshi, Araki, Yuko, Kambe, Daiji, Ohmichi, Mari, Tokura, Seiken, Aoki, Takeshi, Ohtake, Norikazu, Kawamoto, Hiroshi
Published in Bioorganic & medicinal chemistry (15.03.2015)
Published in Bioorganic & medicinal chemistry (15.03.2015)
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Triterpenoid total synthesis. Part 5. Synthetic disproof of the triterpene structure proposed for naurol A, a cytotoxic metabolite of a Pacific sponge
Nozawa, D, Takikawa, H, Mori, K
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
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Synthesis of sphingosine relatives. Part 22. Synthesis of sulfobacin A, B and flavocristamide A, new sulfonolipids isolated from Chryseobacterium sp
Takikawa, H, Nozawa, D, Kayo, A, Muto, S, Mori, K
Published in Journal of the Chemical Society, Perkin Transactions 1 (1999)
Published in Journal of the Chemical Society, Perkin Transactions 1 (1999)
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