Abstract A047: Discovery of potent and paralog selective PROTAC degraders of CBP or p300 proteins for the treatment of various cancers
Abbineni, Chandrasekhar, Thiyagarajan, Saravanan, T, Krishna Chaitanya, Apte, Achala, R, Naveen Kumar, Kumar, Avinash, Babu, Dabbeeru Madhu, S, Shwetha, Kamath, Aishwarya B, Mandal, Monalisha, Panigrahi, Rituparna, Marappan, Sivapriya, Mukherjee, Subhendu, Nellore, Kavitha, Chelur, Shekar, Ramachandra, Murali, Samajdar, Susanta
Published in Molecular cancer therapeutics (01.12.2023)
Published in Molecular cancer therapeutics (01.12.2023)
Get full text
Journal Article
Abstract 3303: Paralogue selective p300 degraders induce synthetic lethality in pre-clinical models of CBP-deficient and p300-dependent malignancies
Thiyagarajan, Saravanan, Abbineni, Chandrasekhar, Chaitanya T, Krishna, Apte, Achala, Iqbal, Iram Khan, Kumar R, Naveen, A B, Aravind, Kumar, Avinash, Babu, Dabbeeru Madhu, Shwetha, Shwetha, Manna, Ankita, Mandal, Monalisha, Panigrahi, Rituparna, Marappan, Sivapriya, Gore, Suraj T, Fairus, Mohamad, Jin, Lim Yang, Mukherjee, Subhendu, Daginakatte, Girish, Chelur, Shekar, Nellore, Kavitha, Ramachandra, Murali, Samajdar, Susanta
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Get full text
Journal Article
Abstract LB-317: Identification of a novel preclinical candidate for CDK7 inhibition
Satyam, Leena K., Poddutoori, Ramulu, Mukherjee, Subhendu, Marappan, Sivapriya, Gopinath, Sreevalsam, Basavaraju, Aravind, Kaza, Lakshmi Narayana, Pothuganti, Manoj Kumar, Nayak, Shilpa, C, Nandish, A, Amith, MV, Ravindra, Babu, Dabbeeru Madhu, A, Nagaraju, Tgore, Suraj, Antony, Thomas, Pandit, Chetan, Ramachandra, Murali, Chelur, Shekar, Daginakatte, Girish, Samajdar, Susanta
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Get full text
Journal Article
Pyrrolo [2,3-B] pyridine CDK9 kinase inhibitors
Risi Roberto M, Hansen Todd M, Curtin Michael, Mastracchio Anthony, Penning Thomas, Gong Jianchun, Song Xiaohong, Dabbeeru Madhu Babu, Goswami Rajeev, Iguturi Omprakash Reddy, Tong Yunsong, Zhu Guidong, Tao Zhi-fu, Michaelides Michael, Miyashiro Juliem, Clark Richard F, Lai Chunqiu, Bruncko Milan, Ji Zhiqin, Souers Andrew, Frey Robin R, Woods Keith W, Florjancic Alan S
Year of Publication 24.10.2017
Get full text
Year of Publication 24.10.2017
Patent
PYRROLO[2,3-B]PYRIDINE CDK9 KINASE INHIBITORS
CURTIN, Michael L, GONG, Jianchun, PENNING, Thomas, TAO, Zhi-fu, GOSWAMI, Rajeev, LAI, Chunqiu, WOODS, Keith W, FLORJANCIC, Alan S, MIYASHIRO, Juliem, DABBEERU, Madhu Babu, HANSEN, Todd M, SOUERS, Andrew, JI, Zhiqin, TONG, Yunsong, BRUNCKO, Milan, CLARK, Richard F, IQUTURI, Omprakash Reddy, MICHAELIDES, Michael, ZHU, Guidong, RISI, Roberto M, MASTRACCHIO, Anthony, SONG, Xiaohong, FREY, Robin R
Year of Publication 07.12.2016
Get full text
Year of Publication 07.12.2016
Patent
PYRROLO [2,3-B] PYRIDINE CDK9 KINASE INHIBITORS
GONG JIANCHUN, RISI ROBERTO M, FLORJANCIC ALAN S, TAO ZHI-FU, TONG YUNSONG, CURTIN MICHAEL, GOSWAMI RAJEEV, HANSEN TODD M, JI ZHIQIN, SONG XIAOHONG, WOODS KEITH W, DABBEERU MADHU BABU, MASTRACCHIO ANTHONY, MICHAELIDES MICHAEL, SOUERS ANDREW, IQUTURI OMPRAKASH REDDY, BRUNCKO MILAN, MIYASHIRO JULIEM, LAI CHUNQIU, ZHU GUIDONG, PENNING THOMAS, CLARK RICHARD F, FREY ROBIN R
Year of Publication 03.03.2016
Get full text
Year of Publication 03.03.2016
Patent
PYRROLO[2,3-B]PYRIDINE CDK9 KINASE INHIBITORS
TAO, ZHI-FU, ZHU, GUIDONG, MICHAELIDES, MICHAEL, FLORJANCIC, ALAN S, CLARK, RICHARD F, GOSWAMI, RAJEEV, FREY, ROBIN R, LAI, CHUNQIU, SONG, XIAOHONG, TONG, YUNSONG, GONG, JIANCHUN, RISI, ROBERTO M, JI, ZHIQIN, MASTRACCHIO, ANTHONY, MIYASHIRO, JULIEM, WOODS, KEITH W, BRUNCKO, MILAN, HANSEN, TODD M, IQUTURI, OMPRAKASH REDDY, DABBEERU, MADHU BABU, CURTIN, MICHAEL L, SOUERS, ANDREW, PENNING, THOMAS
Year of Publication 20.01.2016
Get full text
Year of Publication 20.01.2016
Patent
Pyrrolo[2, 3-b]pyridine cdk9 kinase inhibitors
GONG JIANCHUN, RISI ROBERTO M, FLORJANCIC ALAN S, TAO ZHI-FU, TONG YUNSONG, GOSWAMI RAJEEV, HANSEN TODD M, JI ZHIQIN, SONG XIAOHONG, WOODS KEITH W, DABBEERU MADHU BABU, MASTRACCHIO ANTHONY, MICHAELIDES MICHAEL, SOUERS ANDREW, IQUTURI OMPRAKASH REDDY, BRUNCKO MILAN, MIYASHIRO JULIEM, LAI CHUNQIU, ZHU GUIDONG, PENNING THOMAS, CURTIN MICHAEL L, CLARK RICHARD F, FREY ROBIN R
Year of Publication 13.01.2016
Get full text
Year of Publication 13.01.2016
Patent
Pyrrolo[2,3-b]pyridine CDK9 kinase inhibitors
TAO, ZHI-FU, ZHU, GUIDONG, MICHAELIDES, MICHAEL, FLORJANCIC, ALAN S, CLARK, RICHARD F, GOSWAMI, RAJEEV, FREY, ROBIN R, LAI, CHUNQIU, SONG, XIAOHONG, TONG, YUNSONG, GONG, JIANCHUN, RISI, ROBERTO M, JI, ZHIQIN, MASTRACCHIO, ANTHONY, MIYASHIRO, JULIEM, WOODS, KEITH W, BRUNCKO, MILAN, HANSEN, TODD M, IQUTURI, OMPRAKASH REDDY, DABBEERU, MADHU BABU, CURTIN, MICHAEL L, SOUERS, ANDREW, PENNING, THOMAS
Year of Publication 01.10.2015
Get full text
Year of Publication 01.10.2015
Patent
PYRROLO[2,3-B]PYRIDINE CDK9 KINASE INHIBITORS
TAO, ZHI-FU, ZHU, GUIDONG, MICHAELIDES, MICHAEL, FLORJANCIC, ALAN S, CLARK, RICHARD F, GOSWAMI, RAJEEV, FREY, ROBIN R, LAI, CHUNQIU, SONG, XIAOHONG, TONG, YUNSONG, GONG, JIANCHUN, RISI, ROBERTO M, JI, ZHIQIN, MASTRACCHIO, ANTHONY, MIYASHIRO, JULIEM, WOODS, KEITH W, BRUNCKO, MILAN, HANSEN, TODD M, IQUTURI, OMPRAKASH REDDY, DABBEERU, MADHU BABU, CURTIN, MICHAEL L, SOUERS, ANDREW, PENNING, THOMAS
Year of Publication 18.09.2014
Get full text
Year of Publication 18.09.2014
Patent
PYRROLO[2,3-B]PYRIDINE CDK9 KINASE INHIBITORS
TAO, ZHI-FU, ZHU, GUIDONG, MICHAELIDES, MICHAEL, FLORJANCIC, ALAN S, CLARK, RICHARD F, GOSWAMI, RAJEEV, FREY, ROBIN R, LAI, CHUNQIU, SONG, XIAOHONG, TONG, YUNSONG, GONG, JIANCHUN, RISI, ROBERTO M, JI, ZHIQIN, MASTRACCHIO, ANTHONY, MIYASHIRO, JULIEM, WOODS, KEITH W, BRUNCKO, MILAN, HANSEN, TODD M, IQUTURI, OMPRAKASH REDDY, DABBEERU, MADHU BABU, CURTIN, MICHAEL L, SOUERS, ANDREW, PENNING, THOMAS
Year of Publication 18.09.2014
Get full text
Year of Publication 18.09.2014
Patent
inibidores de pirrolo[2,3 - b] piridina cdk9 kinase
JULIEM MIYASHIRO, YUNSONG TONG, ALAN S. FLORJANCIC, ANTHONY MASTRACCHIO, RICHARD F. CLARK, ROBIN R. FREY, TODD M. HANSEN, MICHAEL L. CURTIN, RAJEEV GOSWAMI, GUIDONG ZHU, MICHAEL MICHAELIDES, KEITH W. WOODS, OMPRAKASH REDDY IQUTURI, ZHI-FU TAO, ROBERTO M. RISI, THOMAS PENNING, CHUNQIU LAI, ZHIQIN JI, JIANCHUN GONG, MADHU BABU DABBEERU, XIAOHONG SONG, MILAN BRUNCKO
Year of Publication 18.07.2017
Get full text
Year of Publication 18.07.2017
Patent
INHIBIDORES DE CDK9 QUINASA DE PIRROLO[2,3-B]PIRIDINA
JULIEM MIYASHIRO, YUNSONG TONG, ANTHONY MASTRACCHIO, ALAN S. FLORJANCIC, ROBIN R. FREY, ANDREW SOUERS, RAJEEV GOSWAMI, MICHAEL L. CURTIN, GUIDONG ZHU, MICHAEL MICHAELIDES, ZHI TAO, OMPRAKASH REDDY IQUTURI, KEITH W. WOODS, THOMAS PENNING, XIAOHONG FU - SONG, CHUNQIU LAI, RICHARD CLARK, ZHIQIN JI, JIANCHUN GONG, MADHU BABU DABBEERU, MILAN BRUNCKO
Year of Publication 28.12.2016
Get full text
Year of Publication 28.12.2016
Patent
PYRROLO[2,3-B]PYRIDINE CDK9 KINASE INHIBITORS
JULIEM MIYASHIRO, YUNSONG TONG, ALAN S. FLORJANCIC, ANTHONY MASTRACCHIO, RICHARD F. CLARK, ROBIN R. FREY, TODD M. HANSEN, ANDREW SOUERS, MICHAEL L. CURTIN, RAJEEV GOSWAMI, GUIDONG ZHU, MICHAEL MICHAELIDES, KEITH W. WOODS, ZHI-FU TAO, OMPRAKASH REDDY IQUTURI, ROBERTO M. RISI, THOMAS PENNING, CHUNQIU LAI, ZHIQIN JI, JIANCHUN GONG, MADHU BABU DABBEERU, XIAOHONG SONG, MILAN BRUNCKO
Year of Publication 02.06.2016
Get full text
Year of Publication 02.06.2016
Patent
Pyrrolo[2,3-B]pyridine CDK9 kinase inhibitors
TAO, ZHI-FU, JI, ZHI-QIN, ZHU, GUIDONG, MICHAELIDES, MICHAEL, FLORJANCIC, ALAN S, CLARK, RICHARD F, GOSWAMI, RAJEEV, FREY, ROBIN R, SONG, XIAO-HONG, LAI, CHUNQIU, TONG, YUNSONG, GONG, JIANCHUN, RISI, ROBERTO M, MASTRACCHIO, ANTHONY, MIYASHIRO, JULIEM, WOODS, KEITH W, BRUNCKO, MILAN, HANSEN, TODD M, IQUTURI, OMPRAKASH REDDY, DABBEERU, MADHU BABU, CURTIN, MICHAEL L, SOUERS, ANDREW, PENNING, THOMAS
Year of Publication 16.12.2014
Get full text
Year of Publication 16.12.2014
Patent
INHIBIDORES DE CDK9 QUINASA DE PIRROLO (2,3- B) PIRIDINA
TAO, ZHI-FU, ZHU, GUIDONG, MICHAELIDES, MICHAEL, FLORJANCIC, ALAN S, CLARK, RICHARD F, GOSWAMI, RAJEEV, FREY, ROBIN R, LAI, CHUNQIU, SONG, XIAOHONG, TONG, YUNSONG, BRUNCKO,MILAN, GONG, JIANCHUN, JI, ZHIQIN, MASTRACCHIO, ANTHONY, MIYASHIRO, JULIEM, WOODS, KEITH W, IQUTURI, OMPRAKASH REDDY, DABBEERU, MADHU BABU, SOUERS, ANDREW, CURTIN, MICHAEL L, PENNING, THOMAS
Year of Publication 31.10.2014
Get full text
Year of Publication 31.10.2014
Patent