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A Dipolar Cycloaddition Reaction To Access 6‑Methyl-4,5,6,7-tetrahydro‑1H‑[1,2,3]triazolo[4,5‑c]pyridines Enables the Discovery Synthesis and Preclinical Profiling of a P2X7 Antagonist Clinical Candidate
Chrovian, Christa C, Soyode-Johnson, Akinola, Peterson, Alexander A, Gelin, Christine F, Deng, Xiaohu, Dvorak, Curt A, Carruthers, Nicholas I, Lord, Brian, Fraser, Ian, Aluisio, Leah, Coe, Kevin J, Scott, Brian, Koudriakova, Tatiana, Schoetens, Freddy, Sepassi, Kia, Gallacher, David J, Bhattacharya, Anindya, Letavic, Michael A
Published in Journal of medicinal chemistry (11.01.2018)
Published in Journal of medicinal chemistry (11.01.2018)
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A Dipolar Cycloaddition Reaction To Access 6-Methyl-4,5,6,7-tetrahydro-1H-1,2,3triazolo4,5-cpyridines Enables the Discovery Synthesis and Preclinical Profiling of a P2X7 Antagonist Clinical Candidate
Chrovian, Christa C, Soyode-Johnson, Akinola, Peterson, Alexander A, Gelin, Christine F, Deng, Xiaohu, Dvorak, Curt A, Carruthers, Nicholas I, Lord, Brian, Fraser, Ian, Aluisio, Leah, Coe, Kevin J, Scott, Brian, Koudriakova, Tatiana, Schoetens, Freddy, Sepassi, Kia, Gallacher, David J, Bhattacharya, Anindya, Letavic, Michael A
Published in Journal of medicinal chemistry (11.01.2018)
Published in Journal of medicinal chemistry (11.01.2018)
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Designing Next-Generation Drug-Like Molecules for Medicinal Applications
Year of Publication 2025
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Diels–Alder Cycloaddition to the Bay Region of Perylene and Its Derivatives as an Attractive Strategy for PAH Core Expansion: Theoretical and Practical Aspects
Kurpanik, Aneta, Matussek, Marek, Lodowski, Piotr, Szafraniec-Gorol, Grażyna, Krompiec, Michał, Krompiec, Stanisław
Published in Molecules (Basel, Switzerland) (17.11.2020)
Published in Molecules (Basel, Switzerland) (17.11.2020)
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Total synthesis of atropurpuran
Gong, Jing, Chen, Huan, Liu, Xiao-Yu, Wang, Zhi-Xiu, Nie, Wei, Qin, Yong
Published in Nature communications (08.07.2016)
Published in Nature communications (08.07.2016)
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Benzannulation via Ruthenium-Catalyzed Diol–Diene [4+2] Cycloaddition: One- and Two-Directional Syntheses of Fluoranthenes and Acenes
Geary, Laina M, Chen, Te-Yu, Montgomery, T. Patrick, Krische, Michael J
Published in Journal of the American Chemical Society (23.04.2014)
Published in Journal of the American Chemical Society (23.04.2014)
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The inverse electron demand Diels–Alder cycloaddition with carbon‐11 and fluorine‐18: A gateway to pretargeted imaging across the blood–brain barrier
Zientek, Simon H., Thompson, Stephen, Sephton, Selena Milicevic, Aigbirhio, Franklin I.
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.2023)
Published in Journal of labelled compounds & radiopharmaceuticals (01.07.2023)
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Glycoclusters on oligonucleotide and PNA scaffolds: synthesis and applications
Spinelli, Nicolas, Defrancq, Eric, Morvan, François
Published in Chemical Society reviews (01.01.2013)
Published in Chemical Society reviews (01.01.2013)
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Chemical synthesis of febrifugine and analogues
Smullen, Shaun, McLaughlin, Noel P., Evans, Paul
Published in Bioorganic & medicinal chemistry (15.05.2018)
Published in Bioorganic & medicinal chemistry (15.05.2018)
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Recent Developments in the Synthesis and Functionalization of Nitrogen Heterocycles: Volume II
Year of Publication 2024
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Recent Developments in the Synthesis and Functionalization of Nitrogen Heterocycles: Volume I
Year of Publication 2024
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Strategies Towards the Synthesis of N2-Substituted 1,2,3-Triazoles
SOUZA, RODRIGO OCTÁVIO M.A. DE, MIRANDA, LEANDRO S. DE MARIZ E
Published in Anais da Academia Brasileira de Ciências (14.02.2019)
Published in Anais da Academia Brasileira de Ciências (14.02.2019)
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