Antiviral Activity and Crystal Structures of HIV-1 gp120 Antagonists
Curreli, Francesca, Kwon, Young D, Nicolau, Isabella, Burgos, Giancarla, Altieri, Andrea, Kurkin, Alexander V, Verardi, Raffaello, Kwong, Peter D, Debnath, Asim K
Published in International journal of molecular sciences (15.12.2022)
Published in International journal of molecular sciences (15.12.2022)
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Journal Article
Comparative Pharmacokinetics of a Dual Inhibitor of HIV-1, NBD-14189, in Rats and Dogs with a Proof-of-Concept Evaluation of Antiviral Potency in SCID-hu Mouse Model
Stoddart, Cheryl A, Curreli, Francesca, Horrigan, Stephen, Altieri, Andrea, Kurkin, Alexander V, Debnath, Asim K
Published in Viruses (01.10.2022)
Published in Viruses (01.10.2022)
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Journal Article
Synthesis of 5-Arylpyrrole-2-carboxylic Acids as Key Intermediates for NBD Series HIV-1 Entry Inhibitors
Belov, Dmitry S., Ivanov, Vladimir N., Curreli, Francesca, Kurkin, Alexander V., Altieri, Andrea, Debnath, Asim K.
Published in Synthesis (Stuttgart) (16.08.2017)
Published in Synthesis (Stuttgart) (16.08.2017)
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Journal Article
Discovery of Highly Potent Small Molecule Pan-Coronavirus Fusion Inhibitors
Curreli, Francesca, Chau, Kent, Tran, Thanh-Thuy, Nicolau, Isabella, Ahmed, Shahad, Das, Pujita, Hillyer, Christopher D, Premenko-Lanier, Mary, Debnath, Asim K
Published in Viruses (01.04.2023)
Published in Viruses (01.04.2023)
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Journal Article
Binding mode characterization of NBD series CD4-mimetic HIV-1 entry inhibitors by X-ray structure and resistance study
Curreli, Francesca, Kwon, Young Do, Zhang, Hongtao, Yang, Yongping, Scacalossi, Daniel, Kwong, Peter D, Debnath, Asim K
Published in Antimicrobial agents and chemotherapy (01.09.2014)
Published in Antimicrobial agents and chemotherapy (01.09.2014)
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Journal Article
Design, synthesis and evaluation of small molecule CD4-mimics as entry inhibitors possessing broad spectrum anti-HIV-1 activity
Curreli, Francesca, Belov, Dmitry S., Ramesh, Ranjith R., Patel, Naisargi, Altieri, Andrea, Kurkin, Alexander V., Debnath, Asim K.
Published in Bioorganic & medicinal chemistry (15.11.2016)
Published in Bioorganic & medicinal chemistry (15.11.2016)
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Journal Article
Virtual screening based identification of novel small-molecule inhibitors targeted to the HIV-1 capsid
Curreli, Francesca, Zhang, Hongtao, Zhang, Xihui, Pyatkin, Ilya, Victor, Zagorodnikov, Altieri, Andrea, Debnath, Asim K.
Published in Bioorganic & medicinal chemistry (01.01.2011)
Published in Bioorganic & medicinal chemistry (01.01.2011)
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Journal Article
Discovery of Highly Potent Fusion Inhibitors with Potential Pan-Coronavirus Activity That Effectively Inhibit Major COVID-19 Variants of Concern (VOCs) in Pseudovirus-Based Assays
Curreli, Francesca, Ahmed, Shahad, Victor, Sofia M B, Drelich, Aleksandra, Panda, Siva S, Altieri, Andrea, Kurkin, Alexander V, Tseng, Chien-Te K, Hillyer, Christopher D, Debnath, Asim K
Published in Viruses (31.12.2021)
Published in Viruses (31.12.2021)
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Journal Article
Synthesis, antiviral activity and resistance of a novel small molecule HIV-1 entry inhibitor
Curreli, Francesca, Haque, Kashfia, Xie, Lihua, Qiu, Qian, Xu, Jinfeng, Yong, Weizhong, Tong, Xiaohe, Debnath, Asim K.
Published in Bioorganic & medicinal chemistry (15.12.2015)
Published in Bioorganic & medicinal chemistry (15.12.2015)
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Journal Article
Antiviral activity of α-helical stapled peptides designed from the HIV-1 capsid dimerization domain
Zhang, Hongtao, Curreli, Francesca, Zhang, Xihui, Bhattacharya, Shibani, Waheed, Abdul A, Cooper, Alan, Cowburn, David, Freed, Eric O, Debnath, Asim K
Published in Retrovirology (03.05.2011)
Published in Retrovirology (03.05.2011)
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Journal Article
Dual-acting stapled peptides target both HIV-1 entry and assembly
Zhang, Hongtao, Curreli, Francesca, Waheed, Abdul A, Mercredi, Peter Y, Mehta, Mansi, Bhargava, Pallavi, Scacalossi, Daniel, Tong, Xiaohe, Lee, Shawn, Cooper, Alan, Summers, Michael F, Freed, Eric O, Debnath, Asim K
Published in Retrovirology (15.11.2013)
Published in Retrovirology (15.11.2013)
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Journal Article
Antiviral Activity of Dual-acting Hydrocarbon-stapled Peptides against HIV-1 Predominantly Circulating in China
WANG, Yan, CURRELI, Francesca, XU, Wei Si, LI, Zhen Peng, KONG, De Sheng, REN, Li, HONG, Kun Xue, JIANG, Shi Bo, SHAO, Yi Ming, DEBNATH, Asim K, MA, Li Ying
Published in Biomedical and environmental sciences (01.06.2017)
Published in Biomedical and environmental sciences (01.06.2017)
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Journal Article
Transcriptional Downregulation of ORF50/Rta by Methotrexate Inhibits the Switch of Kaposi's Sarcoma-Associated Herpesvirus/Human Herpesvirus 8 from Latency to Lytic Replication
Curreli, Francesca, Cerimele, Francesca, Muralidhar, Sumitra, Rosenthal, Leonard J, Cesarman, Ethel, Friedman-Kien, Alvin E, Flore, Ornella
Published in Journal of Virology (01.05.2002)
Published in Journal of Virology (01.05.2002)
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Journal Article
α‐Helix‐Mimetic Foldamers for Targeting HIV‐1 TAR RNA
Maity, Debabrata, Kumar, Sunil, Curreli, Francesca, Debnath, Asim K., Hamilton, Andrew D.
Published in Chemistry : a European journal (28.05.2019)
Published in Chemistry : a European journal (28.05.2019)
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Journal Article
HIV‑1 gp120 Antagonists Also Inhibit HIV‑1 Reverse Transcriptase by Bridging the NNRTI and NRTI Sites
Losada, Natalie, Ruiz, Francesc X, Curreli, Francesca, Gruber, Kevin, Pilch, Alyssa, Das, Kalyan, Debnath, Asim K, Arnold, Eddy
Published in Journal of medicinal chemistry (25.11.2021)
Published in Journal of medicinal chemistry (25.11.2021)
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Journal Article
Synthesis, Antiviral Potency, in Vitro ADMET, and X‑ray Structure of Potent CD4 Mimics as Entry Inhibitors That Target the Phe43 Cavity of HIV‑1 gp120
Curreli, Francesca, Kwon, Young Do, Belov, Dmitry S, Ramesh, Ranjith R, Kurkin, Alexander V, Altieri, Andrea, Kwong, Peter D, Debnath, Asim K
Published in Journal of medicinal chemistry (13.04.2017)
Published in Journal of medicinal chemistry (13.04.2017)
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Journal Article
Stapled Peptides Based on Human Angiotensin-Converting Enzyme 2 (ACE2) Potently Inhibit SARS-CoV-2 Infection In Vitro
Curreli, Francesca, Victor, Sofia M B, Ahmed, Shahad, Drelich, Aleksandra, Tong, Xiaohe, Tseng, Chien-Te K, Hillyer, Christopher D, Debnath, Asim K
Published in mBio (11.12.2020)
Published in mBio (11.12.2020)
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