An investigation into the structure-activity relationships associated with the systematic modification of the beta(2)-adrenoceptor agonist indacaterol
Beattie, David, Beer, David, Bradley, Michelle E., Bruce, Ian, Charlton, Steven J., Cuenoud, Bernard M., Fairhurst, Robin A., Farr, David, Fozard, John R., Janus, Diana, Rosethorne, Elizabeth M., Sandham, David A., Sykes, David A., Trifilieff, Alexandre, Turner, Katharine L., Wissler, Elke
Published in Bioorganic & medicinal chemistry letters (01.10.2012)
Published in Bioorganic & medicinal chemistry letters (01.10.2012)
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Journal Article
An investigation into the structure–activity relationships associated with the systematic modification of the β2-adrenoceptor agonist indacaterol
Beattie, David, Beer, David, Bradley, Michelle E., Bruce, Ian, Charlton, Steven J., Cuenoud, Bernard M., Fairhurst, Robin A., Farr, David, Fozard, John R., Janus, Diana, Rosethorne, Elizabeth M., Sandham, David A., Sykes, David A., Trifilieff, Alexandre, Turner, Katharine L., Wissler, Elke
Published in Bioorganic & medicinal chemistry letters (01.10.2012)
Published in Bioorganic & medicinal chemistry letters (01.10.2012)
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Journal Article
A physical properties based approach for the exploration of a 4-hydroxybenzothiazolone series of β2-adrenoceptor agonists as inhaled long-acting bronchodilators
BEATTIE, David, BRADLEY, Michelle, LEWIS, Christine, MCCARTHY, Clive, OAKMAN, Helen, STRINGER, Rowan, TAYLOR, Roger J, TUFFNELL, Andrew, BREARLEY, Andrew, CHARLTON, Steven J, CUENOUD, Bernard M, FAIRHURST, Robin A, GEDECK, Peter, GOSLING, Martin, JANUS, Diana, JONES, Darryl
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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Journal Article
Synthesis and biological properties of novel glucocorticoid androstene C-17 furoate esters
Sandham, David A., Barker, Lucy, Beattie, David, Beer, David, Bidlake, Louise, Bentley, David, Butler, Keith D., Craig, Sarah, Farr, David, Ffoulkes-Jones, Claire, Fozard, John R., Haberthuer, Sandra, Howes, Colin, Hynx, Deborah, Jeffers, Sarah, Keller, Thomas H., Kirkham, Paul A., Maas, Janet C., Mazzoni, Lazzaro, Nicholls, Andrew, Pilgrim, Gaynor E., Schaebulin, Elisabeth, Spooner, Gillian M., Stringer, Rowan, Tranter, Pamela, Turner, Katharine L., Tweed, Morris F., Walker, Christoph, Watson, Simon J., Cuenoud, Bernard M.
Published in Bioorganic & medicinal chemistry (01.10.2004)
Published in Bioorganic & medicinal chemistry (01.10.2004)
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Journal Article
Long-chain formoterol analogues: an investigation into the effect of increasing amino-substituent chain length on the β2-adrenoceptor activity
ALIKHANI, Vahid, BEER, David, JORDAN, Lynne, LEWIS, Christine, SMITHIES, Kirsty, WISSLER, Elke, BENTLEY, David, BRUCE, Ian, CUENOUD, Bernard M, FAIRHURST, Robin A, GEDECK, Peter, HABERTHUER, Sandra, HAYDEN, Claire, JANUS, Diana
Published in Bioorganic & medicinal chemistry letters (01.09.2004)
Published in Bioorganic & medicinal chemistry letters (01.09.2004)
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Journal Article
An investigation into the structure-activity relationships associated with the systematic modification of the [beta]2-adrenoceptor agonist indacaterol
Beattie, David, Beer, David, Bradley, Michelle E, Bruce, Ian, Charlton, Steven J, Cuenoud, Bernard M, Fairhurst, Robin A, Farr, David, Fozard, John R, Janus, Diana, Rosethorne, Elizabeth M, Sandham, David A, Sykes, David A, Trifilieff, Alexandre, Turner, Katharine L, Wissler, Elke
Published in Bioorganic & medicinal chemistry letters (01.10.2012)
Published in Bioorganic & medicinal chemistry letters (01.10.2012)
Get full text
Journal Article
Long-chain formoterol analogues: an investigation into the effect of increasing amino-substituent chain length on the β 2-adrenoceptor activity
Alikhani, Vahid, Beer, David, Bentley, David, Bruce, Ian, Cuenoud, Bernard M., Fairhurst, Robin A., Gedeck, Peter, Haberthuer, Sandra, Hayden, Claire, Janus, Diana, Jordan, Lynne, Lewis, Christine, Smithies, Kirsty, Wissler, Elke
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
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Journal Article
A physical properties based approach for the exploration of a 4-hydroxybenzothiazolone series of β 2-adrenoceptor agonists as inhaled long-acting bronchodilators
Beattie, David, Bradley, Michelle, Brearley, Andrew, Charlton, Steven J., Cuenoud, Bernard M., Fairhurst, Robin A., Gedeck, Peter, Gosling, Martin, Janus, Diana, Jones, Darryl, Lewis, Christine, McCarthy, Clive, Oakman, Helen, Stringer, Rowan, Taylor, Roger J., Tuffnell, Andrew
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
A physical properties based approach for the exploration of a 4-hydroxybenzothiazolone series of beta2-adrenoceptor agonists as inhaled long-acting bronchodilators
Beattie, David, Bradley, Michelle, Brearley, Andrew, Charlton, Steven J, Cuenoud, Bernard M, Fairhurst, Robin A, Gedeck, Peter, Gosling, Martin, Janus, Diana, Jones, Darryl, Lewis, Christine, McCarthy, Clive, Oakman, Helen, Stringer, Rowan, Taylor, Roger J, Tuffnell, Andrew
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Get full text
Journal Article
Long-chain formoterol analogues: an investigation into the effect of increasing amino-substituent chain length on the beta2-adrenoceptor activity
Alikhani, Vahid, Beer, David, Bentley, David, Bruce, Ian, Cuenoud, Bernard M, Fairhurst, Robin A, Gedeck, Peter, Haberthuer, Sandra, Hayden, Claire, Janus, Diana, Jordan, Lynne, Lewis, Christine, Smithies, Kirsty, Wissler, Elke
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
Get full text
Published in Bioorganic & medicinal chemistry letters (20.09.2004)
Journal Article