HIV Protease Inhibitors Stimulate Hepatic Triglyceride Synthesis
Lenhard, James M, Croom, Dallas K, Weiel, James E, Winegar, Deborah A
Published in Arteriosclerosis, thrombosis, and vascular biology (01.12.2000)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.12.2000)
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Journal Article
Discovery of 6,7-Dihydro‑5H‑pyrrolo[2,3‑a]pyrimidines as Orally Available G Protein-Coupled Receptor 119 Agonists
Katamreddy, Subba R, Carpenter, Andrew J, Ammala, Carina E, Boros, Eric E, Brashear, Ron L, Briscoe, Celia P, Bullard, Sarah R, Caldwell, Richard D, Conlee, Christopher R, Croom, Dallas K, Hart, Shane M, Heyer, Dennis O, Johnson, Paul R, Kashatus, Jennifer A, Minick, Doug J, Peckham, Gregory E, Ross, Sean A, Roller, Shane G, Samano, Vicente A, Sauls, Howard R, Tadepalli, Sarva M, Thompson, James B, Xu, Yun, Way, James M
Published in Journal of medicinal chemistry (27.12.2012)
Published in Journal of medicinal chemistry (27.12.2012)
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Journal Article
Optimization of 3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines as Potent, Orally Active CCK-A Agonists
Henke, Brad R, Aquino, Christopher J, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Queen, Kennedy L, Sherrill, Ronald G, Sugg, Elizabeth E, Suh, Edward M, Szewczyk, Jerzy W, Unwalla, Rayomand J, Yingling, Jeff, Willson, Timothy M
Published in Journal of medicinal chemistry (15.08.1997)
Published in Journal of medicinal chemistry (15.08.1997)
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Journal Article
Dietary Fat Alters HIV Protease Inhibitor–Induced Metabolic Changes in Mice
Lenhard, James M., Croom, Dallas K., Weiel, James E., Spaltenstein, Andrew, Reynolds, David J., Furfine, Eric S.
Published in The Journal of nutrition (01.09.2000)
Published in The Journal of nutrition (01.09.2000)
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Journal Article
Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity. 1. Optimization of the Agonist “Trigger”
Aquino, Christopher J, Armour, Duncan R, Berman, Judd M, Birkemo, Larry S, Carr, Robin A. E, Croom, Dallas K, Dezube, Milana, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Head, Julie E, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Miller, Laurence J, Queen, Kennedy L, Rimele, Thomas J, Smith, David N, Sugg, Elizabeth E
Published in Journal of medicinal chemistry (19.01.1996)
Published in Journal of medicinal chemistry (19.01.1996)
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Journal Article
1,4-Benzodiazepine Peripheral Cholecystokinin (CCK-A) Receptor Agonists
Sherrill, Ronald G, Berman, Judd M, Birkemo, Lawrence, Croom, Dallas K, Dezube, Milana, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Vanmiddlesworth, Frank, Sugg, Elizabeth E
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
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Journal Article
3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines: CCK-A Agonists That Demonstrate Oral Activity as Satiety Agents
Henke, Brad R, Willson, Timothy M, Sugg, Elizabeth E, Croom, Dallas K, Dougherty, Robert W, Queen, Kennedy L, Birkemo, Larry S, Ervin, Gregory N, Grizzle, Mary K, Johnson, Michael F, James, Michael K
Published in Journal of medicinal chemistry (05.07.1996)
Published in Journal of medicinal chemistry (05.07.1996)
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Journal Article
3-[2-(N-Phenylacetamide)]-1,5-benzodiazepines: Orally Active, Binding Selective CCK-A Agonists
Willson, Timothy M, Henke, Brad R, Momtahen, Tanya M, Myers, Peter L, Sugg, Elizabeth E, Unwalla, Rayomand J, Croom, Dallas K, Dougherty, Robert W, Grizzle, Mary K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Yingling, Jeffrey D, James, Michael K
Published in Journal of medicinal chemistry (19.07.1996)
Published in Journal of medicinal chemistry (19.07.1996)
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Journal Article
Modification of Receptor Selectivity and Functional Activity in Cholecystokinin Peptoid Ligands
Dezube, Milana, Sugg, Elizabeth E, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F
Published in Journal of medicinal chemistry (01.08.1995)
Published in Journal of medicinal chemistry (01.08.1995)
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Journal Article
Structure-Activity Relationships for Inhibition of Type 1 and 2 Human 5.alpha.-Reductase and Human Adrenal 3.beta.-Hydroxy-.DELTA.5-steroid Dehydrogenase/3-Keto-.DELTA.5-steroid Isomerase by 6-Azaandrost-4-en-3-ones: Optimization of the C17 Substituent
Frye, Stephen V, Haffner, Curt D, Maloney, Patrick R, Hiner, Roger N, Dorsey, George F, Noe, Robert A, Unwalla, Rayomand J, Batchelor, Kenneth W, Bramson, H. Neal, Stuart, J. Darren, Schweiker, Stephanie L, Van Arnold, John, Bickett, D. Mark, Moss, Marcia L, Tian, Gaochoa, Lee, Frank W, Tippin, Timothy K, James, Michael K, Grizzle, Mary K, Long, James E, Croom, Dallas K
Published in Journal of medicinal chemistry (01.07.1995)
Published in Journal of medicinal chemistry (01.07.1995)
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Journal Article
Discovery of 6,7-Dihydro-5 H -pyrrolo[2,3- a ]pyrimidines as Orally Available G Protein-Coupled Receptor 119 Agonists
Katamreddy, Subba R., Carpenter, Andrew J., Ammala, Carina E., Boros, Eric E., Brashear, Ron L., Briscoe, Celia P., Bullard, Sarah R., Caldwell, Richard D., Conlee, Christopher R., Croom, Dallas K., Hart, Shane M., Heyer, Dennis O., Johnson, Paul R., Kashatus, Jennifer A., Minick, Doug J., Peckham, Gregory E., Ross, Sean A., Roller, Shane G., Samano, Vicente A., Sauls, Howard R., Tadepalli, Sarva M., Thompson, James B., Xu, Yun, Way, James M.
Published in Journal of medicinal chemistry (27.12.2012)
Published in Journal of medicinal chemistry (27.12.2012)
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Journal Article
Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity (II): Optimization of the C3 Amino Substituent
Hirst, Gavin C., Aquino, Christopher, Birkemo, Lawrence, Croom, Dallas K., Dezube, Milana, Dougherty, Robert W., Ervin, Gregory N., Grizzle, Mary K., Henke, Brad, James, Michael K., Johnson, Michael F., Momtahen, Tanya, Queen, Kennedy L., Sherrill, Ronald G., Szewczyk, Jerzy, Willson, Timothy M., Sugg, Elizabeth E.
Published in Journal of medicinal chemistry (20.12.1996)
Published in Journal of medicinal chemistry (20.12.1996)
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Journal Article
4-Substituted Uridine 5′-Triphosphates as Agonists of the P2Y2 Purinergic Receptor
Shaver, Sammy R., Pendergast, William, Siddiqi, Suhaib M., Yerxa, Benjamin R., Croom, Dallas K., Dougherty, Robert W., James, Michael K., Jones, A. Neil, Rideout, Janet L.
Published in Nucleosides & nucleotides (01.07.1997)
Published in Nucleosides & nucleotides (01.07.1997)
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Journal Article
4-Substituted Uridine 5′-Triphosphates as Agonists of the P 2Y2 Purinergic Receptor
Shaver, Sammy R., Pendergast, William, Siddiqi, Suhaib M., Yerxa, Benjamin R., Croom, Dallas K., Dougherty, Robert W., James, Michael K., Jones, A. Neil, Rideout, Janet L.
Published in Nucleosides & nucleotides (01.07.1997)
Published in Nucleosides & nucleotides (01.07.1997)
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Journal Article