Abstract B129: Preclinical studies with DCC-3116, an ULK kinase inhibitor designed to inhibit autophagy as a potential strategy to address mutant RAS cancers
Smith, Bryan D, Vogeti, Lakshminarayana, Gupta, Anu, Singh, Jarnail, Al-Ani, Gada, Bulfer, Stacie L, Caldwell, Timothy M, Timson, Mary J, Vogeti, Subha, Ahn, Yu Mi, Al-Hashimi, Hikmat, Crawley, Chase K, Heiniger, Cale L, Leary, Cynthia B, Proto, Justin T, Shen, Quanrong, Telikepalli, Hanumaiah, Yates, Karen, Lu, Wei-Ping, Flynn, Daniel L
Published in Molecular cancer therapeutics (01.12.2019)
Published in Molecular cancer therapeutics (01.12.2019)
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Journal Article
Abstract 593: DCC-3084, a brain penetrant RAF dimer inhibitor, broadly inhibits BRAF class I, II, and III alterations leading to growth inhibition of intracranially implanted tumors in preclinical models
Al-Ani, Gada, Bulfer, Stacie L., Zwicker, Jefferey D., Crawley, Chase K., Elliot, Kristin M., Javed, Salim, Groer, Qi, Hood, Molly M., Large, Joshua W., Luther, Kylie, Romero, Yeni K., Stanley, Forrest A., Tanner, Daniel C., Telikepalli, Hanumaiah, Le Bourdonnec, Bertrand, Smith, Bryan D., Flynn, Daniel L.
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Journal Article
Abstract 4045: DCC-3084, a RAF dimer inhibitor, broadly inhibits BRAF class I, II, III, BRAF fusions, and RAS-driven solid tumors leading to tumor regression in preclinical models
Bulfer, Stacie L., Bourdonnec, Bertrand Le, Zwicker, Jeffery D., Ahn, Yu Mi, Al-Ani, Gada, Al-Hashimi, Hikmat, Crawley, Chase, Elliott, Kristin M., Faisal, Saqib, Harned, Andrew M., Heiniger, Cale L., Hood, Molly M., Javed, Salim, Kennedy, Michael, Large, Joshua W., Leary, Cynthia B., Lu, Wei-Ping, Luther, Kylie, Petty, Max D., Picard, Hunter R., Proto, Justin T., Romero, Yeni K., Stanley, Forrest A., Stoltz, Kristen L., Tanner, Daniel C., Telikepalli, Hanumaiah, Timson, Mary J., Vogeti, Lakshminarayana, Vogeti, Subha, Yang, Sihyung, Zhong, Lexy H., Smith, Bryan D., Flynn, Daniel L.
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Journal Article
RAF KINASE INHIBITORS AND METHODS OF USE THEREOF
VOGETI, Lakshminarayana, CRAWLEY, Chase Kenyon, AHN, Yu Mi, FLYNN, Daniel L, LE BOURDONNEC, Bertrand
Year of Publication 11.07.2024
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Year of Publication 11.07.2024
Patent
RAF KINASE INHIBITORS AND METHODS OF USE THEREOF
FLYNN, DANIEL L, CRAWLEY, CHASE KENYON, LE BOURDONNEC, BERTRAND, AHN, YU MI, VOGETI, LAKSHMINARAYANA
Year of Publication 15.06.2023
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Year of Publication 15.06.2023
Patent