Cryo-EM structures of the TMEM16A calcium-activated chloride channel
Dang, Shangyu, Feng, Shengjie, Tien, Jason, Peters, Christian J, Bulkley, David, Lolicato, Marco, Zhao, Jianhua, Zuberbühler, Kathrin, Ye, Wenlei, Qi, Lijun, Chen, Tingxu, Craik, Charles S, Jan, Yuh Nung, Minor, Jr, Daniel L, Cheng, Yifan, Jan, Lily Yeh
Published in Nature (London) (21.12.2017)
Published in Nature (London) (21.12.2017)
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Journal Article
Mapping the catalytic conformations of an assembly-line polyketide synthase module
Cogan, Dillon P, Zhang, Kaiming, Li, Xiuyuan, Li, Shanshan, Pintilie, Grigore D, Roh, Soung-Hun, Craik, Charles S, Chiu, Wah, Khosla, Chaitan
Published in Science (American Association for the Advancement of Science) (05.11.2021)
Published in Science (American Association for the Advancement of Science) (05.11.2021)
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Structure- and function-based design of Plasmodium-selective proteasome inhibitors
Li, Hao, O'Donoghue, Anthony J, van der Linden, Wouter A, Xie, Stanley C, Yoo, Euna, Foe, Ian T, Tilley, Leann, Craik, Charles S, da Fonseca, Paula C A, Bogyo, Matthew
Published in Nature (London) (11.02.2016)
Published in Nature (London) (11.02.2016)
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Journal Article
Characterising proteolysis during SARS-CoV-2 infection identifies viral cleavage sites and cellular targets with therapeutic potential
Meyer, Bjoern, Chiaravalli, Jeanne, Gellenoncourt, Stacy, Brownridge, Philip, Bryne, Dominic P, Daly, Leonard A, Grauslys, Arturas, Walter, Marius, Agou, Fabrice, Chakrabarti, Lisa A, Craik, Charles S, Eyers, Claire E, Eyers, Patrick A, Gambin, Yann, Jones, Andrew R, Sierecki, Emma, Verdin, Eric, Vignuzzi, Marco, Emmott, Edward
Published in Nature communications (21.09.2021)
Published in Nature communications (21.09.2021)
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Journal Article
Quantitative MS-based enzymology of caspases reveals distinct protein substrate specificities, hierarchies, and cellular roles
Julien, Olivier, Zhuang, Min, Wiita, Arun P., O’Donoghue, Anthony J., Knudsen, Giselle M., Craik, Charles S., Wells, James A.
Published in Proceedings of the National Academy of Sciences - PNAS (05.04.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (05.04.2016)
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Journal Article
Mechanisms of Macromolecular Protease Inhibitors
Farady, Christopher J, Craik, Charles S
Published in Chembiochem : a European journal of chemical biology (22.11.2010)
Published in Chembiochem : a European journal of chemical biology (22.11.2010)
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Journal Article
Combination of Antifungal Drugs and Protease Inhibitors Prevent Candida albicans Biofilm Formation and Disrupt Mature Biofilms
Lohse, Matthew B, Gulati, Megha, Craik, Charles S, Johnson, Alexander D, Nobile, Clarissa J
Published in Frontiers in microbiology (25.05.2020)
Published in Frontiers in microbiology (25.05.2020)
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Assessment of human virus removal during municipal wastewater treatment in Edmonton, Canada
Qiu, Y., Lee, B.E., Neumann, N., Ashbolt, N., Craik, S., Maal‐Bared, R., Pang, X.L.
Published in Journal of applied microbiology (01.12.2015)
Published in Journal of applied microbiology (01.12.2015)
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Journal Article
Subnanometre-resolution electron cryomicroscopy structure of a heterodimeric ABC exporter
Kim, JungMin, Wu, Shenping, Tomasiak, Thomas M, Mergel, Claudia, Winter, Michael B, Stiller, Sebastian B, Robles-Colmanares, Yaneth, Stroud, Robert M, Tampé, Robert, Craik, Charles S, Cheng, Yifan
Published in Nature (London) (15.01.2015)
Published in Nature (London) (15.01.2015)
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Journal Article
Phosphorylation of tau at a single residue inhibits binding to the E3 ubiquitin ligase, CHIP
Nadel, Cory M, Pokhrel, Saugat, Wucherer, Kristin, Oehler, Abby, Thwin, Aye C, Basu, Koli, Callahan, Matthew D, Southworth, Daniel R, Mordes, Daniel A, Craik, Charles S, Gestwicki, Jason E
Published in Nature communications (12.09.2024)
Published in Nature communications (12.09.2024)
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Structural and mechanistic basis of the EMC-dependent biogenesis of distinct transmembrane clients
Miller-Vedam, Lakshmi E, Bräuning, Bastian, Popova, Katerina D, Schirle Oakdale, Nicole T, Bonnar, Jessica L, Prabu, Jesuraj R, Boydston, Elizabeth A, Sevillano, Natalia, Shurtleff, Matthew J, Stroud, Robert M, Craik, Charles S, Schulman, Brenda A, Frost, Adam, Weissman, Jonathan S
Published in eLife (25.11.2020)
Published in eLife (25.11.2020)
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Substrate Profiling of Cysteine Proteases Using a Combinatorial Peptide Library Identifies Functionally Unique Specificities
Choe, Youngchool, Leonetti, Francesco, Greenbaum, Doron C., Lecaille, Fabien, Bogyo, Matthew, Brömme, Dieter, Ellman, Jonathan A., Craik, Charles S.
Published in The Journal of biological chemistry (05.05.2006)
Published in The Journal of biological chemistry (05.05.2006)
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Journal Article
Structural requirements for the collagenase and elastase activity of cathepsin K and its selective inhibition by an exosite inhibitor
Sharma, Vidhu, Panwar, Preety, O'Donoghue, Anthony J, Cui, Haoran, Guido, Rafael V C, Craik, Charles S, Brömme, Dieter
Published in Biochemical journal (01.01.2015)
Published in Biochemical journal (01.01.2015)
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Journal Article
Predicting CD4 T-cell epitopes based on antigen cleavage, MHCII presentation, and TCR recognition
Schneidman-Duhovny, Dina, Khuri, Natalia, Dong, Guang Qiang, Winter, Michael B, Shifrut, Eric, Friedman, Nir, Craik, Charles S, Pratt, Kathleen P, Paz, Pedro, Aswad, Fred, Sali, Andrej
Published in PloS one (06.11.2018)
Published in PloS one (06.11.2018)
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Continuous Imaging of Plasmon Rulers in Live Cells Reveals Early-Stage Caspase-3 Activation at the Single-Molecule Level
Jun, Young-wook, Sheikholeslami, Sassan, Hostetter, Daniel R., Tajon, Cheryl, Craik, Charles S., Alivisatos, A. Paul
Published in Proceedings of the National Academy of Sciences - PNAS (20.10.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (20.10.2009)
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Journal Article
Global substrate profiling of proteases in human neutrophil extracellular traps reveals consensus motif predominantly contributed by elastase
O'Donoghue, Anthony J, Jin, Ye, Knudsen, Giselle M, Perera, Natascha C, Jenne, Dieter E, Murphy, John E, Craik, Charles S, Hermiston, Terry W
Published in PloS one (20.09.2013)
Published in PloS one (20.09.2013)
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Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery
Kryštůfek, Robin, Šácha, Pavel, Starková, Jana, Brynda, Jiří, Hradilek, Martin, Tloušt’ová, Eva, Grzymska, Justyna, Rut, Wioletta, Boucher, Michael J, Drąg, Marcin, Majer, Pavel, Hájek, Miroslav, Řezáčová, Pavlína, Madhani, Hiten D, Craik, Charles S, Konvalinka, Jan
Published in Journal of medicinal chemistry (27.05.2021)
Published in Journal of medicinal chemistry (27.05.2021)
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Journal Article
Vinyl Sulfones as Antiparasitic Agents and a Structural Basis for Drug Design
Kerr, Iain D., Lee, Ji H., Farady, Christopher J., Marion, Rachael, Rickert, Mathias, Sajid, Mohammed, Pandey, Kailash C., Caffrey, Conor R., Legac, Jennifer, Hansell, Elizabeth, McKerrow, James H., Craik, Charles S., Rosenthal, Philip J., Brinen, Linda S.
Published in The Journal of biological chemistry (18.09.2009)
Published in The Journal of biological chemistry (18.09.2009)
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