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Isotopic Perturbation of Intramolecular Hydrogen Bonds in Rigid 1,3-Diols: NMR Studies Reveal Unusually Large Equilibrium Isotope Effects
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Efficient Synthesis of NK1 Receptor Antagonist Aprepitant Using a Crystallization-Induced Diastereoselective Transformation
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Published in Journal of the American Chemical Society (26.02.2003)
Published in Journal of the American Chemical Society (26.02.2003)
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Synthesis of a Potent hNK-1 Receptor Antagonist via an SN2 Reaction of an Enantiomerically Pure α-Alkoxy Sulfonate
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Published in Organic letters (06.01.2005)
Published in Organic letters (06.01.2005)
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Synthesis of a Potent hNK-1 Receptor Antagonist via an S N 2 Reaction of an Enantiomerically Pure α-Alkoxy Sulfonate
Nelson, Todd D., Rosen, Jonathan D., Smitrovich, Jacqueline H., Payack, Joseph, Craig, Bridgette, Matty, Louis, Huffman, Mark A., McNamara, James
Published in Organic letters (01.01.2005)
Published in Organic letters (01.01.2005)
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Efficient synthesis of NK(1) receptor antagonist aprepitant using a crystallization-induced diastereoselective transformation
Brands, Karel M J, Payack, Joseph F, Rosen, Jonathan D, Nelson, Todd D, Candelario, Alexander, Huffman, Mark A, Zhao, Matthew M, Li, Jing, Craig, Bridgette, Song, Zhiguo J, Tschaen, David M, Hansen, Karl, Devine, Paul N, Pye, Philip J, Rossen, Kai, Dormer, Peter G, Reamer, Robert A, Welch, Christopher J, Mathre, David J, Tsou, Nancy N, McNamara, James M, Reider, Paul J
Published in Journal of the American Chemical Society (26.02.2003)
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Published in Journal of the American Chemical Society (26.02.2003)
Journal Article
Efficient Synthesis of NK 1 Receptor Antagonist Aprepitant Using a Crystallization-Induced Diastereoselective Transformation
Brands, Karel M. J., Payack, Joseph F., Rosen, Jonathan D., Nelson, Todd D., Candelario, Alexander, Huffman, Mark A., Zhao, Matthew M., Li, Jing, Craig, Bridgette, Song, Zhiguo J., Tschaen, David M., Hansen, Karl, Devine, Paul N., Pye, Philip J., Rossen, Kai, Dormer, Peter G., Reamer, Robert A., Welch, Christopher J., Mathre, David J., Tsou, Nancy N., McNamara, James M., Reider, Paul J.
Published in Journal of the American Chemical Society (01.02.2003)
Published in Journal of the American Chemical Society (01.02.2003)
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Process Development and Scale-up of AG035029
Saenz, James, Mitchell, Mark, Bahmanyar, Sami, Stankovic, Nebojsa, Perry, Michael, Craig-Woods, Bridgette, Kline, Billie, Yu, Shu, Albizati, Kim
Published in Organic process research & development (01.01.2007)
Published in Organic process research & development (01.01.2007)
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Synthesis of a Potent hNK-1 Receptor Antagonist (I) via an SN2 Reaction of an Enantiomerically Pure α-Alkoxy Sulfonate
Nelson, Todd D., Rosen, Jonathan D., Smitrovich, Jacqueline H., Payack, Joseph, Craig, Bridgette, Matty, Louis, Huffman, Mark A., McNamara, James
Published in ChemInform (26.04.2005)
Published in ChemInform (26.04.2005)
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Journal Article
Synthesis of a Potent hNK‐1 Receptor Antagonist (I) via an S N 2 Reaction of an Enantiomerically Pure α‐Alkoxy Sulfonate
Nelson, Todd D., Rosen, Jonathan D., Smitrovich, Jacqueline H., Payack, Joseph, Craig, Bridgette, Matty, Louis, Huffman, Mark A., McNamara, James
Published in ChemInform (26.04.2005)
Published in ChemInform (26.04.2005)
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