A Mechanistic Study of the Lewis Base-Directed Cycloaddition of 2‑Pyrones and Alkynylboranes
Crépin, Damien F. P, Harrity, Joseph P. A, Jiang, Julong, Meijer, Anthony J. H. M, Nassoy, Anne-Chloé M. A, Raubo, Piotr
Published in Journal of the American Chemical Society (18.06.2014)
Published in Journal of the American Chemical Society (18.06.2014)
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Journal Article
Multiple Rhodium-Catalyzed Cleavages of Single C–C bonds
Aïssa, Christophe, Crépin, Damien, Tetlow, Daniel J, Ho, Kelvin Y. T
Published in Organic letters (15.03.2013)
Published in Organic letters (15.03.2013)
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Journal Article
Design, synthesis, and evaluation of 1-( N-benzylamino)-2-phenyl-3-(1 H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents
Giraud, Francis, Logé, Cédric, Pagniez, Fabrice, Crepin, Damien, Le Pape, Patrice, Le Borgne, Marc
Published in Bioorganic & medicinal chemistry (15.03.2008)
Published in Bioorganic & medicinal chemistry (15.03.2008)
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Journal Article
Design, Synthesis, and in vitro Antifungal Activity of 1-[(4-Substituted-benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols
Guillon, Rémi, Pagniez, Fabrice, Giraud, Francis, Crépin, Damien, Picot, Carine, Le Borgne, Marc, Morio, Florent, Duflos, Muriel, Logé, Cédric, Le Pape, Patrice
Published in ChemMedChem (02.05.2011)
Published in ChemMedChem (02.05.2011)
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Journal Article
Design, synthesis and evaluation of 3-(imidazol- 1-ylmethyl)indoles as antileishmanial agents. Part II
Giraud, Francis, Loge, Cedric, Pagniez, Fabrice, Crepin, Damien, Barres, Sophie, Picot, Carine, Le Pape, Patrice, Le Borgne, Marc
Published in Journal of enzyme inhibition and medicinal chemistry (01.10.2009)
Published in Journal of enzyme inhibition and medicinal chemistry (01.10.2009)
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Journal Article
Abstract 5692: Identification of novel CDK12 inhibitors that synergize with PARP inhibition through induction of ‘BRCAness’ phenotype
Ainscow, Edward K., Bahl, Ashwani, Thompson, Stuart, Flatt, Luke, Crepin, Damien, Stevenson, Brett
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
Abstract P051: Identification of an orally bioavailable dual Cyclin K glue degrader - CDK12/13 inhibitor
Ainscow, Edward K., Campbell, Adrian, Cripps, Michael, Workman, Robert, Thomson, Stuart, Chohan, Kam, Crepin, Damien, Sunose, Mahiro, Patient, Jamie, Kendrew, Jane, Bahl, Ash
Published in Molecular cancer therapeutics (01.12.2021)
Published in Molecular cancer therapeutics (01.12.2021)
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Journal Article
In Vitro and In Vivo Antifungal Profile of a Novel and Long-Acting Inhaled Azole, PC945, on Aspergillus fumigatus Infection
Colley, Thomas, Alanio, Alexandre, Kelly, Steven L, Sehra, Gurpreet, Kizawa, Yasuo, Warrilow, Andrew G S, Parker, Josie E, Kelly, Diane E, Kimura, Genki, Anderson-Dring, Lauren, Nakaoki, Takahiro, Sunose, Mihiro, Onions, Stuart, Crepin, Damien, Lagasse, Franz, Crittall, Matthew, Shannon, Jonathan, Cooke, Michael, Bretagne, Stéphane, King-Underwood, John, Murray, John, Ito, Kazuhiro, Strong, Pete, Rapeport, Garth
Published in Antimicrobial agents and chemotherapy (01.05.2017)
Published in Antimicrobial agents and chemotherapy (01.05.2017)
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Journal Article
In Vitro and In Vivo Efficacy of a Novel and Long-Acting Fungicidal Azole, PC1244, on Aspergillus fumigatus Infection
Colley, Thomas, Sehra, Gurpreet, Chowdhary, Anuradha, Alanio, Alexandre, Kelly, Steven L, Kizawa, Yasuo, Armstrong-James, Darius, Fisher, Matthew C, Warrilow, Andrew G S, Parker, Josie E, Kelly, Diane E, Kimura, Genki, Nishimoto, Yuki, Sunose, Mihiro, Onions, Stuart, Crepin, Damien, Lagasse, Franz, Crittall, Matthew, Shannon, Jonathan, McConville, Matthew, King-Underwood, John, Naylor, Alan, Bretagne, Stéphane, Murray, John, Ito, Kazuhiro, Strong, Pete, Rapeport, Garth
Published in Antimicrobial agents and chemotherapy (01.05.2018)
Published in Antimicrobial agents and chemotherapy (01.05.2018)
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Journal Article
Facile and chemoselective rhodium-catalysed intramolecular hydroacylation of [small alpha],[small alpha]-disubstituted 4-alkylidenecyclopropanals
Crepin, Damien, Tugny, Coralie, Murray, James H, Aissa, Christophe
Published in Chemical communications (Cambridge, England) (01.01.2011)
Published in Chemical communications (Cambridge, England) (01.01.2011)
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Journal Article
Conformationally restricted benzothienoazepine respiratory syncytial virus inhibitors: their synthesis, structural analysis and biological activitiesElectronic supplementary information (ESI) available. See DOI: 10.1039/c8md00033f
Fordyce, Euan A. F, Fraser Hunt, S, Crepin, Damien, Onions, Stuart T, Parra, Guillaume F, Sleigh, Chris J, King-Underwood, John, Finch, Harry, Murray, John
Year of Publication 20.03.2018
Year of Publication 20.03.2018
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Conformationally restricted benzothienoazepine respiratory syncytial virus inhibitors: their synthesis, structural analysis and biological activities† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8md00033f
Fordyce, Euan A. F., Fraser Hunt, S., Crepin, Damien, Onions, Stuart T., Parra, Guillaume F., Sleigh, Chris J., King-Underwood, John, Finch, Harry, Murray, John
Published in MedChemComm (20.02.2018)
Published in MedChemComm (20.02.2018)
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Journal Article
Conformationally restricted benzothienoazepine respiratory syncytial virus inhibitors: their synthesis, structural analysis and biological activities
Fordyce, Euan A. F., Hunt, S. Fraser, Crepin, Damien, Onions, Stuart T., Parra, Guillaume F., Sleigh, Chris J., King-Underwood, John, Finch, Harry, Murray, John
Published in MedChemComm (01.03.2018)
Published in MedChemComm (01.03.2018)
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