The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold
Sandoval, Elena, Lafuente-Monasterio, María José, Almela, María J, Castañeda, Pablo, Jiménez Díaz, María Belén, Martínez-Martínez, María S, Vidal, Jaume, Angulo-Barturen, Íñigo, Bamborough, Paul, Burrows, Jeremy, Cammack, Nicholas, Chaparro, María J, Coterón, José M, de Cozar, Cristina, Crespo, Benigno, Díaz, Beatriz, Drewes, Gerard, Fernández, Esther, Ferrer-Bazaga, Santiago, Fraile, María Teresa, Gamo, Francisco J, Ghidelli-Disse, Sonja, Gómez, Rubén, Haselden, John, Huss, Sophie, León, María Luisa, de Mercado, Jaime, Macdonald, Simon J. F, Martín Hernando, José Ignacio, Prats, Sara, Puente, Margarita, Rodríguez, Anne, de la Rosa, Juan C, Rueda, Lourdes, Selenski, Carolyn, Willis, Paul, Wilson, David M, Witty, Michael, Calderón, Félix
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article
Case Study of Small Molecules As Antimalarials: 2‑Amino-1-phenylethanol (APE) Derivatives
Chaparro, María J, Vidal, Jaume, Angulo-Barturen, Íñigo, Bueno, José M, Burrows, Jeremy, Cammack, Nicholas, Castañeda, Pablo, Colmenarejo, Gonzalo, Coterón, José M, de las Heras, Laura, Fernández, Esther, Ferrer, Santiago, Gabarró, Raquel, Gamo, Francisco J, García, Mercedes, Jiménez-Díaz, María B, Lafuente, María J, León, María L, Martínez, María S, Minick, Douglas, Prats, Sara, Puente, Margarita, Rueda, Lourdes, Sandoval, Elena, Santos-Villarejo, Ángel, Witty, Michael, Calderón, Félix
Published in ACS medicinal chemistry letters (12.06.2014)
Published in ACS medicinal chemistry letters (12.06.2014)
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Journal Article
Falcipain Inhibitors: Optimization Studies of the 2-Pyrimidinecarbonitrile Lead Series
Coterón, Jose M, Catterick, David, Castro, Julia, Chaparro, María J, Díaz, Beatriz, Fernández, Esther, Ferrer, Santiago, Gamo, Francisco J, Gordo, Mariola, Gut, Jiri, de las Heras, Laura, Legac, Jennifer, Marco, Maria, Miguel, Juan, Muñoz, Vicente, Porras, Esther, de la Rosa, Juan C, Ruiz, Jose R, Sandoval, Elena, Ventosa, Pilar, Rosenthal, Philip J, Fiandor, Jose M
Published in Journal of medicinal chemistry (26.08.2010)
Published in Journal of medicinal chemistry (26.08.2010)
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Journal Article
Correction to The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold
Sandoval, Elena, Lafuente-Monasterio, María José, Almela, María J., Castañeda, Pablo, Jiménez Díaz, María Belén, Martínez-Martínez, María S., Vidal, Jaume, Angulo-Barturen, Íñigo, Bamborough, Paul, Burrows, Jeremy, Cammack, Nicholas, Chaparro, María J., Coterón, José M., de Cozar, Cristina, Crespo, Benigno, Díaz, Beatriz, Drewes, Gerard, Fernández, Esther, Ferrer-Bazaga, Santiago, Fraile, María Teresa, Gamo, Francisco J., Ghidelli-Disse, Sonja, Gómez, Rubén, Haselden, John, Huss, Sophie, León, María Luisa, de Mercado, Jaime, Macdonald, Simon J. F., Martín Hernando, José Ignacio, Prats, Sara, Puente, Margarita, Rodríguez, Anne, de la Rosa, Juan C., Rueda, Lourdes, Selenski, Carolyn, Willis, Paul, Wilson, David M., Witty, Michael, Calderón, Félix
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Journal Article
Stereoselective synthesis of the antifungal GM222712
Bueno, José M, Coterón, José M, Chiara, Jose Luis, Fernández-Mayoralas, Alfonso, Fiandor, José M, Valle, Nuria
Published in Tetrahedron letters (08.06.2000)
Published in Tetrahedron letters (08.06.2000)
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Journal Article
Corrections to Falcipain Inhibitors: Optimization Studies of the 2-Pyrimidinecarbonitrile Lead Series
Coterón, Jose M, Catterick, David, Castro, Julia, Chaparro, María J, Díaz, Beatriz, Fernández, Esther, Ferrer, Santiago, Gamo, Francisco J, Gordo, Mariola, Gut, Jiri, de las Heras, Laura, Legac, Jennifer, Marco, Maria, Miguel, Juan, Muñoz, Vicente, Porras, Esther, de la Rosa, Juan C, Ruiz, Jose R, Sandoval, Elena, Ventosa, Pilar, Rosenthal, Philip J, Fiandor, Jose M
Published in Journal of medicinal chemistry (11.11.2010)
Published in Journal of medicinal chemistry (11.11.2010)
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Journal Article
Tetrahydro-2-naphthyl and 2‑Indanyl Triazolopyrimidines Targeting Plasmodium falciparum Dihydroorotate Dehydrogenase Display Potent and Selective Antimalarial Activity
Kokkonda, Sreekanth, Deng, Xiaoyi, White, Karen L, Coteron, Jose M, Marco, Maria, de las Heras, Laura, White, John, El Mazouni, Farah, Tomchick, Diana R, Manjalanagara, Krishne, Rudra, Kakali Rani, Chen, Gong, Morizzi, Julia, Ryan, Eileen, Kaminsky, Werner, Leroy, Didier, Martínez-Martínez, María Santos, Jimenez-Diaz, Maria Belen, Bazaga, Santiago Ferrer, Angulo-Barturen, Iñigo, Waterson, David, Burrows, Jeremy N, Matthews, Dave, Charman, Susan A, Phillips, Margaret A, Rathod, Pradipsinh K
Published in Journal of medicinal chemistry (09.06.2016)
Published in Journal of medicinal chemistry (09.06.2016)
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Journal Article
Glycophanes, cyclodextrin-cyclophane hybrid receptors for apolar binding in aqueous solutions. A stereoselective carbohydrate-carbohydrate interaction in water
Coteron, Jose M, Vicent, Cristina, Bosso, Claude, Penades, Soledad
Published in Journal of the American Chemical Society (01.11.1993)
Published in Journal of the American Chemical Society (01.11.1993)
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Journal Article
Structure-Guided Lead Optimization of Triazolopyrimidine-Ring Substituents Identifies Potent Plasmodium falciparum Dihydroorotate Dehydrogenase Inhibitors with Clinical Candidate Potential
Coteron, Jose M, Marco, María, Esquivias, Jorge, Deng, Xiaoyi, White, Karen L, White, John, Koltun, Maria, El Mazouni, Farah, Kokkonda, Sreekanth, Katneni, Kasiram, Bhamidipati, Ravi, Shackleford, David M, Angulo-Barturen, Iñigo, Ferrer, Santiago B, Jiménez-Díaz, María Belén, Gamo, Francisco-Javier, Goldsmith, Elizabeth J, Charman, William N, Bathurst, Ian, Floyd, David, Matthews, David, Burrows, Jeremy N, Rathod, Pradipsinh K, Charman, Susan A, Phillips, Margaret A
Published in Journal of medicinal chemistry (11.08.2011)
Published in Journal of medicinal chemistry (11.08.2011)
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Journal Article
A Replicative In Vitro Assay for Drug Discovery against Leishmania donovani
Tegazzini, Diana, Díaz, Rosario, Aguilar, Fernando, Peña, Imanol, Presa, Jesús L, Yardley, Vanessa, Martin, Julio J, Coteron, Jose M, Croft, Simon L, Cantizani, Juan
Published in Antimicrobial agents and chemotherapy (01.06.2016)
Published in Antimicrobial agents and chemotherapy (01.06.2016)
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Journal Article
Stereocontrolled glycosylation of sordaricin in the presence of ammonium salts
Coterón, José M., Chiara, José L., Fernández-Mayoralas, Alfonso, Fiandor, José M., Valle, Nuria
Published in Tetrahedron letters (08.06.2000)
Published in Tetrahedron letters (08.06.2000)
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Journal Article
Oligosaccharides Structurally Related to E-Selectin Ligands Are Inhibitors of Neural Cell Division: Synthesis, Conformational Analysis, and Biological Activity
Coteron, Jose M, Singh, Kamaljit, Asensio, Juan L, Dominguez-Dalda, Maria, Fernandez-Mayoralas, Alfonso, Jimenez-Barbero, Jesus, Martin-Lomas, Manuel, Nieto-Sampedro, Manuel
Published in Journal of organic chemistry (01.03.1995)
Published in Journal of organic chemistry (01.03.1995)
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Journal Article
The complexation of glucose and other monosaccharides with cyclodextrins
Hacket, Frank, Coteron, Jose-Miguel, Schneider, Hans-Jörg, Kazachenko, Vladimir P
Published in Canadian journal of chemistry (01.01.1997)
Published in Canadian journal of chemistry (01.01.1997)
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