A semi-synthetic neolignan derivative from dihydrodieugenol B selectively affects the bioenergetic system of Leishmania infantum and inhibits cell division
Amaral, Maiara, de Sousa, Fernanda S, Silva, Thais A Costa, Junior, Andrés Jimenez G, Taniwaki, Noemi N, Johns, Deidre M, Lago, João Henrique G, Anderson, Edward A, Tempone, Andre G
Published in Scientific reports (16.04.2019)
Published in Scientific reports (16.04.2019)
Get full text
Journal Article
Chemical Constituents from Aerial Parts of Baccharis sphenophylla and Effects against Intracellular Forms of Trypanosoma cruzi
Silva, Matheus L., Costa‐Silva, Thais A., Antar, Guilherme M., Tempone, Andre G., Lago, João Henrique G.
Published in Chemistry & biodiversity (01.10.2021)
Published in Chemistry & biodiversity (01.10.2021)
Get full text
Journal Article
Essential Oils from Different Myrtaceae Species from Brazilian Atlantic Forest Biome – Chemical Dereplication and Evaluation of Antitrypanosomal Activity
Silva Maiolini, Tatiane Cristina, Rosa, Welton, Oliveira Miranda, Daniel, Costa‐Silva, Thais A., Tempone, Andre G., Pires Bueno, Paula Carolina, Ferreira Dias, Danielle, Aparecida Chagas de Paula, Daniela, Sartorelli, Patricia, Lago, João Henrique G., Gomes Soares, Marisi
Published in Chemistry & biodiversity (01.06.2022)
Published in Chemistry & biodiversity (01.06.2022)
Get full text
Journal Article
Simplified Derivatives of Dibenzylbutyrolactone Lignans from Hydrocotyle bonariensis as Antitrypanosomal Candidates
Souza, Dalete Christine S., Costa‐Silva, Thais A., Morais, Thiago R., Brito, Juliana R., Ferreira, Edgard A., Antar, Guilherme M., Sartorelli, Patricia, Tempone, Andre G., Lago, João Henrique G.
Published in Chemistry & biodiversity (01.10.2021)
Published in Chemistry & biodiversity (01.10.2021)
Get full text
Journal Article
γ‐Lactones from Persea americana and Persea fulva – in Vitro and in Silico Evaluation of Trypanosoma cruzi Activity
Reis, Isabella Mary A., Umehara, Eric, Conceição, Rodrigo S., M. Oliveira, Larissa, Coelho dos S. Junior, Manoelito, Costa‐Silva, Thais A., Amaral, Maiara, Tempone, Andre G., Branco, Alexsandro, Lago, João Henrique G.
Published in Chemistry & biodiversity (01.09.2021)
Published in Chemistry & biodiversity (01.09.2021)
Get full text
Journal Article
Aporphine Alkaloids from Ocotea puberula with Anti‐Trypanosoma Cruzi Potential – Activity of Dicentrine‐β‐N‐Oxide in the Plasma Membrane Electric Potentials
Barbosa, Henrique, Costa‐Silva, Thais A., Alves Conserva, Geanne A., Araujo, Adelson J., Lordello, Ana Luísa L., Antar, Guilherme M., Amaral, Maiara, Soares, Marisi G., Tempone, Andre G., Lago, João Henrique G.
Published in Chemistry & biodiversity (01.04.2021)
Published in Chemistry & biodiversity (01.04.2021)
Get full text
Journal Article
Synthesis of New Dehydrodieugenol Derivatives via Olefin Cross Metathesis and In Vitro Evaluation of Their Trypanocidal Activity
Galhardo, Thalita S, Ueno, Anderson K, Carvalho, Wagner A, Costa-Silva, Thais A, Gonçalves, Marina M, Abiuzi, Mariana B, Tempone, Andre G, Lago, João Henrique G, Mandelli, Dalmo, Fischmeister, Cedric, Bruneau, Christian
Published in Catalysts (01.07.2023)
Published in Catalysts (01.07.2023)
Get full text
Journal Article
Antileishmanial activity and immunomodulatory effect of secosubamolide, a butanolide isolated from Nectandra oppositifolia (Lauraceae)
Costa-Silva, Thais A. da, Conserva, Geanne A. Alves, Galisteo Jr, Andrés J., Tempone, Andre G., Lago, João Henrique G.
Published in The journal of venomous animals and toxins including tropical diseases (2019)
Published in The journal of venomous animals and toxins including tropical diseases (2019)
Get full text
Journal Article
Enyne acetogenins from Porcelia macrocarpa displayed anti-Trypanosoma cruzi activity and cause a reduction in the intracellular calcium level
Thevenard, Fernanda, Brito, Ivanildo A, Costa-Silva, Thais A, Tempone, Andre G, Lago, João Henrique G
Published in Scientific reports (24.06.2023)
Published in Scientific reports (24.06.2023)
Get full text
Journal Article
Structure-activity relationship study of antitrypanosomal analogues of gibbilimbol B using multivariate analysis and computation-aided drug design
Leão, Luiz P.M.O., de B. Vieira, Nátalie, Oliveira, Paula P.S., Chagas-Paula, Daniela A., Soares, Marisi G., Souza, Thiago B., Baldim, João L., Costa-Silva, Thais A., Tempone, Andre G., Dias, Danielle F., Lago, João Henrique G.
Published in Bioorganic & medicinal chemistry letters (01.03.2023)
Published in Bioorganic & medicinal chemistry letters (01.03.2023)
Get full text
Journal Article
Evaluation of the effects in cellular membrane models of antitrypanosomal poly-thymolformaldehyde (PTF) using Langmuir monolayers
Parolin, Giovana A., Gonçalves, Giulia E.G., Costa-Silva, Thais A., Tempone, Andre G., Caseli, Luciano, Lago, João Henrique G., Péres, Laura O.
Published in Biochimica et biophysica acta. Biomembranes (01.02.2021)
Published in Biochimica et biophysica acta. Biomembranes (01.02.2021)
Get full text
Journal Article
Discovery of New Hits as Antitrypanosomal Agents by In Silico and In Vitro Assays Using Neolignan-Inspired Natural Products from Nectandra leucantha
Araujo, Sheila C., Sousa, Fernanda S., Costa-Silva, Thais A., Tempone, Andre G., Lago, João Henrique G., Honorio, Kathia M.
Published in Molecules (Basel, Switzerland) (06.07.2021)
Published in Molecules (Basel, Switzerland) (06.07.2021)
Get full text
Journal Article
Metabolite profile of Nectandra oppositifolia Nees & Mart. and assessment of antitrypanosomal activity of bioactive compounds through efficiency analyses
Alves Conserva, Geanne A, Quirós-Guerrero, Luis M, Costa-Silva, Thais A, Marcourt, Laurence, Pinto, Erika G, Tempone, Andre G, Fernandes, João Paulo S, Wolfender, Jean-Luc, Queiroz, Emerson F, Lago, João Henrique G
Published in PloS one (25.02.2021)
Published in PloS one (25.02.2021)
Get full text
Journal Article
Antileishmanial Effects of Acetylene Acetogenins from Seeds of Porcelia macrocarpa (Warm.) R.E. Fries (Annonaceae) and Semisynthetic Derivatives
Brito, Ivanildo A, Thevenard, Fernanda, Costa-Silva, Thais A, Oliveira, Samuel S, Cunha, Rodrigo L O R, de Oliveira, Emerson A, Sartorelli, Patricia, Guadagnin, Rafael C, Romanelli, Maiara M, Tempone, Andre G, Lago, João Henrique G
Published in Molecules (Basel, Switzerland) (28.01.2022)
Published in Molecules (Basel, Switzerland) (28.01.2022)
Get full text
Journal Article
Interaction of dicentrinone, an antitrypanosomal aporphine alkaloid isolated from Ocotea puberula (Lauraceae), in cell membrane models at the air-water interface
Barbosa, Henrique, da Silva, Rafael Leonardo C.G., Costa-Silva, Thais A., Tempone, Andre G., Antar, Guilherme M., Lago, João Henrique G., Caseli, Luciano
Published in Bioorganic chemistry (01.08.2020)
Published in Bioorganic chemistry (01.08.2020)
Get full text
Journal Article
Neolignans from leaves of Nectandra leucantha (Lauraceae) display in vitro antitrypanosomal activity via plasma membrane and mitochondrial damages
Grecco, Simone S., Costa-Silva, Thais A., Jerz, Gerold, de Sousa, Fernanda S., Londero, Vinicius S., Galuppo, Mariana K., Lima, Marta L., Neves, Bruno J., Andrade, Carolina H., Tempone, Andre G., Lago, João Henrique G.
Published in Chemico-biological interactions (01.11.2017)
Published in Chemico-biological interactions (01.11.2017)
Get full text
Journal Article
Differential lethal action of C17:2 and C17:0 anacardic acid derivatives in Trypanosoma cruzi – A mechanistic study
Umehara, Eric, Costa Silva, Thais A., Mendes, Viviane M., Guadagnin, Rafael C., Sartorelli, Patricia, Tempone, Andre G., Lago, João Henrique G.
Published in Bioorganic chemistry (01.09.2020)
Published in Bioorganic chemistry (01.09.2020)
Get full text
Journal Article
Investigation of the Anti-Leishmania (Leishmania) infantum Activity of Some Natural Sesquiterpene Lactones
Wulsten, Imke F, Costa-Silva, Thais A, Mesquita, Juliana T, Lima, Marta L, Galuppo, Mariana K, Taniwaki, Noemi N, Borborema, Samanta E T, Da Costa, Fernando B, Schmidt, Thomas J, Tempone, Andre G
Published in Molecules (Basel, Switzerland) (25.04.2017)
Published in Molecules (Basel, Switzerland) (25.04.2017)
Get full text
Journal Article
Structure-activity relationship study of antitrypanosomal chalcone derivatives using multivariate analysis
Gomes, Kaio S., da Costa-Silva, Thais A., Oliveira, Igor H., Aguilar, Andrea M., Oliveira-Silva, Diogo, Uemi, Miriam, Silva, Wender A., Melo, Lennine R., Andrade, Carlos Kleber Z., Tempone, Andre G., Baldim, João L., Lago, João Henrique G.
Published in Bioorganic & medicinal chemistry letters (15.06.2019)
Published in Bioorganic & medicinal chemistry letters (15.06.2019)
Get full text
Journal Article
IgG4 specific to Toxoplasma gondii excretory/secretory antigens in serum and/or cerebrospinal fluid support the cerebral toxoplasmosis diagnosis in HIV-infected patients
Meira, Cristina S., Vidal, José E., Costa-Silva, Thais A., Motoie, Gabriela, Gava, Ricardo, Hiramoto, Roberto M., Pereira-Chioccola, Vera L.
Published in Journal of immunological methods (30.09.2013)
Published in Journal of immunological methods (30.09.2013)
Get full text
Journal Article