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Discovery of Anticancer Agents of Diverse Natural Origin
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Preclinical Evaluation of the Novel BTK Inhibitor Acalabrutinib in Canine Models of B-Cell Non-Hodgkin Lymphoma
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Nonsteroidal Selective Androgen Receptor Modulators (SARMs): Dissociating the Anabolic and Androgenic Activities of the Androgen Receptor for Therapeutic Benefit
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Published in Journal of medicinal chemistry (25.06.2009)
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Decoupling FcRn and tumor contributions to elevated immune checkpoint inhibitor clearance in cancer cachexia
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Published in Pharmacological research (01.01.2024)
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Inhibition of androgen/AR signaling inhibits diethylnitrosamine (DEN) induced tumour initiation and remodels liver immune cell networks
Helms, Timothy H., Mullins, Riley D., Thomas-Ahner, Jennifer M., Kulp, Samuel K., Campbell, Moray J., Lucas, Fabienne, Schmidt, Nathan, LeMoine, Dana M., Getaneh, Surafel, Xie, Zhiliang, Phelps, Mitch A., Clinton, Steven K., Coss, Christopher C.
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Phyllanthusmin Derivatives Induce Apoptosis and Reduce Tumor Burden in High-Grade Serous Ovarian Cancer by Late-Stage Autophagy Inhibition
Young, Alexandria N, Herrera, Denisse, Huntsman, Andrew C, Korkmaz, Melissa A, Lantvit, Daniel D, Mazumder, Sarmistha, Kolli, Shamalatha, Coss, Christopher C, King, Salane, Wang, Hongyan, Swanson, Steven M, Kinghorn, A Douglas, Zhang, Xiaoli, Phelps, Mitch A, Aldrich, Leslie N, Fuchs, James R, Burdette, Joanna E
Published in Molecular cancer therapeutics (01.10.2018)
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The Neonatal Fc Receptor Is Elevated in Monocyte-Derived Immune Cells in Pancreatic Cancer
Thomas, Justin, Torok, Molly A, Agrawal, Kriti, Pfau, Timothy, Vu, Trang T, Lyberger, Justin, Chang, Hsiaochi, Castillo, Alyssa Marie M, Chen, Min, Remaily, Bryan, Kim, Kyeongmin, Xie, Zhiliang, Dillhoff, Mary E, Kulp, Samuel K, Behbehani, Gregory K, Cruz-Monserrate, Zobeida, Ganesan, Latha P, Owen, Dwight H, Phelps, Mitch A, Coss, Christopher C, Mace, Thomas A
Published in International journal of molecular sciences (25.06.2022)
Published in International journal of molecular sciences (25.06.2022)
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Overcoming resistance to anabolic SARM therapy in experimental cancer cachexia with an HDAC inhibitor
Liva, Sophia G, Tseng, Yu‐Chou, Dauki, Anees M, Sovic, Michael G, Vu, Trang, Henderson, Sally E, Kuo, Yi‐Chiu, Benedict, Jason A, Zhang, Xiaoli, Remaily, Bryan C, Kulp, Samuel K, Campbell, Moray, Bekaii‐Saab, Tanios, Phelps, Mitchell A, Chen, Ching‐Shih, Coss, Christopher C
Published in EMBO molecular medicine (07.02.2020)
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Activity of Estrogen Receptor β Agonists in Therapy-Resistant Estrogen Receptor-Positive Breast Cancer
Datta, Jharna, Willingham, Natalie, Manouchehri, Jasmine M, Schnell, Patrick, Sheth, Mirisha, David, Joel J, Kassem, Mahmoud, Wilson, Tyler A, Radomska, Hanna S, Coss, Christopher C, Bennett, Chad E, Ganju, Ramesh K, Sardesai, Sagar D, Lustberg, Maryam, Ramaswamy, Bhuvaneswari, Stover, Daniel G, Cherian, Mathew A
Published in Frontiers in oncology (25.04.2022)
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Narayanan, Ramesh, Coss, Christopher C., Dalton, James T.
Published in Molecular and cellular endocrinology (15.04.2018)
Published in Molecular and cellular endocrinology (15.04.2018)
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Target specificity, in vivo pharmacokinetics, and efficacy of the putative STAT3 inhibitor LY5 in osteosarcoma, Ewing's sarcoma, and rhabdomyosarcoma
Yu, Peter Y, Gardner, Heather L, Roberts, Ryan, Cam, Hakan, Hariharan, Seethalakshmi, Ren, Ling, LeBlanc, Amy K, Xiao, Hui, Lin, Jiayuh, Guttridge, Denis C, Mo, Xiaokui, Bennett, Chad E, Coss, Christopher C, Ling, Yonghua, Phelps, Mitch A, Houghton, Peter, London, Cheryl A
Published in PloS one (27.07.2017)
Published in PloS one (27.07.2017)
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Selective Androgen Receptor Modulator Treatment Improves Muscle Strength and Body Composition and Prevents Bone Loss in Orchidectomized Rats
Gao, Wenqing, Reiser, Peter J, Coss, Christopher C, Phelps, Mitch A, Kearbey, Jeffrey D, Miller, Duane D, Dalton, James T
Published in Endocrinology (Philadelphia) (01.11.2005)
Published in Endocrinology (Philadelphia) (01.11.2005)
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Discovery and preclinical characterization of novel small molecule TRK and ROS1 tyrosine kinase inhibitors for the treatment of cancer and inflammation
Narayanan, Ramesh, Yepuru, Muralimohan, Coss, Christopher C, Wu, Zhongzhi, Bauler, Matthew N, Barrett, Christina M, Mohler, Michael L, Wang, Yun, Kim, Juhyun, Snyder, Linda M, He, Yali, Levy, Nelson, Miller, Duane D, Dalton, James T
Published in PloS one (26.12.2013)
Published in PloS one (26.12.2013)
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Role and pharmacologic significance of cytochrome P‐450 2D6 in oxidative metabolism of toremifene and tamoxifen
Kim, Juhyun, Coss, Christopher C., Barrett, Christina M., Mohler, Michael L., Bohl, Casey E., Li, Chien‐Ming, He, Yali, Veverka, Karen A., Dalton, James T.
Published in International journal of cancer (15.03.2013)
Published in International journal of cancer (15.03.2013)
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Murine cancer cachexia models replicate elevated catabolic pembrolizumab clearance in humans
Castillo, Alyssa Marie M., Vu, Trang T., Liva, Sophia G., Chen, Min, Xie, Zhiliang, Thomas, Justin, Remaily, Bryan, Guo, Yizhen, Subrayan, Uma L., Costa, Travis, Helms, Timothy H., Irby, Donald J., Kim, Kyeongmin, Owen, Dwight H., Kulp, Samuel K., Mace, Thomas A., Phelps, Mitch A., Coss, Christopher C.
Published in JCSM rapid communications (01.07.2021)
Published in JCSM rapid communications (01.07.2021)
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Cachectic Cancer Patients: Immune to Checkpoint Inhibitor Therapy?
Coss, Christopher C, Clinton, Steven K, Phelps, Mitch A
Published in Clinical cancer research (01.12.2018)
Published in Clinical cancer research (01.12.2018)
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