Discovery of PF-06873600, a CDK2/4/6 Inhibitor for the Treatment of Cancer
Freeman-Cook, Kevin D, Hoffman, Robert L, Behenna, Douglas C, Boras, Britton, Carelli, Jordan, Diehl, Wade, Ferre, Rose Ann, He, You-Ai, Hui, Andrea, Huang, Buwen, Huser, Nanni, Jones, Rhys, Kephart, Susan E, Lapek, John, McTigue, Michele, Miller, Nichol, Murray, Brion W, Nagata, Asako, Nguyen, Lisa, Niessen, Sherry, Ninkovic, Sacha, O’Doherty, Inish, Ornelas, Martha A, Solowiej, James, Sutton, Scott C, Tran, Khanh, Tseng, Elaine, Visswanathan, Ravi, Xu, Meirong, Zehnder, Luke, Zhang, Qin, Zhang, Cathy, Dann, Stephen
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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Journal Article
Lipophilic efficiency: the most important efficiency metric in medicinal chemistry
Freeman-Cook, Kevin D, Hoffman, Robert L, Johnson, Ted W
Published in Future medicinal chemistry (01.02.2013)
Published in Future medicinal chemistry (01.02.2013)
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Journal Article
Development of catchment water quality models within a realtime status and forecast system for the Great Barrier Reef
Khan, Urooj, Cook, Freeman J., Laugesen, Richard, Hasan, Mohammad M., Plastow, Kevin, Amirthanathan, Gnanathikkam E., Bari, Mohammed A., Tuteja, Narendra K.
Published in Environmental modelling & software : with environment data news (01.10.2020)
Published in Environmental modelling & software : with environment data news (01.10.2020)
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Journal Article
Groundwater recharge from overbank floods
Doble, Rebecca C., Crosbie, Russell S., Smerdon, Brian D., Peeters, Luk, Cook, Freeman J.
Published in Water resources research (01.09.2012)
Published in Water resources research (01.09.2012)
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Journal Article
Design of Selective, ATP-Competitive Inhibitors of Akt
Freeman-Cook, Kevin D, Autry, Christopher, Borzillo, Gary, Gordon, Deborah, Barbacci-Tobin, Elsa, Bernardo, Vincent, Briere, David, Clark, Tracey, Corbett, Matthew, Jakubczak, John, Kakar, Shefali, Knauth, Elizabeth, Lippa, Blaise, Luzzio, Michael J, Mansour, Mahmoud, Martinelli, Gary, Marx, Matthew, Nelson, Kendra, Pandit, Jayvardhan, Rajamohan, Francis, Robinson, Shaughnessy, Subramanyam, Chakrapani, Wei, Liuqing, Wythes, Martin, Morris, Joel
Published in Journal of medicinal chemistry (24.06.2010)
Published in Journal of medicinal chemistry (24.06.2010)
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Journal Article
Justice for Incarcerated Moms Act of 2021: Reflections and recommendations
Shlafer, Rebecca J, Gerrity, Erica, Norris, Chauntel, Freeman-Cook, Rachel, B Sufrin, Carolyn
Published in Women's Health (01.04.2022)
Published in Women's Health (01.04.2022)
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Book Review
Journal Article
Analysis of soil wetting and solute transport in subsurface trickle irrigation
Cote, Claire M., Bristow, Keith L., Charlesworth, Philip B., Cook, Freeman J., Thorburn, Peter J.
Published in Irrigation science (01.11.2003)
Published in Irrigation science (01.11.2003)
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Journal Article
Discovery of small molecule isozyme non-specific inhibitors of mammalian acetyl-CoA carboxylase 1 and 2
Corbett, Jeffrey W., Freeman-Cook, Kevin D., Elliott, Richard, Vajdos, Felix, Rajamohan, Francis, Kohls, Darcy, Marr, Eric, Zhang, Hailong, Tong, Liang, Tu, Meihua, Murdande, Sharad, Doran, Shawn D., Houser, Janet A., Song, Wei, Jones, Christopher J., Coffey, Steven B., Buzon, Leanne, Minich, Martha L., Dirico, Kenneth J., Tapley, Susan, Kirk McPherson, R., Sugarman, Eliot, James Harwood, H., Esler, William
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
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Journal Article
Conserved Locus-Specific Silencing Functions of Schizosaccharomyces pombe sir2
Freeman-Cook, Lisa L, Gomez, Eliana B, Spedale, Erik J, Marlett, John, Forsburg, Susan L, Pillus, Lorraine, Laurenson, Patricia
Published in Genetics (Austin) (01.03.2005)
Published in Genetics (Austin) (01.03.2005)
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Journal Article
Maximizing Lipophilic Efficiency: The Use of Free-Wilson Analysis in the Design of Inhibitors of Acetyl-CoA Carboxylase
Freeman-Cook, Kevin D, Amor, Paul, Bader, Scott, Buzon, Leanne M, Coffey, Steven B, Corbett, Jeffrey W, Dirico, Kenneth J, Doran, Shawn D, Elliott, Richard L, Esler, William, Guzman-Perez, Angel, Henegar, Kevin E, Houser, Janet A, Jones, Christopher S, Limberakis, Chris, Loomis, Katherine, McPherson, Kirk, Murdande, Sharad, Nelson, Kendra L, Phillion, Dennis, Pierce, Betsy S, Song, Wei, Sugarman, Eliot, Tapley, Susan, Tu, Meihua, Zhao, Zhengrong
Published in Journal of medicinal chemistry (26.01.2012)
Published in Journal of medicinal chemistry (26.01.2012)
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Journal Article
Selection and Characterization of Small Random Transmembrane Proteins that Bind and Activate the Platelet-derived Growth Factor β Receptor
Freeman-Cook, Lisa L., Dixon, Ann M., Frank, Jennifer B., Xia, Yu, Ely, Lara, Gerstein, Mark, Engelman, Donald M., DiMaio, Daniel
Published in Journal of molecular biology (14.05.2004)
Published in Journal of molecular biology (14.05.2004)
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Journal Article
Packing contacts can mediate highly specific interactions between artificial transmembrane proteins and the PDGFβ receptor
Ptacek, Jennifer B, Edwards, Anne P.B, Freeman-Cook, Lisa L, DiMaio, Daniel
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2007)
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2007)
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Journal Article
Identification of Tetrahydropyrido[4,3‑d]pyrimidine Amides as a New Class of Orally Bioavailable TGR5 Agonists
Piotrowski, David W, Futatsugi, Kentaro, Warmus, Joseph S, Orr, Suvi T. M, Freeman-Cook, Kevin D, Londregan, Allyn T, Wei, Liuqing, Jennings, Sandra M, Herr, Michael, Coffey, Steven B, Jiao, Wenhua, Storer, Gregory, Hepworth, David, Wang, Jian, Lavergne, Sophie Y, Chin, Janice E, Hadcock, John R, Brenner, Martin B, Wolford, Angela C, Janssen, Ann M, Roush, Nicole S, Buxton, Joanne, Hinchey, Terri, Kalgutkar, Amit S, Sharma, Raman, Flynn, Declan A
Published in ACS medicinal chemistry letters (10.01.2013)
Published in ACS medicinal chemistry letters (10.01.2013)
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Journal Article
Designing glucokinase activators with reduced hypoglycemia risk: discovery of N,N-dimethyl-5-(2-methyl-6-((5-methylpyrazin-2-yl)-carbamoyl)benzofuran-4-yloxy)pyrimidine-2-carboxamide as a clinical candidate for the treatment of type 2 diabetes mellitus
Pfefferkorn, Jeffrey A., Guzman-Perez, Angel, Oates, Peter J., Litchfield, John, Aspnes, Gary, Basak, Arindrajit, Benbow, John, Berliner, Martin A., Bian, Jianwei, Choi, Chulho, Freeman-Cook, Kevin, Corbett, Jeffrey W., Didiuk, Mary, Dunetz, Joshua R., Filipski, Kevin J., Hungerford, William M., Jones, Christopher S., Karki, Kapil, Ling, Anthony, Li, Jian-Cheng, Patel, Leena, Perreault, Christian, Risley, Hud, Saenz, James, Song, Wei, Tu, Meihua, Aiello, Robert, Atkinson, Karen, Barucci, Nicole, Beebe, David, Bourassa, Patricia, Bourbounais, Francis, Brodeur, Anne M., Burbey, Rena, Chen, Jing, D'Aquila, Theresa, Derksen, David R., Haddish-Berhane, Nahor, Huang, Cong, Landro, James, Lee Lapworth, Amanda, MacDougall, Margit, Perregaux, David, Pettersen, John, Robertson, Alan, Tan, Beijing, Treadway, Judith L., Liu, Shenping, Qiu, Xiayang, Knafels, John, Ammirati, Mark, Song, Xi, DaSilva-Jardine, Paul, Liras, Spiros, Sweet, Laurel, Rolph, Timothy P.
Published in MedChemComm (01.09.2011)
Published in MedChemComm (01.09.2011)
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Journal Article
Packing contacts can mediate highly specific interactions between artificial transmembrane proteins and the PDGFb receptor
Ptacek, Jennifer B, Edwards, Anne PB, Freeman-Cook, Lisa L, DiMaio, Daniel
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2007)
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2007)
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Journal Article