Chemically induced degradation of CDK9 by a proteolysis targeting chimera (PROTAC)
Robb, Caroline M., Contreras, Jacob I., Kour, Smit, Taylor, Margaret A., Abid, Mohammad, Sonawane, Yogesh A., Zahid, Muhammad, Murry, Daryl J., Natarajan, Amarnath, Rana, Sandeep
Published in Chemical communications (Cambridge, England) (04.07.2017)
Published in Chemical communications (Cambridge, England) (04.07.2017)
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Journal Article
Cyclin Dependent Kinase 9 Inhibitors for Cancer Therapy
Sonawane, Yogesh A, Taylor, Margaret A, Napoleon, John Victor, Rana, Sandeep, Contreras, Jacob I, Natarajan, Amarnath
Published in Journal of medicinal chemistry (13.10.2016)
Published in Journal of medicinal chemistry (13.10.2016)
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Journal Article
Isatin Derived Spirocyclic Analogues with α‑Methylene-γ-butyrolactone as Anticancer Agents: A Structure–Activity Relationship Study
Rana, Sandeep, Blowers, Elizabeth C, Tebbe, Calvin, Contreras, Jacob I, Radhakrishnan, Prakash, Kizhake, Smitha, Zhou, Tian, Rajule, Rajkumar N, Arnst, Jamie L, Munkarah, Adnan R, Rattan, Ramandeep, Natarajan, Amarnath
Published in Journal of medicinal chemistry (26.05.2016)
Published in Journal of medicinal chemistry (26.05.2016)
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Journal Article
CDK5 Inhibitor Downregulates Mcl-1 and Sensitizes Pancreatic Cancer Cell Lines to Navitoclax
Kour, Smit, Rana, Sandeep, Contreras, Jacob I, King, Hannah M, Robb, Caroline M, Sonawane, Yogesh A, Bendjennat, Mourad, Crawford, Ayrianne J, Barger, Carter J, Kizhake, Smitha, Luo, Xu, Hollingsworth, Michael A, Natarajan, Amarnath
Published in Molecular pharmacology (01.10.2019)
Published in Molecular pharmacology (01.10.2019)
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Journal Article
Structure activity relationship (SAR) study identifies a quinoxaline urea analog that modulates IKKβ phosphorylation for pancreatic cancer therapy
Sagar, Satish, Singh, Sarbjit, Mallareddy, Jayapal Reddy, Sonawane, Yogesh A., Napoleon, John V., Rana, Sandeep, Contreras, Jacob I., Rajesh, Christabelle, Ezell, Edward L., Kizhake, Smitha, Garrison, Jered C., Radhakrishnan, Prakash, Natarajan, Amarnath
Published in European journal of medicinal chemistry (15.10.2021)
Published in European journal of medicinal chemistry (15.10.2021)
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Journal Article
Symbiotic prodrugs (SymProDs) dual targeting of NFkappaB and CDK
Rana, Sandeep, Kour, Smit, Sonawane, Yogesh A., Robb, Caroline M., Contreras, Jacob I., Kizhake, Smitha, Zahid, Muhammad, Karpf, Adam R., Natarajan, Amarnath
Published in Chemical biology & drug design (01.08.2020)
Published in Chemical biology & drug design (01.08.2020)
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Journal Article
Development of 1‑((1,4-trans)‑4-Aryloxycyclohexyl)-3-arylurea Activators of Heme-Regulated Inhibitor as Selective Activators of the Eukaryotic Initiation Factor 2 Alpha (eIF2α) Phosphorylation Arm of the Integrated Endoplasmic Reticulum Stress Response
Yefidoff-Freedman, Revital, Fan, Jing, Yan, Lu, Zhang, Qingwen, dos Santos, Guillermo Rodrigo Reis, Rana, Sandeep, Contreras, Jacob I, Sahoo, Rupam, Wan, Debin, Young, Jun, Dias Teixeira, Karina Luiza, Morisseau, Christophe, Halperin, Jose, Hammock, Bruce, Natarajan, Amarnath, Wang, Peimin, Chorev, Michael, Aktas, Bertal H
Published in Journal of medicinal chemistry (13.07.2017)
Published in Journal of medicinal chemistry (13.07.2017)
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Journal Article
Characterization of CDK(5) inhibitor, 20-223 (aka CP668863) for colorectal cancer therapy
Robb, Caroline M, Kour, Smit, Contreras, Jacob I, Agarwal, Ekta, Barger, Carter J, Rana, Sandeep, Sonawane, Yogesh, Neilsen, Beth K, Taylor, Margaret, Kizhake, Smitha, Thakare, Rhishikesh N, Chowdhury, Sanjib, Wang, Jing, Black, Jennifer D, Hollingsworth, Michael A, Brattain, Michael G, Natarajan, Amarnath
Published in Oncotarget (12.01.2018)
Published in Oncotarget (12.01.2018)
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Journal Article
Discovery and characterization of small molecule Rac1 inhibitors
Arnst, Jamie L, Hein, Ashley L, Taylor, Margaret A, Palermo, Nick Y, Contreras, Jacob I, Sonawane, Yogesh A, Wahl, Andrew O, Ouellette, Michel M, Natarajan, Amarnath, Yan, Ying
Published in Oncotarget (23.05.2017)
Published in Oncotarget (23.05.2017)
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Journal Article
Chemical Genetic Screens Identify Kinase Inhibitor Combinations that Target Anti-Apoptotic Proteins for Cancer Therapy
Contreras, Jacob I, Robb, Caroline M, King, Hannah M, Baxter, Jared, Crawford, Ayrianne J, Kour, Smit, Kizhake, Smitha, Sonawane, Yogesh A, Rana, Sandeep, Hollingsworth, Michael A, Luo, Xu, Natarajan, Amarnath
Published in ACS chemical biology (18.05.2018)
Published in ACS chemical biology (18.05.2018)
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Journal Article
Developing Polyamine‐Based Peptide Amphiphiles with Tunable Morphology and Physicochemical Properties
Samad, Mehdi Bin, Chhonker, Yashpal Singh, Contreras, Jacob I., McCarthy, Alec, McClanahan, Megan M., Murry, Daryl J., Conda‐Sheridan, Martin
Published in Macromolecular bioscience (01.08.2017)
Published in Macromolecular bioscience (01.08.2017)
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Journal Article
Correction: Characterization of CDK(5) inhibitor, 20-223 (aka CP668863) for colorectal cancer therapy
Robb, Caroline M, Kour, Smit, Contreras, Jacob I, Agarwal, Ekta, Barger, Carter J, Rana, Sandeep, Sonawane, Yogesh, Neilsen, Beth K, Taylor, Margaret, Kizhake, Smitha, Thakare, Rhishikesh N, Chowdhury, Sanjib, Wang, Jing, Black, Jennifer D, Hollingsworth, Michael A, Brattain, Michael G, Natarajan, Amarnath
Published in Oncotarget (23.06.2020)
Published in Oncotarget (23.06.2020)
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Journal Article
Chemically induced degradation of CDK9 by a proteolysis targeting chimera (PROTAC)Electronic supplementary information (ESI) available. See DOI: 10.1039/c7cc03879h
Robb, Caroline M, Contreras, Jacob I, Kour, Smit, Taylor, Margaret A, Abid, Mohammad, Sonawane, Yogesh A, Zahid, Muhammad, Murry, Daryl J, Natarajan, Amarnath, Rana, Sandeep
Year of Publication 04.07.2017
Year of Publication 04.07.2017
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Journal Article